BG104256A - Лекарствен препарат с контролирано освобождаване на активно съединение - Google Patents

Лекарствен препарат с контролирано освобождаване на активно съединение

Info

Publication number
BG104256A
BG104256A BG104256A BG10425600A BG104256A BG 104256 A BG104256 A BG 104256A BG 104256 A BG104256 A BG 104256A BG 10425600 A BG10425600 A BG 10425600A BG 104256 A BG104256 A BG 104256A
Authority
BG
Bulgaria
Prior art keywords
medicamentous
preparation
active compound
controlled release
cycloprpopyl
Prior art date
Application number
BG104256A
Other languages
English (en)
Other versions
BG64745B1 (bg
Inventor
Hans-Martin Siefert
Patrick Bosche
Heino Stass
Stefan Kettelhoit
Tobias Laich
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of BG104256A publication Critical patent/BG104256A/bg
Publication of BG64745B1 publication Critical patent/BG64745B1/bg

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
BG104256A 1997-09-25 2000-03-20 Лекарствен препарат с контролирано освобождаване на активно съединение BG64745B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19742243 1997-09-25

Publications (2)

Publication Number Publication Date
BG104256A true BG104256A (bg) 2000-12-29
BG64745B1 BG64745B1 (bg) 2006-02-28

Family

ID=7843534

Family Applications (1)

Application Number Title Priority Date Filing Date
BG104256A BG64745B1 (bg) 1997-09-25 2000-03-20 Лекарствен препарат с контролирано освобождаване на активно съединение

Country Status (37)

Country Link
US (1) US6270799B1 (bg)
EP (1) EP1017392B1 (bg)
JP (2) JP2001517625A (bg)
KR (1) KR100531065B1 (bg)
CN (3) CN1895233A (bg)
AR (3) AR013967A1 (bg)
AT (1) ATE220547T1 (bg)
AU (1) AU731693B2 (bg)
BG (1) BG64745B1 (bg)
BR (1) BR9812553B1 (bg)
CA (1) CA2304135C (bg)
CO (1) CO5011082A1 (bg)
CZ (1) CZ293062B6 (bg)
DE (1) DE59804823D1 (bg)
DK (1) DK1017392T3 (bg)
ES (1) ES2179533T3 (bg)
GT (1) GT199800152A (bg)
HK (1) HK1032010A1 (bg)
HN (1) HN1998000144A (bg)
HU (1) HU226583B1 (bg)
ID (1) ID24259A (bg)
IL (1) IL134591A0 (bg)
MY (1) MY129437A (bg)
NO (1) NO327492B1 (bg)
NZ (1) NZ503538A (bg)
PE (1) PE20000224A1 (bg)
PL (1) PL192273B1 (bg)
PT (1) PT1017392E (bg)
SI (1) SI1017392T1 (bg)
SK (1) SK283462B6 (bg)
SV (1) SV1998000119A (bg)
TR (1) TR200000752T2 (bg)
TW (1) TW523412B (bg)
UA (1) UA66812C2 (bg)
UY (1) UY25192A1 (bg)
WO (1) WO1999015172A1 (bg)
ZA (1) ZA988718B (bg)

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AR020661A1 (es) * 1998-09-30 2002-05-22 Alcon Lab Inc Una composicion farmaceutica topica oftalmica, otica o nasal y el uso de la misma para la manufactura de un medicamento
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
DE10031043A1 (de) 2000-06-26 2002-02-14 Bayer Ag Retardzubereitungen von Chinolonantibiotika und Verfahren zu ihrer Herstellung
US20030091634A1 (en) * 2001-09-14 2003-05-15 Pawan Seth Delayed release tablet of venlafaxin
AU2002236132A1 (en) * 2002-03-05 2003-09-16 Ranbaxy Laboratories Limited Modified release oral pharmaceutical composition
ITMI20020515A1 (it) * 2002-03-12 2003-09-12 Jagotec Ag Sistema per il rilasco controllato di uno o piu' principi attivi
US7125563B2 (en) * 2002-04-12 2006-10-24 Dava Pharmaceuticals, Inc. Sustained release pharmaceutical preparations and methods for producing the same
US20050031683A1 (en) * 2003-08-04 2005-02-10 Ashish Kapoor Solid pharmaceutical composition
PL1691787T3 (pl) * 2003-12-04 2008-11-28 Pfizer Prod Inc Sposób wytwarzania farmaceutycznych systemów wielocząstkowych
GB2409204A (en) * 2003-12-19 2005-06-22 Reckitt Benckiser Nv Plasticized thermoplastic polymer
PT1868581E (pt) * 2005-04-11 2012-06-22 Abbott Lab Composições farmacêuticas que possuem perfis de dissolução melhorados para fármacos pouco solúveis
CN1762357B (zh) * 2005-09-21 2010-12-08 深圳市天一时科技开发有限公司 一种莫西沙星口服药物制剂及其制备方法
WO2007033522A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation de gélule contenant de la moxifloxacine et son procédé de préparation
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
EP2837376A3 (de) 2008-12-08 2015-03-25 ratiopharm GmbH Kompaktiertes Moxifloxacin
ITTO20110705A1 (it) * 2011-07-29 2013-01-30 Italiana Sint Spa Procedimento di preparazione della moxifloxacina cloridrato e relativi intermedi
KR20200077712A (ko) 2018-12-21 2020-07-01 한미약품 주식회사 목시플록사신 고형 제제 및 이의 제조방법

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US4207893A (en) 1977-08-29 1980-06-17 Alza Corporation Device using hydrophilic polymer for delivering drug to biological environment
FR2471186A1 (fr) * 1979-12-10 1981-06-19 Roussel Uclaf Nouveaux comprimes a delitescence colique, ainsi que leur procede de preparation
US4503030A (en) * 1983-06-06 1985-03-05 Alza Corporation Device for delivering drug to certain pH environments
CH668187A5 (de) 1986-08-07 1988-12-15 Ciba Geigy Ag Therapeutisches system mit systemischer wirkung.
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SE8704097D0 (sv) * 1987-10-22 1987-10-22 Astra Ab Oral formulation of buspirone and salts thereof
DE3906365A1 (de) * 1988-07-15 1990-01-18 Bayer Ag 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe
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Also Published As

Publication number Publication date
DE59804823D1 (de) 2002-08-22
PL192273B1 (pl) 2006-09-29
CO5011082A1 (es) 2001-02-28
HU226583B1 (hu) 2009-04-28
UY25192A1 (es) 2001-08-27
AU731693B2 (en) 2001-04-05
SK283462B6 (sk) 2003-08-05
CZ20001076A3 (cs) 2000-07-12
NO20001375L (no) 2000-03-16
CA2304135A1 (en) 1999-04-01
ZA988718B (en) 1999-04-01
HUP0003840A2 (hu) 2001-04-28
CN1178659C (zh) 2004-12-08
BR9812553A (pt) 2000-07-25
WO1999015172A1 (de) 1999-04-01
AU9348498A (en) 1999-04-12
ATE220547T1 (de) 2002-08-15
JP2010163455A (ja) 2010-07-29
NO20001375D0 (no) 2000-03-16
CN1271281A (zh) 2000-10-25
PT1017392E (pt) 2002-10-31
CZ293062B6 (cs) 2004-01-14
TR200000752T2 (tr) 2000-09-21
KR100531065B1 (ko) 2005-11-28
BG64745B1 (bg) 2006-02-28
GT199800152A (es) 2000-03-17
AR065072A2 (es) 2009-05-13
US6270799B1 (en) 2001-08-07
SI1017392T1 (en) 2002-12-31
DK1017392T3 (da) 2002-10-21
ES2179533T3 (es) 2003-01-16
BR9812553B1 (pt) 2010-06-01
CA2304135C (en) 2009-01-06
JP2001517625A (ja) 2001-10-09
SV1998000119A (es) 1999-03-02
CN1623533A (zh) 2005-06-08
MY129437A (en) 2007-04-30
PL339349A1 (en) 2000-12-18
KR20010024269A (ko) 2001-03-26
EP1017392B1 (de) 2002-07-17
HK1032010A1 (en) 2001-07-06
IL134591A0 (en) 2001-04-30
NO327492B1 (no) 2009-07-20
AR013967A1 (es) 2001-01-31
AR065073A2 (es) 2009-05-13
EP1017392A1 (de) 2000-07-12
TW523412B (en) 2003-03-11
SK4032000A3 (en) 2000-09-12
CN1895233A (zh) 2007-01-17
ID24259A (id) 2000-07-13
HUP0003840A3 (en) 2006-06-28
NZ503538A (en) 2001-03-30
HN1998000144A (es) 1999-06-02
PE20000224A1 (es) 2000-05-11
UA66812C2 (uk) 2004-06-15

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