BE783440A - Derives de benzofuranne et leur preparation - Google Patents

Derives de benzofuranne et leur preparation

Info

Publication number
BE783440A
BE783440A BE783440A BE783440A BE783440A BE 783440 A BE783440 A BE 783440A BE 783440 A BE783440 A BE 783440A BE 783440 A BE783440 A BE 783440A BE 783440 A BE783440 A BE 783440A
Authority
BE
Belgium
Prior art keywords
preparation
benzofuran derivatives
benzofuran
derivatives
Prior art date
Application number
BE783440A
Other languages
English (en)
French (fr)
Original Assignee
Kakenyaku Kako Cy Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP5233371A external-priority patent/JPS5020062B1/ja
Priority claimed from JP8610971A external-priority patent/JPS5020063B2/ja
Priority claimed from JP439572A external-priority patent/JPS5529993B2/ja
Application filed by Kakenyaku Kako Cy Ltd filed Critical Kakenyaku Kako Cy Ltd
Publication of BE783440A publication Critical patent/BE783440A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/80Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/81Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/86Benzo [b] furans; Hydrogenated benzo [b] furans with an oxygen atom directly attached in position 7

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE783440A 1971-05-13 1972-05-12 Derives de benzofuranne et leur preparation BE783440A (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP3214571 1971-05-13
JP5233371A JPS5020062B1 (es) 1971-07-14 1971-07-14
JP8610971A JPS5020063B2 (es) 1971-10-28 1971-10-28
JP439572A JPS5529993B2 (es) 1972-01-06 1972-01-06

Publications (1)

Publication Number Publication Date
BE783440A true BE783440A (fr) 1972-09-01

Family

ID=27454077

Family Applications (1)

Application Number Title Priority Date Filing Date
BE783440A BE783440A (fr) 1971-05-13 1972-05-12 Derives de benzofuranne et leur preparation

Country Status (8)

Country Link
US (1) US3853923A (es)
BE (1) BE783440A (es)
CA (1) CA989411A (es)
CH (1) CH587261A5 (es)
DE (1) DE2223184C3 (es)
FR (1) FR2137901B1 (es)
GB (1) GB1380129A (es)
NL (1) NL166939C (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2457866A1 (fr) * 1979-05-29 1980-12-26 Anvar Nouveaux derives des cyano-2 hydroxy-3 benzofuranne et benzo(b) thiophene, leur preparation et leur application en therapeutique
JPS5639015A (en) * 1979-09-06 1981-04-14 Kaken Pharmaceut Co Ltd Ophthalmic solution for regulating intraocular tension
FR2515649A1 (fr) * 1981-10-30 1983-05-06 Debat Lab Nouveaux derives appartenant a la famille des 3-amino-1-heteroaryloxy-2-propanols, utilisation en therapeutique et procede de preparation
JPS58157784A (ja) * 1982-03-16 1983-09-19 Kaken Pharmaceut Co Ltd 光学活性な〔s〕−(+)−2−アセチル−7−(2,3−エポキシプロポキシ)ベンゾフランの製造法
JPS60202872A (ja) * 1984-03-27 1985-10-14 Kaken Pharmaceut Co Ltd ベンゾフラン誘導体、その製法およびそれを有効成分とする降圧剤
KR920000799B1 (ko) * 1987-12-11 1992-01-23 미쓰이 세끼유 가가꾸 고오교오 가부시끼가이샤 신규아민류 및 그 용도
TR200101779T2 (tr) 1998-12-18 2001-12-21 Basilea Pharmaceutica Ag Yeni bisiklik bileşenler
GEP20074134B (en) 2002-08-19 2007-06-25 Pfizer Prod Inc Combination therapy for hyperproliferative diseases
GT200600381A (es) 2005-08-25 2007-03-28 Compuestos organicos
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
ATE547394T1 (de) 2006-12-01 2012-03-15 Bristol Myers Squibb Co N-((3-benzyl)-2,2-(bis-phenyl)-propan-1- aminderivate als cetp-hemmer für die behandlung von atherosklerose und herz-kreislauf- erkrankungen
JP5844376B2 (ja) 2010-10-06 2016-01-13 ジェイファーマ株式会社 強力な尿酸トランスポーター阻害剤の開発:それらの尿酸排泄効果のために設計された化合物
SG11201507496UA (en) 2013-04-17 2015-11-27 Pfizer N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
CN107827849B (zh) * 2017-11-14 2020-06-02 沈阳药科大学 6-[2-羟基-3-(烷胺基)丙氧基]苯并呋喃类化合物及其应用
CN107857748B (zh) * 2017-11-14 2020-06-02 沈阳药科大学 5-[2-羟基-3-(烷胺基)丙氧基]苯并呋喃类化合物及其应用
CN107935972B (zh) * 2017-11-14 2020-06-02 沈阳药科大学 5-[2-羟基-3-(异丙胺基)丙氧基]苯并呋喃类衍生物及其应用
SG11202107614PA (en) 2019-01-18 2021-08-30 Astrazeneca Ab Pcsk9 inhibitors and methods of use thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1058822A (en) * 1963-07-30 1967-02-15 Ici Ltd 3-amino-2-hydroxypropoxy heterocyclic derivatives

Also Published As

Publication number Publication date
DE2223184C3 (de) 1980-04-30
DE2223184A1 (de) 1972-11-23
US3853923A (en) 1974-12-10
DE2223184B2 (de) 1979-08-16
NL166939B (nl) 1981-05-15
NL166939C (nl) 1981-10-15
CH587261A5 (es) 1977-04-29
FR2137901B1 (es) 1975-10-31
FR2137901A1 (es) 1972-12-29
CA989411A (en) 1976-05-18
GB1380129A (en) 1975-01-08
NL7206433A (es) 1972-11-15

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Legal Events

Date Code Title Description
RE20 Patent expired

Owner name: KAKENYAKU KAKO CO. LTD

Effective date: 19920512