AU777185B2 - Pharmaceutical form of administration for peptides, methods for its production and use - Google Patents
Pharmaceutical form of administration for peptides, methods for its production and use Download PDFInfo
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- AU777185B2 AU777185B2 AU74041/01A AU7404101A AU777185B2 AU 777185 B2 AU777185 B2 AU 777185B2 AU 74041/01 A AU74041/01 A AU 74041/01A AU 7404101 A AU7404101 A AU 7404101A AU 777185 B2 AU777185 B2 AU 777185B2
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Classifications
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
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| DE10024451 | 2000-05-18 | ||
| DE10024451A DE10024451A1 (de) | 2000-05-18 | 2000-05-18 | Pharmazeutische Darreichungsform für Peptide, Verfahren zu deren Herstellung und Verwendung |
| PCT/EP2001/005555 WO2001087265A2 (de) | 2000-05-18 | 2001-05-16 | Pharmazeutische darreichungsform für peptide, verfahren zu deren herstellung und verwendung |
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| AU7404101A AU7404101A (en) | 2001-11-26 |
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| BR (1) | BR0110892A (cs) |
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| IL (1) | IL152479A (cs) |
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Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US6828415B2 (en) * | 1993-02-19 | 2004-12-07 | Zentaris Gmbh | Oligopeptide lyophilisate, their preparation and use |
| JP4940492B2 (ja) * | 2000-09-04 | 2012-05-30 | 大正製薬株式会社 | 鉄化合物配合内服液剤 |
| DE10157628A1 (de) * | 2001-11-26 | 2003-06-12 | Zentaris Ag | Injektionslösung eines LHRH-Antagonisten |
| US7214662B2 (en) | 2001-11-27 | 2007-05-08 | Zentaris Gmbh | Injectable solution of an LHRH antagonist |
| HRP20050371B1 (hr) * | 2002-09-27 | 2014-09-26 | Zentaris Gmbh | Oblik za primjenu farmaceutiski djelatnih peptida s produljenim oslobađanjem djelatnog sastojka i postupak za njihovu proizvodnju |
| DE10332160A1 (de) | 2003-07-15 | 2005-02-03 | Röhm GmbH & Co. KG | Multipartikuläre Arzneiform, enthaltend mucoadhaesiv formulierte Peptid- oder Protein-Wirkstoffe, sowie ein Verfahren zur Herstellung der Arzneiform |
| ES2297688T3 (es) * | 2004-03-12 | 2008-05-01 | Intercell Ag | Procedimiento para solubizar mezclas de peptidos. |
| EP1674082A1 (de) | 2004-12-22 | 2006-06-28 | Zentaris GmbH | Verfahren zur Herstellung von sterilen Suspensionen oder Lyophilisaten schwerlöslicher basischer Peptidkomplexe, diese enthaltende pharmazeutische Formulierungen sowie ihre Verwendung als Arzneimittel |
| WO2006110119A1 (fr) * | 2005-04-15 | 2006-10-19 | Victor Pavlovich Kutnyak | Produit antineoplasique (et variantes) |
| WO2006110118A1 (fr) * | 2005-04-15 | 2006-10-19 | Victor Pavlovich Kutnyak | Produit cytoprotecteur |
| WO2012077131A1 (en) * | 2010-12-06 | 2012-06-14 | Astron Research Limited | A stable ready-to-use cetrorelix injection |
| CN102144980B (zh) * | 2011-03-07 | 2013-01-09 | 深圳市健元医药科技有限公司 | 一种更加稳定的lhrh拮抗剂冻干粉针剂 |
| CN106456704A (zh) * | 2014-04-16 | 2017-02-22 | Veyx-药物有限公司 | 兽药组合物和其应用 |
| DK3576771T3 (da) * | 2017-01-31 | 2022-05-30 | Veru Inc | Sammensætninger og fremgangsmåder til langvarig frigivelse af antagonister for gonadotropin-frigivende hormon (gnrh) |
| EP3982926A1 (en) * | 2019-06-17 | 2022-04-20 | Intas Pharmaceuticals Ltd. | A stable formulation of cetrorelix |
| PT3811927T (pt) * | 2019-10-24 | 2021-12-14 | Sun Pharmaceutical Ind Ltd | Forma galénica parentérica estável de acetato de cetrorrelix |
| WO2022269572A1 (en) | 2021-06-25 | 2022-12-29 | Extrovis Ag | Pharmaceutical compositions |
| US20240358632A1 (en) * | 2021-08-11 | 2024-10-31 | Rk Pharma Inc. | Ready to use compositions of cetrorelix acetate |
| CN115969954A (zh) * | 2023-01-09 | 2023-04-18 | 开封明仁药业有限公司 | 一种注射用西曲瑞克冻干药物组合物及其制备方法 |
| EP4534074A1 (en) * | 2023-10-04 | 2025-04-09 | Ares Trading S.A. | Liquid cetrorelix composition |
Family Cites Families (41)
| Publication number | Priority date | Publication date | Assignee | Title |
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| DE141996C (cs) | ||||
| DD141996A1 (de) * | 1979-02-21 | 1980-06-04 | Ingrid Wolf | Verfahren zur herstellung von lyophilisierten lhrh-praeparationen |
| JPS5892620A (ja) * | 1981-11-28 | 1983-06-02 | Sunstar Inc | インタ−フエロン安定配合組成物 |
| US4565804A (en) * | 1984-09-07 | 1986-01-21 | The Salk Institute For Biological Studies | GnRH Antagonists VI |
| US4800191A (en) * | 1987-07-17 | 1989-01-24 | Schally Andrew Victor | LHRH antagonists |
| DK163689A (da) * | 1988-04-08 | 1989-10-30 | Sandoz Ag | Peptidderivater |
| JPH0725662B2 (ja) * | 1990-10-22 | 1995-03-22 | アース製薬株式会社 | 使用時調製型上皮細胞成長因子含有水性薬剤の安定化方法 |
| US5643878A (en) * | 1991-09-12 | 1997-07-01 | Ciba-Geigy Corporation | 5-amino-4-hydroxyhexanoic acid derivatives |
| JP3608802B2 (ja) * | 1991-09-20 | 2005-01-12 | 第一サントリーファーマ株式会社 | 安定なカルシトニン医薬組成物及びその製造法 |
| AU4198793A (en) * | 1992-07-24 | 1994-01-27 | Takeda Chemical Industries Ltd. | Microparticle preparation and production thereof |
| EP0666752A4 (en) * | 1992-10-16 | 1996-09-11 | Smithkline Beecham Corp | THERAPEUTIC MICROEMULSIONS. |
| DE4242919A1 (de) * | 1992-12-18 | 1994-06-23 | Boehringer Mannheim Gmbh | Verfahren zur Herstellung von lagerstabilen wässrigen pharmazeutischen Zubereitungen von G-CSF |
| DE4305225A1 (de) * | 1993-02-19 | 1994-08-25 | Asta Medica Ag | Neues Herstellverfahren für Cetrorelix Lyophilisat |
| US6828415B2 (en) * | 1993-02-19 | 2004-12-07 | Zentaris Gmbh | Oligopeptide lyophilisate, their preparation and use |
| JP3636480B2 (ja) * | 1993-05-19 | 2005-04-06 | 科研製薬株式会社 | 凍結乾燥製剤 |
| US6087324A (en) * | 1993-06-24 | 2000-07-11 | Takeda Chemical Industries, Ltd. | Sustained-release preparation |
| JP2915296B2 (ja) * | 1993-08-30 | 1999-07-05 | 宇野 潤 | 抗真菌製剤 |
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| US5595760A (en) | 1994-09-02 | 1997-01-21 | Delab | Sustained release of peptides from pharmaceutical compositions |
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-
2000
- 2000-05-18 DE DE10024451A patent/DE10024451A1/de not_active Ceased
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2001
- 2001-05-16 PL PL363007A patent/PL203958B1/pl unknown
- 2001-05-16 RU RU2002134463/15A patent/RU2253438C2/ru not_active IP Right Cessation
- 2001-05-16 JP JP2001583734A patent/JP4944340B2/ja not_active Expired - Fee Related
- 2001-05-16 CN CNB018177042A patent/CN100342908C/zh not_active Expired - Fee Related
- 2001-05-16 BR BR0110892-1A patent/BR0110892A/pt not_active IP Right Cessation
- 2001-05-16 HU HU0302050A patent/HUP0302050A3/hu unknown
- 2001-05-16 IL IL152479A patent/IL152479A/en active IP Right Grant
- 2001-05-16 UA UA20021210143A patent/UA74578C2/uk unknown
- 2001-05-16 SK SK1716-2002A patent/SK288118B6/sk not_active IP Right Cessation
- 2001-05-16 EP EP01940482.1A patent/EP1282400B1/de not_active Expired - Lifetime
- 2001-05-16 AU AU74041/01A patent/AU777185B2/en not_active Ceased
- 2001-05-16 KR KR1020027015424A patent/KR100580142B1/ko not_active Expired - Fee Related
- 2001-05-16 CZ CZ20023969A patent/CZ303981B6/cs not_active IP Right Cessation
- 2001-05-16 NZ NZ522381A patent/NZ522381A/en not_active IP Right Cessation
- 2001-05-16 TW TW090111674A patent/TWI243059B/zh not_active IP Right Cessation
- 2001-05-16 WO PCT/EP2001/005555 patent/WO2001087265A2/de not_active Ceased
- 2001-05-16 MX MXPA02011389A patent/MXPA02011389A/es active IP Right Grant
- 2001-05-18 US US09/861,009 patent/US7718599B2/en not_active Expired - Fee Related
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- 2001-05-18 AR ARP010102371A patent/AR028588A1/es not_active Application Discontinuation
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2002
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- 2002-11-25 BG BG107312A patent/BG65976B1/bg unknown
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2011
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Legal Events
| Date | Code | Title | Description |
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| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase | ||
| PC1 | Assignment before grant (sect. 113) |
Owner name: ZENTARIS GMBH Free format text: THE FORMER OWNER WAS: ZENTARIS AG |
|
| TC | Change of applicant's name (sec. 104) |
Owner name: ZENTARIS GMBH Free format text: FORMER NAME: ZENTARIS AG |