AU773505B2 - Arylthiazolidinedione and aryloxazolidinedione derivatives - Google Patents

Arylthiazolidinedione and aryloxazolidinedione derivatives Download PDF

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Publication number
AU773505B2
AU773505B2 AU58755/00A AU5875500A AU773505B2 AU 773505 B2 AU773505 B2 AU 773505B2 AU 58755/00 A AU58755/00 A AU 58755/00A AU 5875500 A AU5875500 A AU 5875500A AU 773505 B2 AU773505 B2 AU 773505B2
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AU
Australia
Prior art keywords
propyl
compound
phenyl
methyl
propoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU58755/00A
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English (en)
Other versions
AU5875500A (en
Inventor
Julia K. Boueres
James V. Heck
Victoria K Lombardo
Edward Metzger
Soumya P Sahoo
Conrad Santini
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of AU5875500A publication Critical patent/AU5875500A/en
Application granted granted Critical
Publication of AU773505B2 publication Critical patent/AU773505B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/34—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
AU58755/00A 1999-06-18 2000-06-16 Arylthiazolidinedione and aryloxazolidinedione derivatives Ceased AU773505B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13995399P 1999-06-18 1999-06-18
US60/139953 1999-06-18
PCT/US2000/016586 WO2000078312A1 (en) 1999-06-18 2000-06-16 Arylthiazolidinedione and aryloxazolidinedione derivatives

Publications (2)

Publication Number Publication Date
AU5875500A AU5875500A (en) 2001-01-09
AU773505B2 true AU773505B2 (en) 2004-05-27

Family

ID=22489062

Family Applications (1)

Application Number Title Priority Date Filing Date
AU58755/00A Ceased AU773505B2 (en) 1999-06-18 2000-06-16 Arylthiazolidinedione and aryloxazolidinedione derivatives

Country Status (9)

Country Link
US (1) US6399640B1 (https=)
EP (1) EP1194146B1 (https=)
JP (1) JP2003502369A (https=)
AT (1) ATE333448T1 (https=)
AU (1) AU773505B2 (https=)
CA (1) CA2376919C (https=)
DE (1) DE60029446T2 (https=)
ES (1) ES2265952T3 (https=)
WO (1) WO2000078312A1 (https=)

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Also Published As

Publication number Publication date
EP1194146B1 (en) 2006-07-19
DE60029446T2 (de) 2007-02-08
ES2265952T3 (es) 2007-03-01
JP2003502369A (ja) 2003-01-21
WO2000078312A1 (en) 2000-12-28
EP1194146A1 (en) 2002-04-10
CA2376919C (en) 2008-11-04
US6399640B1 (en) 2002-06-04
DE60029446D1 (de) 2006-08-31
AU5875500A (en) 2001-01-09
EP1194146A4 (en) 2002-07-31
ATE333448T1 (de) 2006-08-15
CA2376919A1 (en) 2000-12-28

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