BR0116129A - Processo para a preparação de composto de diaril-4-aminopiperidinil-1substituìdo, e, composto - Google Patents

Processo para a preparação de composto de diaril-4-aminopiperidinil-1substituìdo, e, composto

Info

Publication number
BR0116129A
BR0116129A BR0116129-6A BR0116129A BR0116129A BR 0116129 A BR0116129 A BR 0116129A BR 0116129 A BR0116129 A BR 0116129A BR 0116129 A BR0116129 A BR 0116129A
Authority
BR
Brazil
Prior art keywords
compound
aminopiperidinyl
preparation
substituted diaryl
substituted
Prior art date
Application number
BR0116129-6A
Other languages
English (en)
Inventor
Andrew Griffin
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/SE2000/002560 external-priority patent/WO2001046263A1/en
Priority claimed from SE0101764A external-priority patent/SE0101764D0/xx
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BR0116129A publication Critical patent/BR0116129A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE COMPOSTO DE DIARIL-4-AMINOPIPERIDINIL-1-SUBSTITUìDO, E, COMPOSTO". A presente invenção descreve um novo e aperfeiçoado processo para a preparação de compostos de diaril-4-amino-piperidinil 1-substituído, por uma dupla arilação de um só pote, seguido pela(s) etapa(s) de desproteção opcional(ais).
BR0116129-6A 2000-12-15 2001-12-13 Processo para a preparação de composto de diaril-4-aminopiperidinil-1substituìdo, e, composto BR0116129A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
PCT/SE2000/002560 WO2001046263A1 (en) 1999-12-20 2000-12-15 Novel compounds
SE0101764A SE0101764D0 (sv) 2001-05-18 2001-05-18 New process
PCT/SE2001/002780 WO2002048108A1 (en) 2000-12-15 2001-12-13 New process for the preparation diaryl-4-amino-piperidinyl compounds

Publications (1)

Publication Number Publication Date
BR0116129A true BR0116129A (pt) 2003-11-04

Family

ID=26655171

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0116129-6A BR0116129A (pt) 2000-12-15 2001-12-13 Processo para a preparação de composto de diaril-4-aminopiperidinil-1substituìdo, e, composto

Country Status (11)

Country Link
US (1) US6835840B2 (pt)
EP (1) EP1343762A1 (pt)
JP (1) JP2004515539A (pt)
CN (1) CN1258529C (pt)
AU (2) AU2002222879B2 (pt)
BR (1) BR0116129A (pt)
CA (1) CA2436263A1 (pt)
IL (1) IL155995A0 (pt)
MX (1) MXPA03005165A (pt)
NZ (1) NZ525982A (pt)
WO (1) WO2002048108A1 (pt)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE623427A (pt) * 1961-10-10
JP2567621B2 (ja) * 1986-08-22 1996-12-25 塩野義製薬株式会社 フエノ−ル類またはフエニルアミン類のオルトシアノ化法
SE9604786D0 (sv) * 1996-12-20 1996-12-20 Astra Pharma Inc New compounds
DK1049676T3 (da) * 1997-12-24 2006-01-16 Ortho Mcneil Pharm Inc 4-[Aryl(piperidin-4-yl)]aminobenzamider, som binder til delta-opioidreceptoren
US6436959B1 (en) * 1998-12-23 2002-08-20 Ortho-Mcneil Pharmaceutical, Inc. 4-[aryl(piperidin-4-yl)]aminobenzamides

Also Published As

Publication number Publication date
NZ525982A (en) 2005-09-30
AU2287902A (en) 2002-06-24
MXPA03005165A (es) 2003-09-22
JP2004515539A (ja) 2004-05-27
WO2002048108A9 (en) 2004-04-15
IL155995A0 (en) 2003-12-23
US6835840B2 (en) 2004-12-28
US20040068112A1 (en) 2004-04-08
WO2002048108B1 (en) 2002-10-10
CN1481362A (zh) 2004-03-10
AU2002222879B2 (en) 2006-02-02
CA2436263A1 (en) 2002-06-20
EP1343762A1 (en) 2003-09-17
WO2002048108A1 (en) 2002-06-20
CN1258529C (zh) 2006-06-07

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: CONFORME ARTIGO 10O DA RESOLUCAO 124/06, CABE SER ARQUIVADO REFERENTE AO NAO RECOLHIMENTO DA 8A, 9AE 10A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2144 DE 07/02/2012.