BE747492A - Nouveaux steroides physiologiquement actifs, et leur procede defabrication - Google Patents
Nouveaux steroides physiologiquement actifs, et leur procede defabricationInfo
- Publication number
- BE747492A BE747492A BE747492DA BE747492A BE 747492 A BE747492 A BE 747492A BE 747492D A BE747492D A BE 747492DA BE 747492 A BE747492 A BE 747492A
- Authority
- BE
- Belgium
- Prior art keywords
- manufacturing process
- physiologically active
- active steroids
- new physiologically
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/14—All rings being cycloaliphatic
- C07C2602/24—All rings being cycloaliphatic the ring system containing nine carbon atoms, e.g. perhydroindane
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
- Physical Or Chemical Processes And Apparatus (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US00807929A US3833622A (en) | 1969-03-17 | 1969-03-17 | Crystalline 25-hydroxycholecalciferol hydrate and structurally related compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BE747492A true BE747492A (fr) | 1970-09-17 |
Family
ID=25197461
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE747492D BE747492A (fr) | 1969-03-17 | 1970-03-17 | Nouveaux steroides physiologiquement actifs, et leur procede defabrication |
Country Status (10)
Country | Link |
---|---|
US (1) | US3833622A (fr) |
JP (1) | JPS4934980B1 (fr) |
BE (1) | BE747492A (fr) |
CA (1) | CA968789A (fr) |
CH (1) | CH528500A (fr) |
DE (1) | DE2012167C2 (fr) |
FR (1) | FR2035000B1 (fr) |
GB (1) | GB1286761A (fr) |
IL (1) | IL33860A (fr) |
NL (1) | NL7003686A (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2571369A1 (fr) * | 1984-10-04 | 1986-04-11 | Wisconsin Alumni Res Found | Derives de la vitamine d et precurseurs de ceux-ci et compositions pharmaceutiques en contenant |
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4012509A (en) * | 1974-06-10 | 1977-03-15 | The Upjohn Company | Composition of matter and process |
US3907843A (en) * | 1974-06-14 | 1975-09-23 | Wisconsin Alumni Res Found | 1{60 -Hydroxyergocalciferol and processes for preparing same |
US3906014A (en) * | 1974-06-17 | 1975-09-16 | Wisconsin Alumni Res Found | 3-Deoxy-1{60 -hydroxycholecalciferol |
US4001096A (en) * | 1975-02-21 | 1977-01-04 | The Upjohn Company | Process for preparing 25-hydroxycholecalciferol intermediates |
US3993675A (en) * | 1975-02-24 | 1976-11-23 | Hoffmann-La Roche Inc. | Process for the preparation of 1α,25-dihydroxycholecalciferol |
US4069321A (en) * | 1975-10-14 | 1978-01-17 | Merck & Co., Inc. | Blocked cholecalciferol and dihydrotachysterol 3 derivatives |
JPS603045B2 (ja) * | 1976-04-19 | 1985-01-25 | 中外製薬株式会社 | 1α―ヒドロキシビタミンD類軟カプセルの製造方法 |
USRE30538E (en) * | 1977-03-07 | 1981-03-03 | Wisconsin Alumni Research Foundation | 3-Deoxy-1α-hydroxycholecalciferol |
US4217288A (en) * | 1977-03-24 | 1980-08-12 | Wisconsin Alumni Research Foundation | Anti-vitamin D compounds |
US4119647A (en) * | 1977-04-11 | 1978-10-10 | Hoffmann-La Roche Inc. | 25-Hydroxycholecalciferol-23,24-3 H and process for the preparation thereof |
JPS6039278B2 (ja) * | 1977-05-23 | 1985-09-05 | 中外製薬株式会社 | ステロイド誘導体 |
US4183852A (en) * | 1977-07-18 | 1980-01-15 | Kaiser Emil T | Process for preparing 25-hydroxycholesterol |
JPS5822479B2 (ja) * | 1977-09-07 | 1983-05-09 | 帝人株式会社 | 1α−ヒドロキシ−24−オキソ−ビタミンD↓3およびその製造法 |
US4188345A (en) * | 1978-07-26 | 1980-02-12 | Wisconsin Alumni Research Foundation | Fluorovitamin D compounds and processes for their preparation |
US4225596A (en) * | 1978-10-13 | 1980-09-30 | Wisconsin Alumni Research Foundation | Method for treating calcium imbalance and improving calcium absorption in mammals |
US4269777A (en) * | 1979-05-21 | 1981-05-26 | Wisconsin Alumni Research Foundation | Isotopically labeled vitamin D derivatives and processes for preparing same |
FR2457282A1 (fr) * | 1979-05-23 | 1980-12-19 | Roussel Uclaf | Nouveau derive du 1a,25 dihydroxy cholecalciferol, son procede de preparation et son application comme medicament |
IL60270A0 (en) * | 1979-06-14 | 1980-09-16 | Diamond Shamrock Corp | Preparation of 25-ydroxycholesterol |
US4252797A (en) * | 1979-07-19 | 1981-02-24 | Walter Rosenthal | Corticosteroid calcium compositions and treatment of rheumatic diseases therewith |
US4260804A (en) * | 1980-02-20 | 1981-04-07 | Wisconsin Alumni Research Foundation | Processes for preparing calcitroic acid and esters thereof |
US5043170A (en) * | 1989-02-14 | 1991-08-27 | Hoffmann-La Roche Inc. | Animal feed composition containing a vitamin D metabolite |
KR960013798B1 (ko) * | 1992-04-24 | 1996-10-10 | 재단법인 한국전자통신연구소 | 평면 도파로형 공간 스위치 |
AU666529B2 (en) * | 1992-04-24 | 1996-02-15 | Wisconsin Alumni Research Foundation | Method of treating osteoporosis with 1 alpha, 24 (R)-dihydroxy-22 (E)-dehydro-vitamin D3 |
US5194431A (en) | 1992-07-08 | 1993-03-16 | Wisconsin Alumni Research Foundation | 24-cyclopropane vitamin D derivatives |
MX9604831A (es) | 1994-04-15 | 1998-05-31 | Upjohn Co | Formas nuevas de cristal de 1-[5-metanosulfonamidoindolil-2-carbonil]-4-[3-(1-metiletila mino)-2-piridinil]-piperazina. |
US6432936B1 (en) | 1999-01-20 | 2002-08-13 | Wisconsin Alumni Research Foundation | Crystalline 1α-hydroxyvitamin D2 and method of purification thereof |
US7235655B2 (en) * | 2002-03-22 | 2007-06-26 | Pharmacia & Upjohn Company | Processes to prepare eplerenone |
PL3095447T3 (pl) | 2006-02-03 | 2022-02-14 | Opko Renal, Llc | Leczenie niedoboru lub deficytu witaminy d 25-hydroksywitaminą d2 i 25- hydroksywitaminą d3 |
SI2037936T1 (sl) | 2006-06-21 | 2014-11-28 | Opko Renal, Llc | Postopek zdravljenja in prepreäśevanja sekundarnega hiperparatiroidizma |
ES2403107T3 (es) | 2007-04-25 | 2013-05-14 | Cytochroma Inc. | Método de tratamiento de insuficiencia y deficiencia de vitamina D |
EP2148683A4 (fr) | 2007-04-25 | 2012-09-12 | Proventiv Therapeutics Llc | Procédé sûr et efficace de traitement et de prévention de l'hyperparathyroïdie secondaire dans les maladies rénales chroniques |
DK2148661T3 (da) | 2007-04-25 | 2013-03-25 | Cytochroma Inc | Orale præparater med kontrolleret afgivelse omfattende vitamin D-forbindelse og voksagtig bærer |
CA2714996C (fr) | 2008-04-02 | 2020-04-07 | Cytochroma Inc. | Procedes, compositions, utilisations, et kits utiles pour la carence en vitamine d et des troubles associes |
PT2552484T (pt) | 2010-03-29 | 2020-04-03 | Opko Ireland Global Holdings Ltd | Métodos e composições para redução dos níveis de parafróides |
KR101847947B1 (ko) | 2013-03-15 | 2018-05-28 | 옵코 아이피 홀딩스 Ⅱ 인코포레이티드 | 안정화되고 변형된 비타민 d 방출 제형 |
CR20170085A (es) | 2014-08-07 | 2017-04-25 | Opko Ireland Global Holdings Ltd | Terapia adjuntiva con 25-hidroxi vitamina d |
BR112018069727A2 (pt) | 2016-03-28 | 2019-02-05 | Opko Ireland Global Holdings Ltd | métodos de tratamento com vitamina d |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1052283B (it) * | 1968-07-01 | 1981-06-20 | Wisconsin Alumni Res Found | Processo per preparare composti del calciferolo e relativi composti |
-
1969
- 1969-03-17 US US00807929A patent/US3833622A/en not_active Expired - Lifetime
-
1970
- 1970-02-04 CA CA073,970A patent/CA968789A/en not_active Expired
- 1970-02-09 IL IL33860A patent/IL33860A/en unknown
- 1970-02-11 GB GB6597/70A patent/GB1286761A/en not_active Expired
- 1970-03-14 DE DE2012167A patent/DE2012167C2/de not_active Expired
- 1970-03-16 FR FR7009330A patent/FR2035000B1/fr not_active Expired
- 1970-03-16 NL NL7003686A patent/NL7003686A/xx unknown
- 1970-03-17 BE BE747492D patent/BE747492A/fr not_active IP Right Cessation
- 1970-03-17 CH CH398070A patent/CH528500A/de not_active IP Right Cessation
- 1970-03-17 JP JP45022231A patent/JPS4934980B1/ja active Pending
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2571369A1 (fr) * | 1984-10-04 | 1986-04-11 | Wisconsin Alumni Res Found | Derives de la vitamine d et precurseurs de ceux-ci et compositions pharmaceutiques en contenant |
Also Published As
Publication number | Publication date |
---|---|
CH528500A (de) | 1972-09-30 |
DE2012167C2 (de) | 1982-09-23 |
GB1286761A (en) | 1972-08-23 |
JPS4934980B1 (fr) | 1974-09-19 |
FR2035000A1 (fr) | 1970-12-18 |
NL7003686A (fr) | 1970-09-21 |
FR2035000B1 (fr) | 1974-01-11 |
IL33860A (en) | 1973-10-25 |
CA968789A (en) | 1975-06-03 |
US3833622A (en) | 1974-09-03 |
IL33860A0 (en) | 1970-04-20 |
DE2012167A1 (de) | 1970-10-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: THE UPJOHN CY Effective date: 19860331 |