BR0114734A - 3,4-dihidropirido [1, 2-a] pirimidinas substituìdas - Google Patents
3,4-dihidropirido [1, 2-a] pirimidinas substituìdasInfo
- Publication number
- BR0114734A BR0114734A BR0114734-0A BR0114734A BR0114734A BR 0114734 A BR0114734 A BR 0114734A BR 0114734 A BR0114734 A BR 0114734A BR 0114734 A BR0114734 A BR 0114734A
- Authority
- BR
- Brazil
- Prior art keywords
- substituted pyrimidines
- compounds
- dihydropyrido
- pharmaceutical preparations
- dihydropyride
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
"3,4-DIHIDROPIRIDO[1,2-a] PIRIMIDINAS SUBSTITUìDAS". Da estrutura geral I a processos para sua produção, a bibliotecas de substâncias contendo as mesmas, a preparados farmacêuticos contendo esses compostos, ao uso desses compostos para a produção de preparados farmacêuticos para o tratamento de dor, incontinência urinária, prurido, tinido e/ou diarréia e a composições farmacêuticas contendo esses compostos.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10050662A DE10050662A1 (de) | 2000-10-13 | 2000-10-13 | Substituierte 3,4-Dihydro-pyrido[1,2-a]pyrimidine |
| PCT/EP2001/011700 WO2002030933A1 (de) | 2000-10-13 | 2001-10-10 | Substituierte 3,4-dihydro-pyrido[1,2-a]pyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0114734A true BR0114734A (pt) | 2003-07-01 |
Family
ID=7659597
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0114734-0A BR0114734A (pt) | 2000-10-13 | 2001-10-10 | 3,4-dihidropirido [1, 2-a] pirimidinas substituìdas |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US7230103B2 (pt) |
| EP (1) | EP1326866B1 (pt) |
| JP (1) | JP4315678B2 (pt) |
| KR (1) | KR20030036924A (pt) |
| CN (1) | CN1255407C (pt) |
| AR (1) | AR034266A1 (pt) |
| AT (1) | ATE297927T1 (pt) |
| AU (2) | AU2002210526B2 (pt) |
| BR (1) | BR0114734A (pt) |
| CA (1) | CA2425666A1 (pt) |
| CO (1) | CO5640115A2 (pt) |
| DE (2) | DE10050662A1 (pt) |
| EC (1) | ECSP034553A (pt) |
| ES (1) | ES2241882T3 (pt) |
| HK (1) | HK1057551A1 (pt) |
| HU (1) | HUP0302464A2 (pt) |
| IL (2) | IL155380A0 (pt) |
| MX (1) | MXPA03003198A (pt) |
| NO (1) | NO20031412L (pt) |
| NZ (1) | NZ525652A (pt) |
| PE (1) | PE20020435A1 (pt) |
| PL (1) | PL361915A1 (pt) |
| PT (1) | PT1326866E (pt) |
| RU (1) | RU2003113966A (pt) |
| SK (1) | SK4142003A3 (pt) |
| WO (1) | WO2002030933A1 (pt) |
| ZA (1) | ZA200303640B (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10310106A1 (de) | 2003-03-06 | 2004-09-16 | Grünenthal GmbH | Substituierte Pyridot [1,2-a]pyrimidin-Verbindungen |
| US20070155738A1 (en) | 2005-05-20 | 2007-07-05 | Alantos Pharmaceuticals, Inc. | Heterobicyclic metalloprotease inhibitors |
| CA2747750A1 (en) * | 2008-12-22 | 2010-07-01 | Theodros Asberom | Gamma secretase modulators |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU178910B (en) * | 1977-08-19 | 1982-07-28 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines |
| US4666912A (en) * | 1984-11-12 | 1987-05-19 | Chinoin Gyogyszer Es Vegyeszeti Termeker Gyara Rt | Treating process |
-
2000
- 2000-10-13 DE DE10050662A patent/DE10050662A1/de not_active Withdrawn
-
2001
- 2001-10-09 AR ARP010104731A patent/AR034266A1/es unknown
- 2001-10-10 BR BR0114734-0A patent/BR0114734A/pt not_active Application Discontinuation
- 2001-10-10 JP JP2002534319A patent/JP4315678B2/ja not_active Expired - Fee Related
- 2001-10-10 AT AT01978402T patent/ATE297927T1/de active
- 2001-10-10 DE DE50106542T patent/DE50106542D1/de not_active Expired - Lifetime
- 2001-10-10 EP EP01978402A patent/EP1326866B1/de not_active Expired - Lifetime
- 2001-10-10 SK SK414-2003A patent/SK4142003A3/sk not_active Application Discontinuation
- 2001-10-10 AU AU2002210526A patent/AU2002210526B2/en not_active Ceased
- 2001-10-10 WO PCT/EP2001/011700 patent/WO2002030933A1/de active IP Right Grant
- 2001-10-10 IL IL15538001A patent/IL155380A0/xx active IP Right Grant
- 2001-10-10 NZ NZ525652A patent/NZ525652A/en unknown
- 2001-10-10 RU RU2003113966/04A patent/RU2003113966A/ru not_active Application Discontinuation
- 2001-10-10 ES ES01978402T patent/ES2241882T3/es not_active Expired - Lifetime
- 2001-10-10 CA CA002425666A patent/CA2425666A1/en not_active Abandoned
- 2001-10-10 AU AU1052602A patent/AU1052602A/xx active Pending
- 2001-10-10 PL PL01361915A patent/PL361915A1/xx not_active Application Discontinuation
- 2001-10-10 CN CNB018205011A patent/CN1255407C/zh not_active Expired - Fee Related
- 2001-10-10 HU HU0302464A patent/HUP0302464A2/hu unknown
- 2001-10-10 MX MXPA03003198A patent/MXPA03003198A/es active IP Right Grant
- 2001-10-10 KR KR10-2003-7005162A patent/KR20030036924A/ko not_active Application Discontinuation
- 2001-10-10 PT PT01978402T patent/PT1326866E/pt unknown
- 2001-10-12 PE PE2001001014A patent/PE20020435A1/es not_active Application Discontinuation
-
2003
- 2003-03-27 NO NO20031412A patent/NO20031412L/no not_active Application Discontinuation
- 2003-04-10 IL IL155380A patent/IL155380A/en not_active IP Right Cessation
- 2003-04-11 CO CO03031095A patent/CO5640115A2/es not_active Application Discontinuation
- 2003-04-11 EC EC2003004553A patent/ECSP034553A/es unknown
- 2003-04-11 US US10/411,390 patent/US7230103B2/en not_active Expired - Fee Related
- 2003-05-12 ZA ZA200303640A patent/ZA200303640B/en unknown
-
2004
- 2004-01-15 HK HK04100342A patent/HK1057551A1/xx not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |