BG60539B2 - Антибактериални средства - Google Patents

Антибактериални средства Download PDF

Info

Publication number
BG60539B2
BG60539B2 BG098514A BG9851494A BG60539B2 BG 60539 B2 BG60539 B2 BG 60539B2 BG 098514 A BG098514 A BG 098514A BG 9851494 A BG9851494 A BG 9851494A BG 60539 B2 BG60539 B2 BG 60539B2
Authority
BG
Bulgaria
Prior art keywords
group
compound
formula
dissolved
carbamoyloxymethyl
Prior art date
Application number
BG098514A
Other languages
Bulgarian (bg)
English (en)
Inventor
Maurizio Foglio
Giovanni Franceschi
Cosimo Scarafile
Federico Arcamone
Aurora Sanfilippo
Original Assignee
Farmitalia Carlo Erba S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba S.P.A. filed Critical Farmitalia Carlo Erba S.P.A.
Publication of BG60539B2 publication Critical patent/BG60539B2/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG098514A 1981-05-06 1994-02-22 Антибактериални средства BG60539B2 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/261,247 US4482565A (en) 1980-02-22 1981-05-06 β-Lactam-containing antibacterial agents and β-lactamase inhibitors

Publications (1)

Publication Number Publication Date
BG60539B2 true BG60539B2 (bg) 1995-07-28

Family

ID=22992480

Family Applications (1)

Application Number Title Priority Date Filing Date
BG098514A BG60539B2 (bg) 1981-05-06 1994-02-22 Антибактериални средства

Country Status (6)

Country Link
US (1) US4482565A (cs)
BG (1) BG60539B2 (cs)
CS (1) CS415491A3 (cs)
GB (1) GB2097786B (cs)
HK (1) HK74587A (cs)
SG (1) SG34487G (cs)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4558042A (en) * 1981-05-06 1985-12-10 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
US4508649A (en) * 1981-12-11 1985-04-02 Farmitalia Carlo Erba Process for preparing optically active penems
NO831160L (no) * 1982-04-08 1983-10-10 Erba Farmitalia Fremstilling av substituerte penem-derivater
US4794109A (en) * 1982-11-16 1988-12-27 Ciba-Geigy Corporation 6-hydroxy-lower alkylpenem compounds, pharmaceutical preparations that contain these compounds, and the use of the latter
GB8300295D0 (en) * 1983-01-06 1983-02-09 Erba Farmitalia Penem esters
US4504485A (en) * 1983-04-04 1985-03-12 Schering Corporation 5R,6S,8R-6-(1-Hydroxyethyl)-2-(2-carbamoyloxyethylthio)-penem-3-carboxylic acid
US4559333A (en) * 1984-03-01 1985-12-17 Schering Corporation Hydrazone substituted penems
GB8416652D0 (en) 1984-06-29 1984-08-01 Erba Farmitalia Penem derivatives
GB8605549D0 (en) * 1986-03-06 1986-04-09 Erba Farmitalia Penem derivatives
GB8713515D0 (en) * 1987-06-10 1987-07-15 Erba Farmitalia Methoxymethyl compounds
GB8714413D0 (en) * 1987-06-19 1987-07-22 Erba Farmitalia 6-substituted penem esters
JP2599610B2 (ja) * 1988-03-01 1997-04-09 大鵬薬品工業株式会社 ２β―置換メチルペニシリン誘導体の製造法
GB8818789D0 (en) 1988-08-08 1988-09-07 Erba Carlo Spa Crystalline(5r 6s)-2-carbamoyloxymethyl-6-((1r)-hydroxyethyl)-2-penem-carboxylic acid & pharmaceutical formulation
US5191075A (en) * 1988-10-19 1993-03-02 Pfizer Inc Process for the preparation of penems
US4992543A (en) * 1988-10-19 1991-02-12 Pfizer Inc. Penem derivatives
GB9006114D0 (en) * 1990-03-19 1990-05-16 Erba Carlo Spa Process for preparing penem esters
IT1239275B (it) * 1990-05-16 1993-10-01 Menarini Farma Ind Penem ditiocarbammati, loro uso e procedimento di fabbricazione relativi
IE65926B1 (en) * 1990-07-19 1995-11-29 Shionogi & Co Thioalkylthio cephalosporin derivatives
EP0597401A3 (en) * 1992-11-11 1995-07-26 Takeda Chemical Industries Ltd Preparation of penemes.
ATE221889T1 (de) * 1998-05-13 2002-08-15 Lg Chemical Ltd Cephalosporin-derivate, verfahren zu ihrer herstellung und diese enthaltende antimikrobielle mittel
US6720445B2 (en) 2000-12-21 2004-04-13 Beacon Laboratories, Inc. Acetyloxymethyl esters and methods for using the same

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU77306A1 (cs) * 1977-05-09 1979-01-18
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
US4374065A (en) * 1979-09-21 1983-02-15 Bristol-Myers Company Antibacterial agents of the β-lactam type
US4340539A (en) * 1980-01-21 1982-07-20 Bristol-Myers Company Derivatives of 6-bromo penicillanic acid

Also Published As

Publication number Publication date
GB2097786B (en) 1984-08-22
GB2097786A (en) 1982-11-10
US4482565A (en) 1984-11-13
CS415491A3 (en) 1992-06-17
US4482565B1 (cs) 1987-11-03
HK74587A (en) 1987-10-23
SG34487G (en) 1987-07-24

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