BE794597A - Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation - Google Patents
Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparationInfo
- Publication number
- BE794597A BE794597A BE794597DA BE794597A BE 794597 A BE794597 A BE 794597A BE 794597D A BE794597D A BE 794597DA BE 794597 A BE794597 A BE 794597A
- Authority
- BE
- Belgium
- Prior art keywords
- piperidinoalcanols
- aryl
- substituted
- preparation process
- piperidino group
- Prior art date
Links
- -1 PIPERIDINO GROUP Chemical group 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22182172A | 1972-01-28 | 1972-01-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE794597A true BE794597A (fr) | 1973-05-16 |
Family
ID=22829539
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE794597D BE794597A (fr) | 1972-01-28 | 1973-01-26 | Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation |
Country Status (26)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3941795A (en) | 1974-02-08 | 1976-03-02 | Richardson-Merrell Inc. | α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4254129A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| US4254130A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| IT1200123B (it) * | 1985-09-27 | 1989-01-05 | Ind Chimica Srl | Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo |
| US4742175A (en) * | 1986-05-07 | 1988-05-03 | Merrell Dow Pharmaceuticals Inc. | Preparation of polymorphically pure terfenadine |
| JPS63101760U (enrdf_load_stackoverflow) * | 1986-12-19 | 1988-07-02 | ||
| IT1205685B (it) * | 1987-05-26 | 1989-03-31 | Erregierre Spa | Processo per la preparazione di alfa-(alchilfenil)-4-(idrossi difenilmetil)-1-piperidina butanolo |
| ZA901360B (en) * | 1989-02-28 | 1990-11-28 | Merrell Dow Pharma | Preparation of the low-melting polymorphic form of terfenadine |
| ZA903145B (en) * | 1989-05-01 | 1991-02-27 | Merrell Dow Pharma | Process for the preparation of the high melting polymorphic form of terfenadine |
| DE3917241A1 (de) * | 1989-05-26 | 1990-11-29 | Schaper & Bruemmer Gmbh | 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate |
| US5466691A (en) * | 1991-08-09 | 1995-11-14 | Yoshitomi Pharmaceutical Industries, Ltd. | Thiophene compound |
| CN1183769A (zh) * | 1995-05-08 | 1998-06-03 | 赫彻斯特马里恩鲁斯公司 | α-(取代的烷基苯基)-4-(羟基二苯基甲基)-1-哌啶丁醇衍生物,其制备和其用作抗组胺剂、抗变应性剂和支气管扩张药的用途 |
| ATE260983T1 (de) * | 1997-03-11 | 2004-03-15 | Aventis Pharma Inc | Verfahren zur herstellung von 4-(4-(4- (hydroxydiphenyl)-1-piperidinyl)-1-hydroxybutyl - alpha,alpha-dimenthylphenylessigsäure und phosphorylierter derivate |
| US7498345B2 (en) * | 2004-09-17 | 2009-03-03 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| US8153385B2 (en) | 2004-10-18 | 2012-04-10 | Reverse Proteomics Research Institute Co., Ltd. | Target protein and target gene in drug designing and screening method |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3081303A (en) * | 1961-10-13 | 1963-03-12 | Searle & Co | 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols |
| GB1242169A (en) * | 1969-04-09 | 1971-08-11 | Ucb Sa | Piperidine derivatives |
-
1972
- 1972-12-04 ZA ZA728544A patent/ZA728544B/xx unknown
- 1972-12-05 IE IE1689/72A patent/IE36983B1/xx unknown
- 1972-12-08 PH PH14156A patent/PH10264A/en unknown
- 1972-12-11 AU AU49893/72A patent/AU467361B2/en not_active Ceased
- 1972-12-12 IL IL41060A patent/IL41060A/xx unknown
- 1972-12-15 GB GB5799572A patent/GB1413138A/en not_active Expired
- 1972-12-20 CH CH1854272A patent/CH587820A5/xx not_active IP Right Cessation
- 1972-12-20 CH CH1381476A patent/CH593259A5/xx not_active IP Right Cessation
- 1972-12-27 JP JP47130136A patent/JPS5115035B2/ja not_active Expired
- 1972-12-29 AT AT246074*1A patent/AT323742B/de not_active IP Right Cessation
- 1972-12-29 AT AT1115372A patent/AT321917B/de not_active IP Right Cessation
-
1973
- 1973-01-08 YU YU34/73A patent/YU36013B/xx unknown
- 1973-01-16 CA CA161,413A patent/CA978946A/en not_active Expired
- 1973-01-17 HU HURI498A patent/HU166477B/hu unknown
- 1973-01-18 ES ES410731A patent/ES410731A1/es not_active Expired
- 1973-01-22 NL NLAANVRAGE7300873,A patent/NL175410C/xx not_active IP Right Cessation
- 1973-01-24 SE SE7300974A patent/SE382058B/xx active Protection Beyond IP Right Term
- 1973-01-24 DE DE2303306A patent/DE2303306C3/de not_active Expired
- 1973-01-24 FR FR7302503A patent/FR2181690B1/fr not_active Expired
- 1973-01-25 DD DD168482A patent/DD103239A5/xx unknown
- 1973-01-26 AR AR246313A patent/AR195314A1/es active
- 1973-01-26 LU LU66916A patent/LU66916A1/xx unknown
- 1973-01-26 DK DK44973AA patent/DK136713B/da not_active IP Right Cessation
- 1973-01-26 PL PL1973160419A patent/PL89095B1/pl unknown
- 1973-01-26 BE BE794597D patent/BE794597A/xx not_active IP Right Cessation
- 1973-01-26 NO NO326/73A patent/NO140057C/no unknown
- 1973-01-26 CS CS630A patent/CS177834B2/cs unknown
- 1973-01-27 SU SU1878074A patent/SU464997A3/ru active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3941795A (en) | 1974-02-08 | 1976-03-02 | Richardson-Merrell Inc. | α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES |
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BE764179A (fr) | " 5-azapyrimidine-nucleosides et leur procede de preparation | |
| BE794598A (fr) | Nouveaux derives olefiniques de piperidines substituees en 4 et leur procede de preparation | |
| BE794669A (fr) | Derives de 3,4-dihydrocarbostyryle et leur procede de preparation | |
| BE825302R (fr) | Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation | |
| BE794597A (fr) | Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation | |
| FR2279744A1 (fr) | Nouveaux composes du type g-lactones et g-lactols et leur procede de preparation | |
| BE794596A (fr) | Piperidinoalcanone-oximes substituees et leur procede de preparation | |
| BE793955A (fr) | Arylpiperazines et leur procede de preparation | |
| BE798059A (fr) | Derives de chromone et leur procede de preparation | |
| BE788050A (fr) | Nouveaux derives de propenylamine et leur procede de preparation | |
| BE807988A (fr) | Nouveaux 2 beta 16 beta-diamino-androstanes et procede pour leur preparation | |
| BE795705A (fr) | Procede de preparation de polyfluoroalcools et leur application | |
| BE814117A (fr) | Aza-2 cycloalkylmethylcetones et leur procede de preparation | |
| BE800830A (fr) | Nouveaux derives d'anilide et leur procede de preparation | |
| BE814118A (fr) | Phenylmethanols et phenylcetones aza-2 cycloalkylmethyl-substitues et leur procede de preparation | |
| BE802336A (fr) | Nouveaux hydroxy-aminosteroides et procede pour leur preparation | |
| BE793252A (fr) | Nouveaux derives de dicycloalkane et leur procede de preparation | |
| BE801315A (fr) | 4-mercapto-azetidinones-(2) et leur procede de preparation | |
| BE807803A (fr) | Nouveaux triazolyl-stilbenes et leur procede de preparation | |
| BE808985A (fr) | Nouveaux derives d'acide de pregnane, et leur procede de preparation | |
| BE751923A (fr) | Nouveaux aminoaryl-ethers et leur procede de preparation | |
| BE801720A (fr) | Derives de benzomorphane et leur procede de preparation | |
| BE799339A (fr) | Nouvelles 2-benzoyl-3-amino-pyridines et leur procede de preparation | |
| BE800121A (fr) | Nouveaux triazolyl-naphtalimides et leur procede de preparation, | |
| BE798165A (fr) | Nouveaux copolymeres et leur procede de preparation |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE20 | Patent expired |
Owner name: MERRELL DOW PHARMACEUTICALS INC. Effective date: 19930126 |