BG36928A3 - Method for preparing pharmacologically active peptides - Google Patents

Method for preparing pharmacologically active peptides

Info

Publication number
BG36928A3
BG36928A3 BG053871A BG5387181A BG36928A3 BG 36928 A3 BG36928 A3 BG 36928A3 BG 053871 A BG053871 A BG 053871A BG 5387181 A BG5387181 A BG 5387181A BG 36928 A3 BG36928 A3 BG 36928A3
Authority
BG
Bulgaria
Prior art keywords
pharmacologically active
active peptides
preparing pharmacologically
preparing
peptides
Prior art date
Application number
BG053871A
Other languages
Bulgarian (bg)
English (en)
Inventor
Paul Gesellchen
Robert Shuman
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of BG36928A3 publication Critical patent/BG36928A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1027—Tetrapeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
BG053871A 1980-10-20 1981-10-16 Method for preparing pharmacologically active peptides BG36928A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/198,900 US4322340A (en) 1980-10-20 1980-10-20 Pharmacologically active peptides

Publications (1)

Publication Number Publication Date
BG36928A3 true BG36928A3 (en) 1985-02-15

Family

ID=22735344

Family Applications (1)

Application Number Title Priority Date Filing Date
BG053871A BG36928A3 (en) 1980-10-20 1981-10-16 Method for preparing pharmacologically active peptides

Country Status (27)

Country Link
US (1) US4322340A (el)
EP (1) EP0050502B1 (el)
JP (1) JPS57108052A (el)
KR (1) KR830007518A (el)
AR (1) AR230046A1 (el)
AT (1) ATE6777T1 (el)
AU (1) AU547221B2 (el)
BG (1) BG36928A3 (el)
CA (1) CA1187871A (el)
DD (1) DD200798A5 (el)
DE (1) DE3162823D1 (el)
DK (1) DK461481A (el)
ES (1) ES506316A0 (el)
FI (1) FI813198L (el)
GB (1) GB2085893B (el)
GR (1) GR75342B (el)
HU (1) HU185320B (el)
IE (1) IE52186B1 (el)
IL (1) IL64083A (el)
NZ (1) NZ198628A (el)
PH (1) PH17006A (el)
PL (1) PL131155B1 (el)
PT (1) PT73839B (el)
RO (1) RO83301B (el)
SU (1) SU1082319A3 (el)
YU (1) YU249081A (el)
ZA (1) ZA817063B (el)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0076557B1 (en) * 1981-06-22 1985-11-13 Imperial Chemical Industries Plc Peptides and pseudopeptides in which the n terminus bears two substituents
US4448717A (en) * 1982-11-12 1984-05-15 Eli Lilly And Company Pharmacologically active peptides
US4510082A (en) * 1983-03-07 1985-04-09 Eli Lilly And Company Pharmacologically active peptides
US4473497A (en) * 1983-03-07 1984-09-25 Eli Lilly And Company Pharmacologically active peptides
DK134784A (da) * 1983-03-07 1984-09-08 Lilly Co Eli Farmakologisk virksomme tripeptid-derivater og fremgangsmaade til fremstilling deraf
US4495178A (en) * 1983-10-06 1985-01-22 G. D. Searle & Co. Enkephalin analogs
JPH0449298A (ja) * 1990-06-19 1992-02-18 Univ New York State 新規なエンケファリン誘導体および鎮痛剤
US5209930A (en) * 1990-12-10 1993-05-11 Rohm And Haas Company Preparation and use of n-iodopropargyl oxycarbonyl amino acid esters and derivatives as antimicrobial agents
US5952465A (en) * 1993-04-23 1999-09-14 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site
AU6770794A (en) * 1993-04-23 1994-11-21 Herbert J. Evans Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site
US6258550B1 (en) 1993-04-23 2001-07-10 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site
US5965698A (en) * 1993-04-23 1999-10-12 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein--protein interaction site
US5928896A (en) * 1993-04-23 1999-07-27 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein--protein interaction site
US6084066A (en) * 1993-10-29 2000-07-04 Virginia Commonwealth University Polypetides that include conformation-constraining groups which flank a protein-protein interaction site

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1577115A (en) * 1976-07-27 1980-10-22 Reckitt & Colmann Prod Ltd Container closure units
CH619686A5 (en) * 1976-02-02 1980-10-15 Sandoz Ag Process for the preparation of novel peptides or peptide derivatives
DK28377A (da) * 1976-02-02 1977-08-03 Sandoz Ag Fremgangsmade til fremstilling af polypeptidderivater
US4264491A (en) * 1977-10-03 1981-04-28 Eli Lilly And Company Analgesic compounds
US4265808A (en) * 1979-12-17 1981-05-05 Eli Lilly And Company Pharmacologically active peptides

Also Published As

Publication number Publication date
FI813198L (fi) 1982-04-21
GB2085893A (en) 1982-05-06
IL64083A (en) 1985-03-31
ZA817063B (en) 1983-05-25
PL233498A1 (el) 1982-05-24
JPS57108052A (en) 1982-07-05
AU547221B2 (en) 1985-10-10
DK461481A (da) 1982-04-21
US4322340A (en) 1982-03-30
ES8306713A1 (es) 1983-06-01
RO83301B (ro) 1984-02-28
HU185320B (en) 1985-01-28
DD200798A5 (de) 1983-06-15
RO83301A (ro) 1984-02-21
NZ198628A (en) 1985-01-31
GB2085893B (en) 1984-03-21
KR830007518A (ko) 1983-10-21
YU249081A (en) 1983-12-31
ES506316A0 (es) 1983-06-01
AR230046A1 (es) 1984-02-29
PT73839A (en) 1981-11-01
GR75342B (el) 1984-07-13
IL64083A0 (en) 1982-01-31
PT73839B (en) 1983-01-17
EP0050502A1 (en) 1982-04-28
IE52186B1 (en) 1987-08-05
IE812442L (en) 1982-04-20
PL131155B1 (en) 1984-10-31
SU1082319A3 (ru) 1984-03-23
ATE6777T1 (de) 1984-04-15
DE3162823D1 (en) 1984-04-26
PH17006A (en) 1984-05-11
CA1187871A (en) 1985-05-28
EP0050502B1 (en) 1984-03-21
AU7657481A (en) 1982-04-29

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