BG108075A - Използване на производни на епотилон за лечение на трудно лечими тумори - Google Patents

Използване на производни на епотилон за лечение на трудно лечими тумори Download PDF

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Publication number
BG108075A
BG108075A BG108075A BG10807503A BG108075A BG 108075 A BG108075 A BG 108075A BG 108075 A BG108075 A BG 108075A BG 10807503 A BG10807503 A BG 10807503A BG 108075 A BG108075 A BG 108075A
Authority
BG
Bulgaria
Prior art keywords
methyl
thiazolyl
ethenyl
dione
dihydroxy
Prior art date
Application number
BG108075A
Other languages
Bulgarian (bg)
English (en)
Inventor
Francis Lee
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23028846&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG108075(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of BG108075A publication Critical patent/BG108075A/bg

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BG108075A 2001-02-20 2003-08-07 Използване на производни на епотилон за лечение на трудно лечими тумори BG108075A (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US26983601P 2001-02-20 2001-02-20

Publications (1)

Publication Number Publication Date
BG108075A true BG108075A (bg) 2005-04-30

Family

ID=23028846

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108075A BG108075A (bg) 2001-02-20 2003-08-07 Използване на производни на епотилон за лечение на трудно лечими тумори

Country Status (18)

Country Link
US (2) US6686380B2 (ru)
EP (1) EP1385529A4 (ru)
JP (1) JP2004522774A (ru)
KR (1) KR20040025895A (ru)
CN (1) CN1774253A (ru)
BG (1) BG108075A (ru)
BR (1) BR0207487A (ru)
CA (1) CA2438610A1 (ru)
EE (1) EE200300396A (ru)
HU (1) HUP0303175A2 (ru)
IL (1) IL156988A0 (ru)
IS (1) IS6918A (ru)
MX (1) MXPA03007394A (ru)
NO (1) NO20033684L (ru)
PL (1) PL363362A1 (ru)
RU (1) RU2003128311A (ru)
WO (1) WO2002066038A1 (ru)
ZA (1) ZA200306173B (ru)

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US7649006B2 (en) 2002-08-23 2010-01-19 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
US6921769B2 (en) 2002-08-23 2005-07-26 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
SI1767535T1 (sl) * 2002-08-23 2010-03-31 Sloan Kettering Inst Cancer Sinteza epotilonov njihovih intermediatov analogov in uporaba le teh
WO2004032866A2 (en) 2002-10-09 2004-04-22 Kosan Biosciences, Inc. Therapeutic formulations
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US20050171167A1 (en) * 2003-11-04 2005-08-04 Haby Thomas A. Process and formulation containing epothilones and analogs thereof
US20090004277A1 (en) * 2004-05-18 2009-01-01 Franchini Miriam K Nanoparticle dispersion containing lactam compound
WO2006017761A2 (en) * 2004-08-05 2006-02-16 Emory University Epothilone analogues as therapeutic agents
ES2306278T3 (es) 2004-11-18 2008-11-01 Bristol-Myers Squibb Company Perla enterica recubierta que comprende ixabepilona.
US20060134214A1 (en) * 2004-11-18 2006-06-22 Ismat Ullah Enteric coated bead comprising epothilone or epothilone analog, and preparation and administration thereof
EP1856255A4 (en) 2005-02-11 2010-01-27 Univ Southern California METHODS OF EXPRESSING PROTEINS WITH DISULFIDE BRIDGES
WO2007130501A2 (en) * 2006-05-01 2007-11-15 University Of Southern California Combination therapy for treatment of cancer
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WO2010056901A2 (en) 2008-11-13 2010-05-20 University Of Southern California Method of expressing proteins with disulfide bridges with enhanced yields and activity
EA035193B1 (ru) 2010-05-18 2020-05-14 Серулин Фарма Инк. Композиции и способы лечения аутоиммунных и других заболеваний
WO2021142202A1 (en) 2020-01-10 2021-07-15 R-Pharm Us Operating Llc Compositions of ixabepilone

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Also Published As

Publication number Publication date
RU2003128311A (ru) 2005-03-10
US20020165258A1 (en) 2002-11-07
PL363362A1 (en) 2004-11-15
MXPA03007394A (es) 2003-12-04
CN1774253A (zh) 2006-05-17
HUP0303175A2 (hu) 2003-12-29
BR0207487A (pt) 2004-08-10
JP2004522774A (ja) 2004-07-29
IL156988A0 (en) 2004-02-08
USRE41393E1 (en) 2010-06-22
EP1385529A4 (en) 2007-05-09
NO20033684D0 (no) 2003-08-19
KR20040025895A (ko) 2004-03-26
CA2438610A1 (en) 2002-08-29
IS6918A (is) 2003-08-18
US6686380B2 (en) 2004-02-03
NO20033684L (no) 2003-10-13
ZA200306173B (en) 2004-11-23
WO2002066038A1 (en) 2002-08-29
EE200300396A (et) 2003-12-15
EP1385529A1 (en) 2004-02-04

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