AU734734B2 - Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction - Google Patents
Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction Download PDFInfo
- Publication number
- AU734734B2 AU734734B2 AU11254/99A AU1125499A AU734734B2 AU 734734 B2 AU734734 B2 AU 734734B2 AU 11254/99 A AU11254/99 A AU 11254/99A AU 1125499 A AU1125499 A AU 1125499A AU 734734 B2 AU734734 B2 AU 734734B2
- Authority
- AU
- Australia
- Prior art keywords
- phosphodiesterase inhibitor
- phosphodiesterase
- type
- formulation
- drug
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US95881697A | 1997-10-28 | 1997-10-28 | |
US08/958816 | 1997-10-28 | ||
US09/181070 | 1998-10-27 | ||
US09/181,070 US6037346A (en) | 1997-10-28 | 1998-10-27 | Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
PCT/US1998/022928 WO1999021558A2 (fr) | 1997-10-28 | 1998-10-28 | Apport local d'inhibiteurs de phosphodiesterases, dans le traitement du dysfonctionnement erectile |
Publications (2)
Publication Number | Publication Date |
---|---|
AU1125499A AU1125499A (en) | 1999-05-17 |
AU734734B2 true AU734734B2 (en) | 2001-06-21 |
Family
ID=25501340
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU11254/99A Ceased AU734734B2 (en) | 1997-10-28 | 1998-10-28 | Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP1027054A4 (fr) |
JP (1) | JP2003525845A (fr) |
AU (1) | AU734734B2 (fr) |
CA (1) | CA2305394C (fr) |
WO (1) | WO1999021558A2 (fr) |
Families Citing this family (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6331543B1 (en) | 1996-11-01 | 2001-12-18 | Nitromed, Inc. | Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use |
CA2295595A1 (fr) | 1997-07-09 | 1999-01-21 | Androsolutions, Inc. | Compositions et procedes perfectionnes de traitement des troubles de l'erection chez l'homme |
US6103765A (en) | 1997-07-09 | 2000-08-15 | Androsolutions, Inc. | Methods for treating male erectile dysfunction |
US6548490B1 (en) * | 1997-10-28 | 2003-04-15 | Vivus, Inc. | Transmucosal administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
US6403597B1 (en) | 1997-10-28 | 2002-06-11 | Vivus, Inc. | Administration of phosphodiesterase inhibitors for the treatment of premature ejaculation |
US6472425B1 (en) | 1997-10-31 | 2002-10-29 | Nitromed, Inc. | Methods for treating female sexual dysfunctions |
US6541487B1 (en) * | 1998-05-01 | 2003-04-01 | R.T. Alamo Ventures I, Llc | PDE III inhibitors for treating sexual dysfunction |
DE19834506A1 (de) * | 1998-07-31 | 2000-02-03 | Hexal Ag | Transmucosales therapeutisches System zur Anwendung von Sildenafil |
EP1157694A4 (fr) * | 1998-12-07 | 2002-08-28 | Nissan Chemical Ind Ltd | Agent therapeutique pour le traitement de la dyserection |
IT1312310B1 (it) * | 1999-05-07 | 2002-04-15 | Recordati Ind Chimica E Farma | Uso di antagonisti selettivi del recettore adrenergico a 1b per ilmiglioramento della disfunzione sessuale |
IL130968A (en) * | 1999-07-15 | 2002-12-01 | Shmuel Simon | Pharmaceutical composition comprising sildenafil or its analogs, useful for the treatment of tinnitus and hearing loss |
US6323241B1 (en) * | 2000-01-10 | 2001-11-27 | Nexmed (Holdings) Inc. | Prostaglandin compositions and methods of treatment for male erectile dysfunction |
AU2001273636A1 (en) | 2000-06-27 | 2002-01-08 | Qualilife Pharmaceuticals Inc. | Compositions and methods for treating females sexual response |
US6503894B1 (en) | 2000-08-30 | 2003-01-07 | Unimed Pharmaceuticals, Inc. | Pharmaceutical composition and method for treating hypogonadism |
US6821978B2 (en) | 2000-09-19 | 2004-11-23 | Schering Corporation | Xanthine phosphodiesterase V inhibitors |
FI20002755A0 (fi) * | 2000-12-15 | 2000-12-15 | Orion Yhtymae Oyj | Menetelmä erektiilin dysfunktion hoitamiseen |
CA2431077A1 (fr) * | 2000-12-19 | 2002-06-27 | Merck Patent Gesellschaft Mit Beschraenkter Haftung | Formulation pharmaceutique contenant des pyrazolo[4,3-d]pyrimidines et des antithrombotiques, des antagonistes de calcium, des prostaglandines ou des derives de prostaglandine |
US20040058940A1 (en) * | 2000-12-19 | 2004-03-25 | Hans-Michael Eggenweiler | Pharmaceutical formulation comprising thienopyrimidines and antithrombotics, calcium antagonists, prostaglandins or prostaglandin derivatives (2) |
HUP0303289A2 (hu) * | 2000-12-19 | 2004-01-28 | Merck Patent Gmbh. | Tienopirimidineket és trombózisellenes szereket, kalcium antagonistákat, prosztaglandinokat vagy prosztaglandinszármazékokat tartalmazó gyógyszerkészítmények |
EP1224933A1 (fr) * | 2001-01-19 | 2002-07-24 | Sanofi-Synthelabo | Nouvelle combinaison d'actifs avec alfuzosine et apomorphine |
US6943171B2 (en) | 2001-11-09 | 2005-09-13 | Schering Corporation | Polycyclic guanine derivative phosphodiesterase V inhibitors |
PT2311432E (pt) | 2002-06-07 | 2015-02-09 | Dyax Corp | Polipeptídeos de domínio kunitz modificado e sua utilização para a redução de isquemia ou aparecimento de uma resposta inflamatória sistémica associada a um procedimento cirúrgico |
WO2004071533A1 (fr) * | 2003-02-14 | 2004-08-26 | Takeda Pharmaceutical Company Limited | Preparation pour administration topique |
WO2005021557A2 (fr) * | 2003-08-29 | 2005-03-10 | Dyax Corp. | Inhibiteurs de protease poly-pegylee |
US7235530B2 (en) | 2004-09-27 | 2007-06-26 | Dyax Corporation | Kallikrein inhibitors and anti-thrombolytic agents and uses thereof |
DK1802277T3 (da) * | 2004-10-18 | 2010-05-17 | Polymun Scient Immunbio Forsch | Liposomal sammensætning indeholdende en aktiv bestanddel til relaksation af glat muskulatur og terapeutisk anvendelse af sammensætningen |
KR20140054312A (ko) * | 2007-02-12 | 2014-05-08 | 디엠아이 바이오사이언시스 인코포레이티드 | 조루 및 발기부전을 동시에 치료하는 방법 |
KR20100050488A (ko) * | 2007-06-26 | 2010-05-13 | 솔베이 파마슈티칼스 비. 브이 | 전구약물로서 실데나필 n-옥사이드 |
KR102555955B1 (ko) | 2014-03-27 | 2023-07-18 | 다케다 파머수티컬 컴패니 리미티드 | 당뇨병성 황반 부종의 치료를 위한 조성물 및 방법 |
WO2021027943A1 (fr) * | 2019-08-14 | 2021-02-18 | 正大天晴药业集团南京顺欣制药有限公司 | Dérivé de pyrimidinopyridazinone et son utilisation médicale |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4801587A (en) * | 1987-03-02 | 1989-01-31 | Gene Voss | Impotence ointment |
US5145852A (en) * | 1989-07-11 | 1992-09-08 | Ronald Virag | Vaso-active medicament to treat impotence |
US5250534A (en) * | 1990-06-20 | 1993-10-05 | Pfizer Inc. | Pyrazolopyrimidinone antianginal agents |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5242391A (en) * | 1990-04-25 | 1993-09-07 | Alza Corporation | Urethral insert for treatment of erectile dysfunction |
GB9114760D0 (en) * | 1991-07-09 | 1991-08-28 | Pfizer Ltd | Therapeutic agents |
GB9301192D0 (en) * | 1993-06-09 | 1993-06-09 | Trott Francis W | Flower shaped mechanised table |
GB9423910D0 (en) * | 1994-11-26 | 1995-01-11 | Pfizer Ltd | Therapeutic agents |
WO1998019672A1 (fr) * | 1996-11-01 | 1998-05-14 | Nitromed Inc. | Composes nitroses et nitrosyles inhibiteurs de la phosphodiesterase, compositions comprenant ces composes et utilisations correspondantes |
JP2001505198A (ja) * | 1996-11-20 | 2001-04-17 | ビイク グルデン ロンベルク ヒエーミツシエ フアブリーク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング | Pde阻害剤としての置換ジヒドロベンゾフラン |
JP2001520999A (ja) * | 1997-10-28 | 2001-11-06 | アシビ, エルエルシー | 女性の性的機能不全の処置 |
-
1998
- 1998-10-28 JP JP2000517716A patent/JP2003525845A/ja active Pending
- 1998-10-28 EP EP19980954032 patent/EP1027054A4/fr not_active Ceased
- 1998-10-28 AU AU11254/99A patent/AU734734B2/en not_active Ceased
- 1998-10-28 WO PCT/US1998/022928 patent/WO1999021558A2/fr not_active Application Discontinuation
- 1998-10-28 CA CA002305394A patent/CA2305394C/fr not_active Expired - Lifetime
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4801587A (en) * | 1987-03-02 | 1989-01-31 | Gene Voss | Impotence ointment |
US5145852A (en) * | 1989-07-11 | 1992-09-08 | Ronald Virag | Vaso-active medicament to treat impotence |
US5250534A (en) * | 1990-06-20 | 1993-10-05 | Pfizer Inc. | Pyrazolopyrimidinone antianginal agents |
Also Published As
Publication number | Publication date |
---|---|
WO1999021558A2 (fr) | 1999-05-06 |
WO1999021558A3 (fr) | 2000-10-26 |
EP1027054A4 (fr) | 2002-11-04 |
CA2305394C (fr) | 2006-12-12 |
EP1027054A1 (fr) | 2000-08-16 |
JP2003525845A (ja) | 2003-09-02 |
AU1125499A (en) | 1999-05-17 |
CA2305394A1 (fr) | 1999-05-06 |
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