BR0104358A - Formulações de taxana tendo solubilidade aperfeiçoada - Google Patents
Formulações de taxana tendo solubilidade aperfeiçoadaInfo
- Publication number
- BR0104358A BR0104358A BR0104358-7A BR0104358A BR0104358A BR 0104358 A BR0104358 A BR 0104358A BR 0104358 A BR0104358 A BR 0104358A BR 0104358 A BR0104358 A BR 0104358A
- Authority
- BR
- Brazil
- Prior art keywords
- improved solubility
- formulations
- taxane
- taxane formulations
- clitaxel
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Patente de Invenção: "FORMULAçõES DE TAXANA TENDO SOLUBILIDADE APERFEIçOADA". A presente invenção refere-se a várias formulações de taxanas tendo solubilidade aperfeiçoada se comparada com clitaxel, particularmente formulações de tais derivados de taxana para administração oral ou parenteral a um paciente.
Applications Claiming Priority (9)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17967400P | 2000-02-02 | 2000-02-02 | |
US17967000P | 2000-02-02 | 2000-02-02 | |
US17978200P | 2000-02-02 | 2000-02-02 | |
US17966900P | 2000-02-02 | 2000-02-02 | |
US17967200P | 2000-02-02 | 2000-02-02 | |
US17967100P | 2000-02-02 | 2000-02-02 | |
US17979300P | 2000-02-02 | 2000-02-02 | |
US17968400P | 2000-02-02 | 2000-02-02 | |
PCT/US2001/003624 WO2001057013A1 (en) | 2000-02-02 | 2001-02-02 | Taxane formulations having improved solubility |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0104358A true BR0104358A (pt) | 2002-01-02 |
Family
ID=27575082
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0104358-7A BR0104358A (pt) | 2000-02-02 | 2001-02-02 | Formulações de taxana tendo solubilidade aperfeiçoada |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP1175414A1 (pt) |
KR (1) | KR20010111580A (pt) |
AU (1) | AU3481001A (pt) |
BR (1) | BR0104358A (pt) |
HU (1) | HUP0200995A3 (pt) |
IL (1) | IL145635A0 (pt) |
NO (1) | NO20014752L (pt) |
NZ (1) | NZ514073A (pt) |
WO (1) | WO2001057013A1 (pt) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6649632B2 (en) | 2000-02-02 | 2003-11-18 | Fsu Research Foundation, Inc. | C10 ester substituted taxanes |
KR20010112395A (ko) | 2000-02-02 | 2001-12-20 | 플로리다 스테이트 유니버시티 리서치 파운데이션, 인크 | 항종양제로서의 c7 카르보네이트 치환된 탁산 |
BR0104350A (pt) | 2000-02-02 | 2002-01-02 | Univ Florida State Res Found | Taxanos de c10 acetato heterossubstituìdo como agentes antitumor |
EP1200424B1 (en) | 2000-02-02 | 2008-11-05 | Florida State University Research Foundation, Inc. | C7 heterosubstituted acetate taxanes as antitumor agents |
AR030188A1 (es) | 2000-02-02 | 2003-08-13 | Univ Florida State Res Found | Compuestos de taxano sustituidos con esteres en el c7; composiciones farmaceuticas que los contienen y proceso para tratar un sujeto mamifero que sufre de una condicion que responde a los taxanos |
US6596737B2 (en) | 2000-02-02 | 2003-07-22 | Fsu Research Foundation, Inc. | C10 carbamoyloxy substituted taxanes |
PL350028A1 (en) | 2000-02-02 | 2002-10-21 | Univ Florida State Res Found | C10 carbonate substituted taxanes as antitumor agents |
CA2354486A1 (en) * | 2001-07-31 | 2003-01-31 | Florida State University Research Foundation, Inc. | C7 ester substituted taxanes |
CA2354478A1 (en) * | 2001-07-31 | 2003-01-31 | Florida State University Research Foundation, Inc. | C10 carbonate substituted taxanes |
CN100522955C (zh) | 2002-08-02 | 2009-08-05 | 伊缪诺金公司 | 含有新型强效紫杉烷的细胞毒性剂及其治疗用途 |
US7390898B2 (en) | 2002-08-02 | 2008-06-24 | Immunogen Inc. | Cytotoxic agents containing novel potent taxanes and their therapeutic use |
PE20050693A1 (es) | 2004-02-13 | 2005-09-27 | Univ Florida State Res Found | Taxanos sustituidos con esteres de ciclopentilo en c10 |
JP2007527432A (ja) | 2004-03-05 | 2007-09-27 | フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド | C7ラクチルオキシ置換タキサン |
JP2011517455A (ja) * | 2008-03-31 | 2011-06-09 | フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド | C(10)エチルエステルおよびc(10)シクロプロピルエステル置換タキサン |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5243045A (en) * | 1991-09-23 | 1993-09-07 | Florida State University | Certain alkoxy substituted taxanes and pharmaceutical compositions containing them |
US5250683A (en) * | 1991-09-23 | 1993-10-05 | Florida State University | Certain substituted taxanes and pharmaceutical compositions containing them |
IL107950A (en) * | 1992-12-15 | 2001-04-30 | Upjohn Co | b 7, b 8 - Matano - Taxols, their preparation and pharmaceutical preparations against malignant tumors containing them |
US5622986A (en) * | 1993-10-20 | 1997-04-22 | Enzon, Inc. | 2'-and/or 7-substituted taxanes |
AU4133096A (en) * | 1994-10-28 | 1996-05-23 | Research Foundation Of The State University Of New York, The | Taxoid derivatives, their preparation and their use as antitumor agents |
US6100411A (en) * | 1994-10-28 | 2000-08-08 | The Research Foundation Of State University Of New York | Taxoid anti-tumor agents and pharmaceutical compositions thereof |
US5801191A (en) * | 1995-06-01 | 1998-09-01 | Biophysica Foundation | Taxoids |
CN1097044C (zh) * | 1996-07-15 | 2002-12-25 | 亚库尔特株式会社总社 | 紫杉烷衍生物以及含有该衍生物的药物 |
JPH1192468A (ja) * | 1997-09-17 | 1999-04-06 | Yakult Honsha Co Ltd | 新規なタキサン誘導体 |
AU758418B2 (en) * | 1997-12-19 | 2003-03-20 | Kabushiki Kaisha Yakult Honsha | Taxane derivatives |
JP2003026673A (ja) * | 1999-03-05 | 2003-01-29 | Asahi Kasei Corp | 骨形成促進剤 |
-
2001
- 2001-02-02 IL IL14563501A patent/IL145635A0/xx unknown
- 2001-02-02 KR KR1020017012367A patent/KR20010111580A/ko not_active Application Discontinuation
- 2001-02-02 BR BR0104358-7A patent/BR0104358A/pt not_active IP Right Cessation
- 2001-02-02 WO PCT/US2001/003624 patent/WO2001057013A1/en not_active Application Discontinuation
- 2001-02-02 EP EP01906972A patent/EP1175414A1/en not_active Withdrawn
- 2001-02-02 HU HU0200995A patent/HUP0200995A3/hu unknown
- 2001-02-02 AU AU34810/01A patent/AU3481001A/en not_active Abandoned
- 2001-02-02 NZ NZ514073A patent/NZ514073A/xx not_active Application Discontinuation
- 2001-10-01 NO NO20014752A patent/NO20014752L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NZ514073A (en) | 2004-02-27 |
WO2001057013A1 (en) | 2001-08-09 |
KR20010111580A (ko) | 2001-12-19 |
HUP0200995A2 (hu) | 2002-07-29 |
IL145635A0 (en) | 2002-06-30 |
EP1175414A1 (en) | 2002-01-30 |
NO20014752D0 (no) | 2001-10-01 |
NO20014752L (no) | 2001-11-27 |
AU3481001A (en) | 2001-08-14 |
HUP0200995A3 (en) | 2005-02-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 1963 DE 19.08.2008. |