BR0008510A - Sistemas policìclicos de 2-amino-tiazol, processo para a sua preparação e medicamento contendo estes compostos - Google Patents
Sistemas policìclicos de 2-amino-tiazol, processo para a sua preparação e medicamento contendo estes compostosInfo
- Publication number
- BR0008510A BR0008510A BR0008510-3A BR0008510A BR0008510A BR 0008510 A BR0008510 A BR 0008510A BR 0008510 A BR0008510 A BR 0008510A BR 0008510 A BR0008510 A BR 0008510A
- Authority
- BR
- Brazil
- Prior art keywords
- polycyclic
- compounds
- preparation
- amino
- medicine containing
- Prior art date
Links
- RAIPHJJURHTUIC-UHFFFAOYSA-N 1,3-thiazol-2-amine Chemical compound NC1=NC=CS1 RAIPHJJURHTUIC-UHFFFAOYSA-N 0.000 title abstract 3
- 125000003367 polycyclic group Chemical group 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- 230000001539 anorectic effect Effects 0.000 abstract 1
- 206010061428 decreased appetite Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Child & Adolescent Psychology (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19908538A DE19908538A1 (de) | 1999-02-26 | 1999-02-26 | Polycyclische 2-Amino-Thiazol Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen |
| PCT/EP2000/000924 WO2000051995A1 (de) | 1999-02-26 | 2000-02-05 | Polycyclische 2-amino-thiazol systeme, verfahren zu ihrer herstellung und arzneimittel enthaltend diese verbindungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0008510A true BR0008510A (pt) | 2002-02-05 |
Family
ID=7899082
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0008510-3A BR0008510A (pt) | 1999-02-26 | 2000-02-05 | Sistemas policìclicos de 2-amino-tiazol, processo para a sua preparação e medicamento contendo estes compostos |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US6251922B1 (https=) |
| EP (1) | EP1157015B1 (https=) |
| JP (1) | JP4728484B2 (https=) |
| KR (1) | KR20010102390A (https=) |
| CN (1) | CN1148362C (https=) |
| AT (1) | ATE295357T1 (https=) |
| AU (1) | AU763111B2 (https=) |
| BR (1) | BR0008510A (https=) |
| CA (1) | CA2364900A1 (https=) |
| DE (2) | DE19908538A1 (https=) |
| ES (1) | ES2240070T3 (https=) |
| HK (1) | HK1043117B (https=) |
| PT (1) | PT1157015E (https=) |
| WO (1) | WO2000051995A1 (https=) |
| ZA (1) | ZA200106198B (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19908537A1 (de) * | 1999-02-26 | 2000-08-31 | Aventis Pharma Gmbh | Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas |
| US7732484B2 (en) * | 2000-08-01 | 2010-06-08 | University Of Virginia Patent Foundation | Use of selective adenosine A1 receptor allosteric enhancers to manipulate angiogenesis |
| JP2005529846A (ja) * | 2002-01-16 | 2005-10-06 | ユニバーシティ オブ バージニア パテント ファウンデーション | Ａ１アデノシン受容体の２−アミノチアゾールアロステリックエンハンサ |
| ES2480994T3 (es) | 2008-03-31 | 2014-07-29 | Genentech, Inc. | Compuestos de tipo benzopirano y benzoxepina inhibidores de PI3K y métodos de uso |
| ES2558742T3 (es) | 2009-09-28 | 2016-02-08 | F. Hoffmann-La Roche Ag | Compuestos inhibidores de PI3K de benzoxepina y métodos de uso |
| ES2570569T3 (es) | 2009-09-28 | 2016-05-19 | Hoffmann La Roche | Compuestos de benzoxazepina como inhibidores de la PI3K y métodos de uso |
| JP5728487B2 (ja) * | 2009-10-29 | 2015-06-03 | ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ | 三環式ヘテロ環化合物 |
| WO2012126901A1 (en) | 2011-03-21 | 2012-09-27 | F. Hoffmann-La Roche Ag | Benzoxazepin compounds selective for pi3k p110 delta and methods of use |
| ES2859478T3 (es) | 2016-09-02 | 2021-10-04 | Bristol Myers Squibb Co | Compuestos heterocíclicos tricíclicos sustituidos |
| WO2019032631A1 (en) | 2017-08-09 | 2019-02-14 | Bristol-Myers Squibb Company | Oxime ether compounds |
| US11046646B2 (en) | 2017-08-09 | 2021-06-29 | Bristol-Myers Squibb Company | Alkylphenyl compounds |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4082773A (en) * | 1972-07-03 | 1978-04-04 | E. R. Squibb & Sons, Inc. | Tricyclic tetrahydro naphthaleneols and related compounds |
| DE2640358A1 (de) * | 1976-09-08 | 1978-03-16 | Hoechst Ag | Thiazolidinderivate und verfahren zu ihrer herstellung |
| CA1292226C (en) * | 1986-01-16 | 1991-11-19 | Terumi Hachiya | Indenothiazole derivative and process for preparing the same |
| IE68593B1 (en) | 1989-12-06 | 1996-06-26 | Sanofi Sa | Heterocyclic substituted acylaminothiazoles their preparation and pharmaceutical compositions containing them |
| TW416953B (en) * | 1996-09-25 | 2001-01-01 | Takeda Chemical Industries Ltd | Tricyclic compounds for eliciting a prostaglandin I2 receptor agonistic effect, their production and use |
| AU3289299A (en) * | 1998-02-19 | 1999-09-06 | Tularik Inc. | Antiviral agents |
| DE19831878C2 (de) * | 1998-07-17 | 2001-05-17 | Aventis Pharma Gmbh | Polycyclische Thiazolidin-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| DE19908537A1 (de) * | 1999-02-26 | 2000-08-31 | Aventis Pharma Gmbh | Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas |
-
1999
- 1999-02-26 DE DE19908538A patent/DE19908538A1/de not_active Withdrawn
-
2000
- 2000-02-05 AU AU32782/00A patent/AU763111B2/en not_active Ceased
- 2000-02-05 BR BR0008510-3A patent/BR0008510A/pt not_active IP Right Cessation
- 2000-02-05 CN CNB008042217A patent/CN1148362C/zh not_active Expired - Fee Related
- 2000-02-05 AT AT00910642T patent/ATE295357T1/de not_active IP Right Cessation
- 2000-02-05 ES ES00910642T patent/ES2240070T3/es not_active Expired - Lifetime
- 2000-02-05 JP JP2000602222A patent/JP4728484B2/ja not_active Expired - Fee Related
- 2000-02-05 PT PT00910642T patent/PT1157015E/pt unknown
- 2000-02-05 DE DE50010285T patent/DE50010285D1/de not_active Expired - Lifetime
- 2000-02-05 CA CA002364900A patent/CA2364900A1/en not_active Abandoned
- 2000-02-05 EP EP00910642A patent/EP1157015B1/de not_active Expired - Lifetime
- 2000-02-05 KR KR1020017010839A patent/KR20010102390A/ko not_active Ceased
- 2000-02-05 WO PCT/EP2000/000924 patent/WO2000051995A1/de not_active Ceased
- 2000-02-05 HK HK02104079.4A patent/HK1043117B/zh not_active IP Right Cessation
- 2000-02-10 US US09/501,208 patent/US6251922B1/en not_active Expired - Lifetime
-
2001
- 2001-07-27 ZA ZA200106198A patent/ZA200106198B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HK1043117B (zh) | 2004-10-08 |
| DE50010285D1 (de) | 2005-06-16 |
| AU763111B2 (en) | 2003-07-10 |
| CN1148362C (zh) | 2004-05-05 |
| JP4728484B2 (ja) | 2011-07-20 |
| ZA200106198B (en) | 2002-05-03 |
| DE19908538A1 (de) | 2000-08-31 |
| ES2240070T3 (es) | 2005-10-16 |
| JP2002538148A (ja) | 2002-11-12 |
| US6251922B1 (en) | 2001-06-26 |
| EP1157015A1 (de) | 2001-11-28 |
| ATE295357T1 (de) | 2005-05-15 |
| PT1157015E (pt) | 2005-08-31 |
| EP1157015B1 (de) | 2005-05-11 |
| KR20010102390A (ko) | 2001-11-15 |
| HK1043117A1 (en) | 2002-09-06 |
| CA2364900A1 (en) | 2000-09-08 |
| WO2000051995A1 (de) | 2000-09-08 |
| AU3278200A (en) | 2000-09-21 |
| CN1344263A (zh) | 2002-04-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A, 8A E 9A ANUIDADES |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009. |