UA66812C2 - Препаративна форма лікарського засобу із регульованим вивільненням активної речовини - Google Patents

Препаративна форма лікарського засобу із регульованим вивільненням активної речовини

Info

Publication number
UA66812C2
UA66812C2 UA2000042347A UA00042347A UA66812C2 UA 66812 C2 UA66812 C2 UA 66812C2 UA 2000042347 A UA2000042347 A UA 2000042347A UA 00042347 A UA00042347 A UA 00042347A UA 66812 C2 UA66812 C2 UA 66812C2
Authority
UA
Ukraine
Prior art keywords
active ingredient
controlled release
drug formulation
therefrom
medicament formulation
Prior art date
Application number
UA2000042347A
Other languages
English (en)
Russian (ru)
Inventor
Ханс-Мартін Зіферт
Патрік Боше
Патрик Боше
Хайно Штасс
Штефан Кеттельхоіт
Тобіас Лаіх
Original Assignee
Баєр Акцієнгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Баєр Акцієнгезельшафт filed Critical Баєр Акцієнгезельшафт
Publication of UA66812C2 publication Critical patent/UA66812C2/uk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Винахід стосується препаративних форм, які як активну речовину містять 1-циклопропіл-7-([S,S]-2,8-діазабіцикло[4.3.0]нон-8-іл)-6-фтор-1,4-дигідро-8-метоксі-4-оксо-3-хінолонкарбонову кислоту або її фармацевтичнo прийнятні солі та/або гідрати, які вивільняють активну речовину, що міститься в них, з певним режимом вивільнення.
UA2000042347A 1997-09-25 1998-09-15 Препаративна форма лікарського засобу із регульованим вивільненням активної речовини UA66812C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19742243 1997-09-25
PCT/EP1998/005842 WO1999015172A1 (de) 1997-09-25 1998-09-15 Arzneimittelformulierung mit kontrollierter wirkstofffreisetzung

Publications (1)

Publication Number Publication Date
UA66812C2 true UA66812C2 (uk) 2004-06-15

Family

ID=7843534

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2000042347A UA66812C2 (uk) 1997-09-25 1998-09-15 Препаративна форма лікарського засобу із регульованим вивільненням активної речовини

Country Status (37)

Country Link
US (1) US6270799B1 (uk)
EP (1) EP1017392B1 (uk)
JP (2) JP2001517625A (uk)
KR (1) KR100531065B1 (uk)
CN (3) CN1178659C (uk)
AR (3) AR013967A1 (uk)
AT (1) ATE220547T1 (uk)
AU (1) AU731693B2 (uk)
BG (1) BG64745B1 (uk)
BR (1) BR9812553B1 (uk)
CA (1) CA2304135C (uk)
CO (1) CO5011082A1 (uk)
CZ (1) CZ293062B6 (uk)
DE (1) DE59804823D1 (uk)
DK (1) DK1017392T3 (uk)
ES (1) ES2179533T3 (uk)
GT (1) GT199800152A (uk)
HK (1) HK1032010A1 (uk)
HN (1) HN1998000144A (uk)
HU (1) HU226583B1 (uk)
ID (1) ID24259A (uk)
IL (1) IL134591A0 (uk)
MY (1) MY129437A (uk)
NO (1) NO327492B1 (uk)
NZ (1) NZ503538A (uk)
PE (1) PE20000224A1 (uk)
PL (1) PL192273B1 (uk)
PT (1) PT1017392E (uk)
SI (1) SI1017392T1 (uk)
SK (1) SK283462B6 (uk)
SV (1) SV1998000119A (uk)
TR (1) TR200000752T2 (uk)
TW (1) TW523412B (uk)
UA (1) UA66812C2 (uk)
UY (1) UY25192A1 (uk)
WO (1) WO1999015172A1 (uk)
ZA (1) ZA988718B (uk)

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US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
AR020661A1 (es) * 1998-09-30 2002-05-22 Alcon Lab Inc Una composicion farmaceutica topica oftalmica, otica o nasal y el uso de la misma para la manufactura de un medicamento
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
DE10031043A1 (de) * 2000-06-26 2002-02-14 Bayer Ag Retardzubereitungen von Chinolonantibiotika und Verfahren zu ihrer Herstellung
US20030091634A1 (en) * 2001-09-14 2003-05-15 Pawan Seth Delayed release tablet of venlafaxin
CN1993109A (zh) * 2002-03-05 2007-07-04 兰贝克赛实验室有限公司 释放得到改良的口服药物组合物
ITMI20020515A1 (it) * 2002-03-12 2003-09-12 Jagotec Ag Sistema per il rilasco controllato di uno o piu' principi attivi
US7125563B2 (en) * 2002-04-12 2006-10-24 Dava Pharmaceuticals, Inc. Sustained release pharmaceutical preparations and methods for producing the same
US20050031683A1 (en) * 2003-08-04 2005-02-10 Ashish Kapoor Solid pharmaceutical composition
SI1691787T1 (sl) * 2003-12-04 2008-10-31 Pfizer Prod Inc Postopek za pripravo farmacevtskih produktov iz več delcev
GB2409204A (en) * 2003-12-19 2005-06-22 Reckitt Benckiser Nv Plasticized thermoplastic polymer
EP2286800A1 (en) * 2005-04-11 2011-02-23 Abbott Laboratories Pharmaceutical compositions having improved dissolution profiles for poorly soluble drugs
CN1762357B (zh) * 2005-09-21 2010-12-08 深圳市天一时科技开发有限公司 一种莫西沙星口服药物制剂及其制备方法
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
WO2007033522A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation de gélule contenant de la moxifloxacine et son procédé de préparation
EP2364141B2 (de) 2008-12-08 2017-08-02 ratiopharm GmbH Kompaktiertes moxifloxacin
ITTO20110705A1 (it) * 2011-07-29 2013-01-30 Italiana Sint Spa Procedimento di preparazione della moxifloxacina cloridrato e relativi intermedi
KR20200077712A (ko) 2018-12-21 2020-07-01 한미약품 주식회사 목시플록사신 고형 제제 및 이의 제조방법

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Also Published As

Publication number Publication date
EP1017392A1 (de) 2000-07-12
HUP0003840A3 (en) 2006-06-28
SV1998000119A (es) 1999-03-02
HUP0003840A2 (hu) 2001-04-28
CN1178659C (zh) 2004-12-08
NO20001375D0 (no) 2000-03-16
US6270799B1 (en) 2001-08-07
ID24259A (id) 2000-07-13
HN1998000144A (es) 1999-06-02
GT199800152A (es) 2000-03-17
UY25192A1 (es) 2001-08-27
CZ20001076A3 (cs) 2000-07-12
JP2001517625A (ja) 2001-10-09
NO327492B1 (no) 2009-07-20
TW523412B (en) 2003-03-11
HK1032010A1 (en) 2001-07-06
KR100531065B1 (ko) 2005-11-28
CZ293062B6 (cs) 2004-01-14
AU9348498A (en) 1999-04-12
AR013967A1 (es) 2001-01-31
CN1623533A (zh) 2005-06-08
BR9812553A (pt) 2000-07-25
AR065073A2 (es) 2009-05-13
CA2304135C (en) 2009-01-06
CA2304135A1 (en) 1999-04-01
PT1017392E (pt) 2002-10-31
SK4032000A3 (en) 2000-09-12
AU731693B2 (en) 2001-04-05
NZ503538A (en) 2001-03-30
HU226583B1 (hu) 2009-04-28
EP1017392B1 (de) 2002-07-17
DK1017392T3 (da) 2002-10-21
WO1999015172A1 (de) 1999-04-01
BR9812553B1 (pt) 2010-06-01
NO20001375L (no) 2000-03-16
PL192273B1 (pl) 2006-09-29
ATE220547T1 (de) 2002-08-15
DE59804823D1 (de) 2002-08-22
SK283462B6 (sk) 2003-08-05
AR065072A2 (es) 2009-05-13
ZA988718B (en) 1999-04-01
TR200000752T2 (tr) 2000-09-21
SI1017392T1 (en) 2002-12-31
KR20010024269A (ko) 2001-03-26
CO5011082A1 (es) 2001-02-28
CN1895233A (zh) 2007-01-17
IL134591A0 (en) 2001-04-30
BG64745B1 (bg) 2006-02-28
PE20000224A1 (es) 2000-05-11
MY129437A (en) 2007-04-30
PL339349A1 (en) 2000-12-18
ES2179533T3 (es) 2003-01-16
BG104256A (en) 2000-12-29
CN1271281A (zh) 2000-10-25
JP2010163455A (ja) 2010-07-29

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