BG61610B2 - Ново пептидно активно вещество и метод за получаването му - Google Patents

Ново пептидно активно вещество и метод за получаването му Download PDF

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Publication number
BG61610B2
BG61610B2 BG100961A BG10096196A BG61610B2 BG 61610 B2 BG61610 B2 BG 61610B2 BG 100961 A BG100961 A BG 100961A BG 10096196 A BG10096196 A BG 10096196A BG 61610 B2 BG61610 B2 BG 61610B2
Authority
BG
Bulgaria
Prior art keywords
pro
val
meval
vai
formula
Prior art date
Application number
BG100961A
Other languages
Bulgarian (bg)
English (en)
Inventor
Wilhelm Amberg
Harald Bernard
Ernst Buschmann
Andreas Haupt
Lothar Janitschke
Bernd Janssen
Ulrich Karl
Andreas Kling
Stefan Mueller
Potzolli Bernd De
Kurt Ritter
Marco Thyes
Thomas Zierke
Original Assignee
Basf Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Aktiengesellschaft filed Critical Basf Aktiengesellschaft
Publication of BG61610B2 publication Critical patent/BG61610B2/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/101—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BG100961A 1994-05-06 1996-11-06 Ново пептидно активно вещество и метод за получаването му BG61610B2 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4415997A DE4415997A1 (de) 1994-05-06 1994-05-06 Neuer peptidischer Wirkstoff und dessen Herstellung
PCT/EP1995/001577 WO1995030691A1 (de) 1994-05-06 1995-04-26 Neuer peptidischer wirkstoff und dessen herstellung

Publications (1)

Publication Number Publication Date
BG61610B2 true BG61610B2 (bg) 1998-01-30

Family

ID=6517453

Family Applications (1)

Application Number Title Priority Date Filing Date
BG100961A BG61610B2 (bg) 1994-05-06 1996-11-06 Ново пептидно активно вещество и метод за получаването му

Country Status (28)

Country Link
US (1) US5864012A (pt)
EP (1) EP0758342B1 (pt)
JP (1) JPH09512803A (pt)
KR (1) KR100336139B1 (pt)
CN (1) CN1113067C (pt)
AT (1) ATE188485T1 (pt)
AU (1) AU688037B2 (pt)
BG (1) BG61610B2 (pt)
BR (1) BR9507623A (pt)
CZ (1) CZ288448B6 (pt)
DE (2) DE4415997A1 (pt)
DK (1) DK0758342T3 (pt)
ES (1) ES2141351T3 (pt)
FI (1) FI119642B (pt)
GR (1) GR3032630T3 (pt)
HR (1) HRP950271B1 (pt)
HU (1) HU220875B1 (pt)
IL (1) IL113544A (pt)
MX (1) MX9605402A (pt)
NO (1) NO317728B1 (pt)
NZ (1) NZ285092A (pt)
PL (1) PL180652B1 (pt)
PT (1) PT758342E (pt)
RU (1) RU2153504C2 (pt)
SI (1) SI9520061B (pt)
TW (1) TW408132B (pt)
WO (1) WO1995030691A1 (pt)
ZA (1) ZA953584B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4415998A1 (de) * 1994-05-06 1995-11-09 Basf Ag Neue Tetrapeptide, ihre Herstellung Verwendung
TW474946B (en) * 1995-12-15 2002-02-01 Basf Ag Novel compounds, the preparation and use thereof
US20010009901A1 (en) 1996-12-11 2001-07-26 Basf Aktiengesellschaft Germany Antineoplastic peptides
US7304750B2 (en) * 1999-12-17 2007-12-04 Nektar Therapeutics Systems and methods for non-destructive mass sensing
KR20020066476A (ko) * 2001-02-12 2002-08-19 쥬가이 세이야쿠 가부시키가이샤 펩타이드 유도체의 제조방법

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2136339C (en) * 1992-05-20 2008-02-05 Andreas Haupt Derivatives of dolastatin

Also Published As

Publication number Publication date
NO964688L (no) 1997-01-02
PT758342E (pt) 2000-04-28
CZ288448B6 (en) 2001-06-13
SI9520061B (sl) 2002-02-28
KR970702880A (ko) 1997-06-10
ES2141351T3 (es) 2000-03-16
NZ285092A (en) 1998-01-26
DE4415997A1 (de) 1995-11-09
EP0758342B1 (de) 2000-01-05
FI119642B (fi) 2009-01-30
DE59507578D1 (de) 2000-02-10
AU2408395A (en) 1995-11-29
HU9603067D0 (en) 1997-01-28
WO1995030691A1 (de) 1995-11-16
NO317728B1 (no) 2004-12-13
DK0758342T3 (da) 2000-05-01
CN1113067C (zh) 2003-07-02
IL113544A0 (en) 1995-07-31
HUT75861A (en) 1997-05-28
IL113544A (en) 2001-01-11
CN1162318A (zh) 1997-10-15
HRP950271A2 (en) 1997-08-31
MX9605402A (es) 1997-12-31
HRP950271B1 (en) 2000-08-31
ZA953584B (en) 1996-11-04
EP0758342A1 (de) 1997-02-19
PL180652B1 (pl) 2001-03-30
FI964448A0 (fi) 1996-11-05
FI964448A (fi) 1996-11-05
RU2153504C2 (ru) 2000-07-27
PL321159A1 (en) 1997-11-24
HU220875B1 (en) 2002-06-29
TW408132B (en) 2000-10-11
US5864012A (en) 1999-01-26
JPH09512803A (ja) 1997-12-22
BR9507623A (pt) 1997-10-07
AU688037B2 (en) 1998-03-05
GR3032630T3 (en) 2000-05-31
KR100336139B1 (ko) 2002-09-25
SI9520061A (en) 1997-06-30
NO964688D0 (no) 1996-11-05
ATE188485T1 (de) 2000-01-15
CZ326096A3 (en) 1997-04-16

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