BE2011C004I2 - - Google Patents

Info

Publication number
BE2011C004I2
BE2011C004I2 BE2011C004C BE2011C004C BE2011C004I2 BE 2011C004 I2 BE2011C004 I2 BE 2011C004I2 BE 2011C004 C BE2011C004 C BE 2011C004C BE 2011C004 C BE2011C004 C BE 2011C004C BE 2011C004 I2 BE2011C004 I2 BE 2011C004I2
Authority
BE
Belgium
Application number
BE2011C004C
Other languages
French (fr)
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of BE2011C004I2 publication Critical patent/BE2011C004I2/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE2011C004C 1999-06-22 2011-02-03 BE2011C004I2 (en(2012))

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US09/338,185 US6403567B1 (en) 1999-06-22 1999-06-22 N-pyrazole A2A adenosine receptor agonists

Publications (1)

Publication Number Publication Date
BE2011C004I2 true BE2011C004I2 (en(2012)) 2019-05-21

Family

ID=23323763

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2011C004C BE2011C004I2 (en(2012)) 1999-06-22 2011-02-03

Country Status (27)

Country Link
US (9) US6403567B1 (en(2012))
EP (1) EP1189916B1 (en(2012))
JP (1) JP4727880B2 (en(2012))
KR (1) KR100463300B1 (en(2012))
CN (1) CN1167709C (en(2012))
AR (1) AR024441A1 (en(2012))
AT (1) ATE256141T1 (en(2012))
AU (1) AU760806B2 (en(2012))
BE (1) BE2011C004I2 (en(2012))
BR (1) BRPI0011856B8 (en(2012))
CA (1) CA2377746C (en(2012))
CY (1) CY2011002I2 (en(2012))
DE (2) DE122011000010I1 (en(2012))
DK (1) DK1189916T3 (en(2012))
ES (1) ES2209974T3 (en(2012))
FR (1) FR11C0004I2 (en(2012))
HK (1) HK1044952B (en(2012))
IL (2) IL147198A0 (en(2012))
LU (1) LU91785I2 (en(2012))
MX (1) MXPA01013325A (en(2012))
NO (2) NO322457B1 (en(2012))
NZ (1) NZ516334A (en(2012))
PT (1) PT1189916E (en(2012))
TR (1) TR200200588T2 (en(2012))
TW (1) TWI230161B (en(2012))
WO (1) WO2000078779A2 (en(2012))
ZA (1) ZA200200301B (en(2012))

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WO2000078779A2 (en) 2000-12-28
ATE256141T1 (de) 2003-12-15
CY2011002I1 (el) 2012-01-25
US20110144320A1 (en) 2011-06-16
TWI230161B (en) 2005-04-01
NO20016350D0 (no) 2001-12-21
US20140073596A1 (en) 2014-03-13
CA2377746C (en) 2007-04-10
FR11C0004I2 (fr) 2012-03-16
JP4727880B2 (ja) 2011-07-20
US6403567B1 (en) 2002-06-11
KR20020028910A (ko) 2002-04-17
CN1358191A (zh) 2002-07-10
DE60007127D1 (de) 2004-01-22
US8278435B2 (en) 2012-10-02
US20040038928A1 (en) 2004-02-26
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US20060052332A1 (en) 2006-03-09
EP1189916B1 (en) 2003-12-10
US6642210B1 (en) 2003-11-04
DE60007127T2 (de) 2004-09-16
BR0011856B1 (pt) 2014-06-17
CN1167709C (zh) 2004-09-22
BRPI0011856B8 (pt) 2021-05-25
US8569260B2 (en) 2013-10-29
ES2209974T3 (es) 2004-07-01
KR100463300B1 (ko) 2004-12-23
DK1189916T3 (da) 2004-03-22
EP1189916A2 (en) 2002-03-27
US7655637B2 (en) 2010-02-02
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