BG17799A3 - Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини - Google Patents
Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидиниInfo
- Publication number
- BG17799A3 BG17799A3 BG016080A BG1773170A BG17799A3 BG 17799 A3 BG17799 A3 BG 17799A3 BG 016080 A BG016080 A BG 016080A BG 1773170 A BG1773170 A BG 1773170A BG 17799 A3 BG17799 A3 BG 17799A3
- Authority
- BG
- Bulgaria
- Prior art keywords
- thieno
- pyrimidines
- furyl
- nitro
- preparation
- Prior art date
Links
- 150000003230 pyrimidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19691959403 DE1959403A1 (de) | 1969-11-26 | 1969-11-26 | Neue 2-(5-Nitro-2-furyl)-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung |
| DE19702050816 DE2050816A1 (de) | 1970-10-16 | 1970-10-16 | Neue 2-(Nitro-2-furyl>thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine |
| DE19702050814 DE2050814A1 (de) | 1970-10-16 | 1970-10-16 | Neue Verfahren zur Herstellung von 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidinen |
| DE19702050815 DE2050815A1 (de) | 1970-10-16 | 1970-10-16 | Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG17799A3 true BG17799A3 (bg) | 1973-12-25 |
Family
ID=27430978
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG016080A BG17799A3 (bg) | 1969-11-26 | 1970-11-17 | Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини |
| BG017732A BG17800A3 (bg) | 1969-11-26 | 1970-11-17 | Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG017732A BG17800A3 (bg) | 1969-11-26 | 1970-11-17 | Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US3661908A (cg-RX-API-DMAC7.html) |
| BE (1) | BE759493A (cg-RX-API-DMAC7.html) |
| BG (2) | BG17799A3 (cg-RX-API-DMAC7.html) |
| CA (1) | CA926865A (cg-RX-API-DMAC7.html) |
| CH (3) | CH567029A5 (cg-RX-API-DMAC7.html) |
| DK (1) | DK128781B (cg-RX-API-DMAC7.html) |
| FR (1) | FR2073416B1 (cg-RX-API-DMAC7.html) |
| GB (1) | GB1321316A (cg-RX-API-DMAC7.html) |
| IE (1) | IE34765B1 (cg-RX-API-DMAC7.html) |
| IL (1) | IL35729A (cg-RX-API-DMAC7.html) |
| NL (1) | NL7017210A (cg-RX-API-DMAC7.html) |
| NO (1) | NO129954B (cg-RX-API-DMAC7.html) |
| SE (1) | SE377938B (cg-RX-API-DMAC7.html) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3932642A (en) * | 1971-04-10 | 1976-01-13 | Boehringer Ingelheim Gmbh | Biocidal compositions containing a 2- (5'-nitro-2'-furyl)-thieno(2,3-d) pyrimidine and methods of use |
| US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
| US6608053B2 (en) * | 2000-04-27 | 2003-08-19 | Yamanouchi Pharmaceutical Co., Ltd. | Fused heteroaryl derivatives |
| US20040138238A1 (en) * | 2002-08-08 | 2004-07-15 | Dhanoa Dale S. | Substituted aminopyrimidine compounds as neurokinin antagonists |
| GB0423653D0 (en) | 2004-10-25 | 2004-11-24 | Piramed Ltd | Pharmaceutical compounds |
| EP2046799B1 (en) * | 2006-04-26 | 2017-07-19 | Genentech, Inc. | Phosphoinositide 3-kinase inhibitor compounds and pharmaceutical compositions containing them |
| NZ572812A (en) * | 2006-04-26 | 2010-09-30 | Hoffmann La Roche | THIENO [3, 2-D] PYRIMIDINE Indazole DERIVATIVE USEFUL AS PI3K INHIBITOR |
| CL2007001167A1 (es) * | 2006-04-26 | 2008-01-25 | Genentech Inc | Compuestos derivados de pirimidina condensada, inhibidores de p13-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicionfarmaceutica. |
| JP5284977B2 (ja) * | 2006-12-07 | 2013-09-11 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | ホスホイノシチド3−キナーゼ阻害剤化合物及び使用方法 |
| WO2008073785A2 (en) * | 2006-12-07 | 2008-06-19 | Genentech, Inc. | Phosphoinositide 3-kinase inhibitor compounds and methods of use |
| EP2158207B1 (en) * | 2007-06-12 | 2011-05-25 | F. Hoffmann-La Roche AG | Thiazoliopyrimidines and their use as inhibitors of phosphatidylinositol-3 kinase |
| EP2207781B1 (en) * | 2007-09-24 | 2012-11-28 | Genentech, Inc. | Thiazolopyrimidine p13k inhibitor compounds and methods of use |
| WO2009055730A1 (en) * | 2007-10-25 | 2009-04-30 | Genentech, Inc. | Process for making thienopyrimidine compounds |
| GB0721095D0 (en) * | 2007-10-26 | 2007-12-05 | Piramed Ltd | Pharmaceutical compounds |
| MX2011009167A (es) | 2009-03-12 | 2011-09-15 | Genentech Inc | Combinaciones de compuestos inhibidores de fosfoinositida 3-cinasa y agentes quimioterapeuticos para el tratamiento contra neoplasia hemotopoyeticas malignas. |
| EP2451811A1 (en) * | 2009-05-27 | 2012-05-16 | F. Hoffmann-La Roche AG | Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use |
| MX2011012520A (es) * | 2009-05-27 | 2011-12-12 | Hoffmann La Roche | Compuestos inhibidores de pi3k de pirimidina biciclicos selectivos para p110 delta y metodos de uso de los mismos. |
| PE20121816A1 (es) * | 2009-10-12 | 2013-01-02 | Hoffmann La Roche | Combinaciones de un inhibidor de pi3k y un inhibidor de mek |
| CA2793892A1 (en) | 2010-04-16 | 2011-10-20 | Elizabeth Punnoose | Foxo3a as predictive biomarker for pi3k/akt kinase pathway inhibitor efficacy |
| US20140004209A1 (en) | 2010-12-22 | 2014-01-02 | Genentech, Inc. | Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms |
| EP2959014B1 (en) | 2013-02-25 | 2019-11-13 | Genentech, Inc. | Methods and compositions for detecting and treating drug resistant akt mutant |
-
0
- BE BE759493D patent/BE759493A/xx unknown
-
1970
- 1970-11-17 BG BG016080A patent/BG17799A3/xx unknown
- 1970-11-17 BG BG017732A patent/BG17800A3/xx unknown
- 1970-11-18 US US90841A patent/US3661908A/en not_active Expired - Lifetime
- 1970-11-23 CH CH1514674A patent/CH567029A5/xx not_active IP Right Cessation
- 1970-11-23 CH CH1514974A patent/CH568324A5/xx not_active IP Right Cessation
- 1970-11-23 CH CH1731270A patent/CH559210A5/xx not_active IP Right Cessation
- 1970-11-25 NO NO04524/70A patent/NO129954B/no unknown
- 1970-11-25 NL NL7017210A patent/NL7017210A/xx unknown
- 1970-11-25 DK DK601570AA patent/DK128781B/da unknown
- 1970-11-25 GB GB5614670A patent/GB1321316A/en not_active Expired
- 1970-11-26 IL IL35729A patent/IL35729A/xx unknown
- 1970-11-26 IE IE1519/70A patent/IE34765B1/xx unknown
- 1970-11-26 FR FR7042531A patent/FR2073416B1/fr not_active Expired
- 1970-11-26 CA CA099166A patent/CA926865A/en not_active Expired
- 1970-11-26 SE SE7016054A patent/SE377938B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CH568324A5 (cg-RX-API-DMAC7.html) | 1975-10-31 |
| GB1321316A (en) | 1973-06-27 |
| IE34765B1 (en) | 1975-08-06 |
| SE377938B (cg-RX-API-DMAC7.html) | 1975-08-04 |
| NO129954B (cg-RX-API-DMAC7.html) | 1974-06-17 |
| DK128781B (da) | 1974-07-01 |
| CH559210A5 (cg-RX-API-DMAC7.html) | 1975-02-28 |
| FR2073416A1 (cg-RX-API-DMAC7.html) | 1971-10-01 |
| BE759493A (fr) | 1971-05-25 |
| IL35729A0 (en) | 1971-01-28 |
| FR2073416B1 (cg-RX-API-DMAC7.html) | 1975-04-18 |
| NL7017210A (cg-RX-API-DMAC7.html) | 1971-05-28 |
| IE34765L (en) | 1971-05-26 |
| IL35729A (en) | 1974-01-14 |
| BG17800A3 (bg) | 1973-12-25 |
| US3661908A (en) | 1972-05-09 |
| CH567029A5 (cg-RX-API-DMAC7.html) | 1975-09-30 |
| CA926865A (en) | 1973-05-22 |
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