BG65878B1 - Многосъставна лекарствена форма, съдържаща най-малко две различни покрити пелетни форми - Google Patents

Многосъставна лекарствена форма, съдържаща най-малко две различни покрити пелетни форми Download PDF

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Publication number
BG65878B1
BG65878B1 BG107147A BG10714702A BG65878B1 BG 65878 B1 BG65878 B1 BG 65878B1 BG 107147 A BG107147 A BG 107147A BG 10714702 A BG10714702 A BG 10714702A BG 65878 B1 BG65878 B1 BG 65878B1
Authority
BG
Bulgaria
Prior art keywords
weight
meth
active ingredient
release
pellet
Prior art date
Application number
BG107147A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG107147A (bg
Inventor
Thomas Beckert
Hans-Ulrich Petereit
Jennifer Dressman
Markus Rudolph
Original Assignee
Roehm Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2001/002679 external-priority patent/WO2002060415A1/de
Application filed by Roehm Gmbh & Co. Kg filed Critical Roehm Gmbh & Co. Kg
Publication of BG107147A publication Critical patent/BG107147A/bg
Publication of BG65878B1 publication Critical patent/BG65878B1/bg

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/60—Salicylic acid; Derivatives thereof
    • A61K31/606—Salicylic acid; Derivatives thereof having amino groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
BG107147A 2001-01-31 2002-09-26 Многосъставна лекарствена форма, съдържаща най-малко две различни покрити пелетни форми BG65878B1 (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10104504 2001-01-31
DE10104880A DE10104880A1 (de) 2001-01-31 2001-02-01 Multipartikuläre Arzneiform, enthaltend mindestens zwei unterschiedlich überzogene Pelletformen
PCT/EP2001/002679 WO2002060415A1 (de) 2001-01-31 2001-03-09 Multipartikuläre arzneiform, enthaltend mindestens zwei unterschiedlich überzogene pelletformen

Publications (2)

Publication Number Publication Date
BG107147A BG107147A (bg) 2003-05-30
BG65878B1 true BG65878B1 (bg) 2010-04-30

Family

ID=7672474

Family Applications (1)

Application Number Title Priority Date Filing Date
BG107147A BG65878B1 (bg) 2001-01-31 2002-09-26 Многосъставна лекарствена форма, съдържаща най-малко две различни покрити пелетни форми

Country Status (5)

Country Link
BG (1) BG65878B1 (pt)
BR (1) BRPI0109640B8 (pt)
DE (1) DE10104880A1 (pt)
IL (1) IL151150A (pt)
MX (1) MX2007010610A (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102008048729A1 (de) * 2008-09-24 2010-03-25 Add Technologies Ltd Advanced Drug Delivery Multipartikuläre Tabletten und Verfahren zur deren Herstellung
GB201118182D0 (en) * 2011-10-21 2011-12-07 Jagotec Ag Improvements in or relating to organic compounds
DE102012105528A1 (de) 2012-06-25 2014-01-02 Hennig Arzneimittel Gmbh & Co. Kg Arzneiform zur Freisetzung von Wirkstoffen

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1617751A1 (de) * 1966-08-12 1971-04-08 Roehm & Haas Gmbh Dragierlack fuer Arzneiformen
EP0181515A2 (de) * 1984-10-19 1986-05-21 Röhm Gmbh Verfahren zur Herstellung einer wässrigen Überzugsmitteldispersion und ihre Verwendung zum Überziehen von Arzneimitteln
EP0629398A1 (en) * 1993-06-18 1994-12-21 Tanabe Seiyaku Co., Ltd. Pharmaceutical preparation for controlled release of a medicinal compound at a targeted site in the intestinal tract
EP0704207A2 (de) * 1994-08-31 1996-04-03 Röhm GmbH Thermoplastischer Kunststoff für darmsaftlösliche Arznei-Umhüllungen
EP0704208A2 (de) * 1994-08-31 1996-04-03 Röhm GmbH Überzugs- und Bindemittel für Arzneiformen sowie damit hergestellte Arzneiform
EP0727205A2 (de) * 1995-02-16 1996-08-21 Röhm Gmbh Thermoplastisches Überzugs- und Bindemittel für Arzneiformen

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1617751A1 (de) * 1966-08-12 1971-04-08 Roehm & Haas Gmbh Dragierlack fuer Arzneiformen
EP0181515A2 (de) * 1984-10-19 1986-05-21 Röhm Gmbh Verfahren zur Herstellung einer wässrigen Überzugsmitteldispersion und ihre Verwendung zum Überziehen von Arzneimitteln
EP0629398A1 (en) * 1993-06-18 1994-12-21 Tanabe Seiyaku Co., Ltd. Pharmaceutical preparation for controlled release of a medicinal compound at a targeted site in the intestinal tract
EP0704207A2 (de) * 1994-08-31 1996-04-03 Röhm GmbH Thermoplastischer Kunststoff für darmsaftlösliche Arznei-Umhüllungen
EP0704208A2 (de) * 1994-08-31 1996-04-03 Röhm GmbH Überzugs- und Bindemittel für Arzneiformen sowie damit hergestellte Arzneiform
EP0727205A2 (de) * 1995-02-16 1996-08-21 Röhm Gmbh Thermoplastisches Überzugs- und Bindemittel für Arzneiformen

Also Published As

Publication number Publication date
MX2007010610A (es) 2009-02-19
BRPI0109640B8 (pt) 2021-05-25
IL151150A (en) 2010-04-15
BG107147A (bg) 2003-05-30
BRPI0109640B1 (pt) 2020-03-10
BR0109640A (pt) 2003-04-22
DE10104880A1 (de) 2002-08-08

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BG65878B1 (bg) Многосъставна лекарствена форма, съдържаща най-малко две различни покрити пелетни форми