BG106727A - Производни на хигромицин - Google Patents

Производни на хигромицин Download PDF

Info

Publication number
BG106727A
BG106727A BG106727A BG10672702A BG106727A BG 106727 A BG106727 A BG 106727A BG 106727 A BG106727 A BG 106727A BG 10672702 A BG10672702 A BG 10672702A BG 106727 A BG106727 A BG 106727A
Authority
BG
Bulgaria
Prior art keywords
alkyl
groups
aryl
independently
hydroxy
Prior art date
Application number
BG106727A
Other languages
Bulgarian (bg)
English (en)
Inventor
Katherine BRIGHTY
Robert LINDE
Matthew Hayward
Takushi Kaneko
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG106727A publication Critical patent/BG106727A/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26Acyclic or carbocyclic radicals, substituted by hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BG106727A 1999-10-29 2002-05-20 Производни на хигромицин BG106727A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16258199P 1999-10-29 1999-10-29
PCT/IB2000/001461 WO2001030795A1 (en) 1999-10-29 2000-10-09 Hygromycin derivatives

Publications (1)

Publication Number Publication Date
BG106727A true BG106727A (bg) 2003-01-31

Family

ID=22586256

Family Applications (1)

Application Number Title Priority Date Filing Date
BG106727A BG106727A (bg) 1999-10-29 2002-05-20 Производни на хигромицин

Country Status (32)

Country Link
US (1) US6562792B1 (pt)
EP (1) EP1224197A1 (pt)
JP (1) JP2003512473A (pt)
KR (1) KR20020063885A (pt)
CN (1) CN1382150A (pt)
AP (1) AP2002002494A0 (pt)
AR (1) AR023282A1 (pt)
AU (1) AU7549400A (pt)
BG (1) BG106727A (pt)
BR (1) BR0015153A (pt)
CA (1) CA2389191A1 (pt)
CO (1) CO5261498A1 (pt)
CZ (1) CZ20021355A3 (pt)
EA (1) EA200200292A1 (pt)
EE (1) EE200200228A (pt)
GT (1) GT200000185A (pt)
HK (1) HK1049672A1 (pt)
HU (1) HUP0203525A3 (pt)
IL (1) IL148577A0 (pt)
IS (1) IS6311A (pt)
MA (1) MA26838A1 (pt)
MX (1) MXPA02004360A (pt)
NO (1) NO20021850L (pt)
OA (1) OA12081A (pt)
PA (1) PA8505801A1 (pt)
PE (1) PE20010763A1 (pt)
PL (1) PL357083A1 (pt)
SK (1) SK5472002A3 (pt)
SV (1) SV2002000211A (pt)
TN (1) TNSN00211A1 (pt)
TR (1) TR200201145T2 (pt)
WO (1) WO2001030795A1 (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EE200200671A (et) 2000-06-02 2004-08-16 Pfizer Products Inc. Hügromütsiin A derivaadid bakteriaalsete ja algloomadest põhjustatud infektsioonide ravimiseks
US6653481B2 (en) * 2000-12-29 2003-11-25 Synthon Bv Process for making amlodipine
US7923439B2 (en) * 2008-10-15 2011-04-12 Tyco Healthcare Group Lp Hydroxamate compositions
US20210275559A1 (en) * 2018-08-20 2021-09-09 Kim Lewis Hygromycin a compounds and methods of treating spirochete diseases
TW202128675A (zh) 2019-12-06 2021-08-01 美商維泰克斯製藥公司 作為鈉通道調節劑之經取代四氫呋喃
PE20241335A1 (es) 2021-06-04 2024-07-03 Vertex Pharma N-(hidroxialquil (hetero)aril) tetrahidrofurano carboxamidas como moduladores de canales de sodio

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100418167B1 (ko) * 1998-12-02 2004-02-11 화이자 프로덕츠 인크. 항균제로서의 하이그로마이신 a 유도체

Also Published As

Publication number Publication date
WO2001030795A1 (en) 2001-05-03
PA8505801A1 (es) 2002-08-26
KR20020063885A (ko) 2002-08-05
HUP0203525A3 (en) 2003-08-28
AR023282A1 (es) 2002-09-04
IL148577A0 (en) 2002-09-12
CO5261498A1 (es) 2003-03-31
US6562792B1 (en) 2003-05-13
SK5472002A3 (en) 2003-02-04
GT200000185A (es) 2002-04-18
TR200201145T2 (tr) 2002-09-23
CN1382150A (zh) 2002-11-27
NO20021850D0 (no) 2002-04-19
CA2389191A1 (en) 2001-05-03
SV2002000211A (es) 2002-07-16
AP2002002494A0 (en) 2002-06-30
IS6311A (is) 2002-03-19
PL357083A1 (en) 2004-07-12
EA200200292A1 (ru) 2002-10-31
JP2003512473A (ja) 2003-04-02
MA26838A1 (fr) 2004-12-20
EP1224197A1 (en) 2002-07-24
AU7549400A (en) 2001-05-08
PE20010763A1 (es) 2001-07-25
TNSN00211A1 (fr) 2005-11-10
EE200200228A (et) 2003-06-16
MXPA02004360A (es) 2002-11-07
HUP0203525A2 (hu) 2003-02-28
CZ20021355A3 (cs) 2002-11-13
NO20021850L (no) 2002-04-19
BR0015153A (pt) 2002-07-16
OA12081A (en) 2006-05-04
HK1049672A1 (zh) 2003-05-23

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