BE849647A - Esters et amides des acides pyrimido (4,5-b) quinolein-4(3h)-one-2-carboxyliques, en tant qu'agents antiulceres - Google Patents
Esters et amides des acides pyrimido (4,5-b) quinolein-4(3h)-one-2-carboxyliques, en tant qu'agents antiulceresInfo
- Publication number
- BE849647A BE849647A BE1007837A BE1007837A BE849647A BE 849647 A BE849647 A BE 849647A BE 1007837 A BE1007837 A BE 1007837A BE 1007837 A BE1007837 A BE 1007837A BE 849647 A BE849647 A BE 849647A
- Authority
- BE
- Belgium
- Prior art keywords
- quinolein
- amids
- pyrimido
- esters
- carboxylic acids
- Prior art date
Links
- 239000003699 antiulcer agent Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/650,714 US4011324A (en) | 1976-01-20 | 1976-01-20 | Esters and amides of pyrimido[4,5-b]quinolin-4(3H)-one-2-carboxylic acids as antiulcer agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BE849647A true BE849647A (fr) | 1977-06-20 |
Family
ID=24609991
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE1007837A BE849647A (fr) | 1976-01-20 | 1976-12-20 | Esters et amides des acides pyrimido (4,5-b) quinolein-4(3h)-one-2-carboxyliques, en tant qu'agents antiulceres |
Country Status (10)
Country | Link |
---|---|
US (1) | US4011324A (da) |
JP (2) | JPS5289700A (da) |
BE (1) | BE849647A (da) |
DE (1) | DE2700216A1 (da) |
DK (1) | DK575776A (da) |
FR (1) | FR2361892A1 (da) |
GB (1) | GB1531681A (da) |
IE (1) | IE43964B1 (da) |
LU (1) | LU76457A1 (da) |
NL (1) | NL168515C (da) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2757915A1 (de) * | 1976-12-28 | 1978-07-06 | Mitsubishi Yuka Pharma | Pyrimidochinoxalinderivate, verfahren zur herstellung derselben und arzneimittel zur behandlung von allergischem asthma |
DE3138550A1 (de) * | 1981-09-28 | 1983-04-07 | Boehringer Ingelheim KG, 6507 Ingelheim | Substituierte 2-phenyl-2-(pyridyloxy)-ethylamine und isostere verbindungen, verfahren zu ihrer herstellung und verwendung |
US4551460A (en) * | 1982-05-10 | 1985-11-05 | Hoffmann-La Roche Inc. | Pyrido[2,1-b]quinazoline derivatives useful as agents for treatment of allergic conditions and vascular disorders involving thrombosis |
DE3232620A1 (de) * | 1982-09-02 | 1984-03-08 | Hoechst Ag, 6230 Frankfurt | 10-phenyl1-1,3,9-triazaanthracene und diese enthaltendes photopolymerisierbares gemisch |
US6545004B1 (en) | 1999-10-27 | 2003-04-08 | Cytokinetics, Inc. | Methods and compositions utilizing quinazolinones |
US7230000B1 (en) | 1999-10-27 | 2007-06-12 | Cytokinetics, Incorporated | Methods and compositions utilizing quinazolinones |
WO2002094790A1 (fr) * | 2001-05-23 | 2002-11-28 | Mitsubishi Pharma Corporation | Compose heterocyclique condense et son utilisation medicale |
ITMI20012060A1 (it) * | 2001-10-05 | 2003-04-05 | Recordati Chem Pharm | Nuovi eterocilcli n-acilati |
US7009049B2 (en) * | 2002-02-15 | 2006-03-07 | Cytokinetics, Inc. | Syntheses of quinazolinones |
JP2006508030A (ja) * | 2002-05-09 | 2006-03-09 | サイトキネティクス・インコーポレーテッド | ピリミジノン化合物、組成物および方法 |
WO2003097053A1 (en) | 2002-05-09 | 2003-11-27 | Cytokinetics, Inc. | Compounds, compositions, and methods |
WO2003103575A2 (en) * | 2002-05-23 | 2003-12-18 | Cytokinetics, Inc. | Compounds, compositions, and methods |
US7041676B2 (en) * | 2002-06-14 | 2006-05-09 | Cytokinetics, Inc. | Compounds, compositions, and methods |
EP1537089A4 (en) * | 2002-07-23 | 2008-04-16 | Cytokinetics Inc | CONNECTIONS, COMPOSITIONS AND PROCEDURES |
JP2005536553A (ja) * | 2002-08-21 | 2005-12-02 | サイトキネティクス・インコーポレーテッド | 化合物、組成物および方法 |
US7557115B2 (en) * | 2002-09-30 | 2009-07-07 | Cytokinetics, Inc. | Compounds, compositions, and methods |
EP1682534A2 (en) * | 2003-11-03 | 2006-07-26 | Cytokinetics, Inc. | Pyrimidin-4-one compounds, compositions, and methods |
US20050148593A1 (en) * | 2003-11-07 | 2005-07-07 | Gustave Bergnes | Compounds, compositions, and methods |
EP1692112A4 (en) * | 2003-12-08 | 2008-09-24 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS, AND METHODS |
EP1740551B9 (en) * | 2004-04-30 | 2013-01-16 | Takeda Pharmaceutical Company Limited | Heterocyclic amide compound and use thereof as an mmp-13 inhibitor |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3414574A (en) * | 1967-04-21 | 1968-12-03 | Sandoz Ag | Certain pyrimido (4, 5-b) indoles and intermediates employed in their preparation |
US3974161A (en) * | 1974-02-20 | 1976-08-10 | Pfizer Inc. | Fused pyrimidin-4(3H)-ones as antiallergy agents |
GB1458205A (en) * | 1973-04-13 | 1976-12-08 | Pfizer | Fused pyrimidin-4- 3h-ones as antiallergy agents |
-
1976
- 1976-01-20 US US05/650,714 patent/US4011324A/en not_active Expired - Lifetime
- 1976-10-21 IE IE2318/76A patent/IE43964B1/en unknown
- 1976-12-20 BE BE1007837A patent/BE849647A/xx unknown
- 1976-12-21 DK DK575776A patent/DK575776A/da not_active Application Discontinuation
- 1976-12-21 FR FR7638523A patent/FR2361892A1/fr active Granted
- 1976-12-21 NL NLAANVRAGE7614191,A patent/NL168515C/xx not_active IP Right Cessation
- 1976-12-22 LU LU76457A patent/LU76457A1/xx unknown
- 1976-12-22 JP JP15479776A patent/JPS5289700A/ja active Pending
-
1977
- 1977-01-05 DE DE19772700216 patent/DE2700216A1/de active Pending
- 1977-01-12 GB GB1181/77A patent/GB1531681A/en not_active Expired
-
1978
- 1978-09-25 JP JP11781478A patent/JPS5470433A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
FR2361892A1 (fr) | 1978-03-17 |
DK575776A (da) | 1977-07-21 |
IE43964B1 (en) | 1981-07-15 |
NL7614191A (nl) | 1977-07-22 |
JPS5470433A (en) | 1979-06-06 |
US4011324A (en) | 1977-03-08 |
FR2361892B1 (da) | 1980-09-19 |
IE43964L (en) | 1977-07-20 |
JPS5289700A (en) | 1977-07-27 |
GB1531681A (en) | 1978-11-08 |
LU76457A1 (da) | 1977-07-05 |
NL168515B (nl) | 1981-11-16 |
DE2700216A1 (de) | 1977-07-28 |
NL168515C (nl) | 1982-04-16 |
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