BR0104354A - Taxanos substituìdos com éster c10 - Google Patents
Taxanos substituìdos com éster c10Info
- Publication number
- BR0104354A BR0104354A BR0104354-4A BR0104354A BR0104354A BR 0104354 A BR0104354 A BR 0104354A BR 0104354 A BR0104354 A BR 0104354A BR 0104354 A BR0104354 A BR 0104354A
- Authority
- BR
- Brazil
- Prior art keywords
- taxanes
- ester
- replaced
- substituent
- side chain
- Prior art date
Links
- 229940123237 Taxane Drugs 0.000 title abstract 3
- 150000002148 esters Chemical class 0.000 title abstract 2
- 125000004185 ester group Chemical group 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
- B65D—CONTAINERS FOR STORAGE OR TRANSPORT OF ARTICLES OR MATERIALS, e.g. BAGS, BARRELS, BOTTLES, BOXES, CANS, CARTONS, CRATES, DRUMS, JARS, TANKS, HOPPERS, FORWARDING CONTAINERS; ACCESSORIES, CLOSURES, OR FITTINGS THEREFOR; PACKAGING ELEMENTS; PACKAGES
- B65D83/00—Containers or packages with special means for dispensing contents
- B65D83/14—Containers for dispensing liquid or semi-liquid contents by internal gaseous pressure, i.e. aerosol containers comprising propellant
- B65D83/75—Aerosol containers not provided for in groups B65D83/16 - B65D83/74
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Dispersion Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Mechanical Engineering (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17978200P | 2000-02-02 | 2000-02-02 | |
| PCT/US2001/003623 WO2001057032A1 (en) | 2000-02-02 | 2001-02-02 | C10 ester substituted taxanes as antitumor agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0104354A true BR0104354A (pt) | 2002-01-02 |
Family
ID=22657972
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0104354-4A BR0104354A (pt) | 2000-02-02 | 2001-02-02 | Taxanos substituìdos com éster c10 |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP1165553B1 (enExample) |
| JP (1) | JP2003522172A (enExample) |
| CN (1) | CN1380882A (enExample) |
| AT (1) | ATE432928T1 (enExample) |
| AU (1) | AU782150B2 (enExample) |
| BG (1) | BG64889B1 (enExample) |
| BR (1) | BR0104354A (enExample) |
| CA (1) | CA2368274C (enExample) |
| CZ (1) | CZ20013430A3 (enExample) |
| DE (1) | DE60138853D1 (enExample) |
| GE (1) | GEP20043323B (enExample) |
| HU (1) | HUP0600302A2 (enExample) |
| IL (1) | IL145638A (enExample) |
| MX (1) | MXPA01009905A (enExample) |
| NO (1) | NO327910B1 (enExample) |
| NZ (1) | NZ514382A (enExample) |
| PL (1) | PL202957B1 (enExample) |
| RO (1) | RO121270B1 (enExample) |
| RU (1) | RU2262506C2 (enExample) |
| SK (1) | SK13692001A3 (enExample) |
| TR (1) | TR200102858T1 (enExample) |
| TW (1) | TWI299732B (enExample) |
| UA (1) | UA75039C2 (enExample) |
| WO (1) | WO2001057032A1 (enExample) |
| ZA (1) | ZA200108055B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6649632B2 (en) | 2000-02-02 | 2003-11-18 | Fsu Research Foundation, Inc. | C10 ester substituted taxanes |
| CA2354471A1 (en) * | 2001-07-31 | 2003-01-31 | Florida State University Research Foundation, Inc. | C10 ester substituted taxanes |
| SG129990A1 (en) * | 2001-08-01 | 2007-03-20 | Univ Florida State Res Found | C10 ester substituted taxanes |
| SV2006002010A (es) | 2004-02-13 | 2006-08-23 | Univ Florida State Res Found | Taxanos sustituidos con esteres de ciclopentilo en c10 |
| WO2006088767A2 (en) * | 2005-02-14 | 2006-08-24 | Florida State University Research Foundation, Inc. | C10 cyclopropyl ester substituted taxane compositions |
| US8242166B2 (en) | 2008-03-31 | 2012-08-14 | Florida State University Research Foundation, Inc. | C(10) ethyl ester and C(10) cyclopropyl ester substituted taxanes |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2601675B1 (fr) * | 1986-07-17 | 1988-09-23 | Rhone Poulenc Sante | Derives du taxol, leur preparation et les compositions pharmaceutiques qui les contiennent |
| US5243045A (en) * | 1991-09-23 | 1993-09-07 | Florida State University | Certain alkoxy substituted taxanes and pharmaceutical compositions containing them |
| US5250683A (en) * | 1991-09-23 | 1993-10-05 | Florida State University | Certain substituted taxanes and pharmaceutical compositions containing them |
| IL108443A0 (en) * | 1993-01-29 | 1994-04-12 | Univ Florida State | C7 taxane derivatives and pharmaceutical compositions containing them |
| CA2158863C (en) * | 1993-03-22 | 2006-12-19 | Robert A. Holton | Taxanes having a pyridyl substituted side-chain |
| EP0690711B1 (en) * | 1993-03-22 | 2000-08-16 | Florida State University | Taxanes having an amino substituted side-chain |
| PT1228759E (pt) * | 1993-03-22 | 2005-04-29 | Univ Florida State | Composicoes farmaceuticas contendo um taxano possuindo uma cadeia lateral substituida com furilo ou tienilo |
| US5475011A (en) * | 1993-03-26 | 1995-12-12 | The Research Foundation Of State University Of New York | Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment |
| US6100411A (en) * | 1994-10-28 | 2000-08-08 | The Research Foundation Of State University Of New York | Taxoid anti-tumor agents and pharmaceutical compositions thereof |
| WO1996013495A1 (en) * | 1994-10-28 | 1996-05-09 | The Research Foundation Of State University Of New York | Taxoid derivatives, their preparation and their use as antitumor agents |
| CA2255615C (en) * | 1996-05-22 | 2006-08-29 | Neuromedica, Inc. | Compositions comprising conjugates of cis-docosahexaenoic acid and docetaxel |
| US5795909A (en) * | 1996-05-22 | 1998-08-18 | Neuromedica, Inc. | DHA-pharmaceutical agent conjugates of taxanes |
| AU758418B2 (en) * | 1997-12-19 | 2003-03-20 | Kabushiki Kaisha Yakult Honsha | Taxane derivatives |
| JP2003026673A (ja) * | 1999-03-05 | 2003-01-29 | Asahi Kasei Corp | 骨形成促進剤 |
-
2001
- 2001-02-02 RO ROA200101083A patent/RO121270B1/ro unknown
- 2001-02-02 CA CA002368274A patent/CA2368274C/en not_active Expired - Fee Related
- 2001-02-02 HU HU0600302A patent/HUP0600302A2/hu unknown
- 2001-02-02 CN CN01800568A patent/CN1380882A/zh active Pending
- 2001-02-02 SK SK1369-2001A patent/SK13692001A3/sk unknown
- 2001-02-02 IL IL145638A patent/IL145638A/en not_active IP Right Cessation
- 2001-02-02 PL PL351380A patent/PL202957B1/pl not_active IP Right Cessation
- 2001-02-02 JP JP2001557864A patent/JP2003522172A/ja active Pending
- 2001-02-02 GE GE4523A patent/GEP20043323B/en unknown
- 2001-02-02 WO PCT/US2001/003623 patent/WO2001057032A1/en not_active Ceased
- 2001-02-02 CZ CZ20013430A patent/CZ20013430A3/cs unknown
- 2001-02-02 NZ NZ514382A patent/NZ514382A/en unknown
- 2001-02-02 UA UA2001106733A patent/UA75039C2/uk unknown
- 2001-02-02 AT AT01906971T patent/ATE432928T1/de not_active IP Right Cessation
- 2001-02-02 DE DE60138853T patent/DE60138853D1/de not_active Expired - Lifetime
- 2001-02-02 EP EP01906971A patent/EP1165553B1/en not_active Expired - Lifetime
- 2001-02-02 MX MXPA01009905A patent/MXPA01009905A/es active IP Right Grant
- 2001-02-02 RU RU2001129501/04A patent/RU2262506C2/ru active
- 2001-02-02 AU AU34809/01A patent/AU782150B2/en not_active Ceased
- 2001-02-02 BR BR0104354-4A patent/BR0104354A/pt not_active IP Right Cessation
- 2001-02-02 TR TR2001/02858T patent/TR200102858T1/xx unknown
- 2001-03-27 TW TW090102238A patent/TWI299732B/zh not_active IP Right Cessation
- 2001-10-01 NO NO20014754A patent/NO327910B1/no not_active IP Right Cessation
- 2001-10-01 ZA ZA200108055A patent/ZA200108055B/en unknown
- 2001-10-01 BG BG105965A patent/BG64889B1/bg unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HUP0600302A2 (en) | 2006-07-28 |
| TR200102858T1 (tr) | 2002-12-23 |
| RU2262506C2 (ru) | 2005-10-20 |
| PL351380A1 (en) | 2003-04-07 |
| ATE432928T1 (de) | 2009-06-15 |
| BG64889B1 (bg) | 2006-08-31 |
| IL145638A (en) | 2011-05-31 |
| IL145638A0 (en) | 2002-06-30 |
| GEP20043323B (en) | 2004-02-10 |
| AU3480901A (en) | 2001-08-14 |
| SK13692001A3 (sk) | 2002-07-02 |
| NZ514382A (en) | 2004-05-28 |
| JP2003522172A (ja) | 2003-07-22 |
| TWI299732B (en) | 2008-08-11 |
| EP1165553B1 (en) | 2009-06-03 |
| RO121270B1 (ro) | 2007-02-28 |
| PL202957B1 (pl) | 2009-08-31 |
| CZ20013430A3 (cs) | 2002-04-17 |
| EP1165553A1 (en) | 2002-01-02 |
| NO20014754D0 (no) | 2001-10-01 |
| AU782150B2 (en) | 2005-07-07 |
| BG105965A (en) | 2002-07-31 |
| UA75039C2 (en) | 2006-03-15 |
| NO327910B1 (no) | 2009-10-19 |
| NO20014754L (no) | 2001-11-29 |
| CN1380882A (zh) | 2002-11-20 |
| ZA200108055B (en) | 2003-12-01 |
| CA2368274C (en) | 2009-10-13 |
| CA2368274A1 (en) | 2001-08-09 |
| MXPA01009905A (es) | 2003-08-20 |
| DE60138853D1 (de) | 2009-07-16 |
| WO2001057032A1 (en) | 2001-08-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE 10A. E 11A. ANUIDADE(S). |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2138 DE 27/12/2011. |