AU644496B2 - Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinoalkylbenzothiazine compounds and processes for their preparation and medicaments containing these compounds - Google Patents

Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinoalkylbenzothiazine compounds and processes for their preparation and medicaments containing these compounds Download PDF

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Publication number
AU644496B2
AU644496B2 AU88091/91A AU8809191A AU644496B2 AU 644496 B2 AU644496 B2 AU 644496B2 AU 88091/91 A AU88091/91 A AU 88091/91A AU 8809191 A AU8809191 A AU 8809191A AU 644496 B2 AU644496 B2 AU 644496B2
Authority
AU
Australia
Prior art keywords
compounds
denotes
general formula
lower alkyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU88091/91A
Other languages
English (en)
Other versions
AU8809191A (en
Inventor
Francois Floc'h
Daniel Jasserand
Richard White
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Products GmbH
Original Assignee
Kali Chemie Pharma GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kali Chemie Pharma GmbH filed Critical Kali Chemie Pharma GmbH
Publication of AU8809191A publication Critical patent/AU8809191A/en
Application granted granted Critical
Publication of AU644496B2 publication Critical patent/AU644496B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU88091/91A 1990-11-24 1991-11-22 Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinoalkylbenzothiazine compounds and processes for their preparation and medicaments containing these compounds Ceased AU644496B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4037427A DE4037427A1 (de) 1990-11-24 1990-11-24 Heterocyclisch substituierte piperazinoalkylbenzoxazin und -thiazin-verbindungen sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE4037427 1990-11-24

Publications (2)

Publication Number Publication Date
AU8809191A AU8809191A (en) 1992-05-28
AU644496B2 true AU644496B2 (en) 1993-12-09

Family

ID=6418854

Family Applications (1)

Application Number Title Priority Date Filing Date
AU88091/91A Ceased AU644496B2 (en) 1990-11-24 1991-11-22 Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinoalkylbenzothiazine compounds and processes for their preparation and medicaments containing these compounds

Country Status (16)

Country Link
EP (1) EP0488008A1 (OSRAM)
JP (1) JPH05140156A (OSRAM)
KR (1) KR920009826A (OSRAM)
CN (1) CN1062140A (OSRAM)
AU (1) AU644496B2 (OSRAM)
CA (1) CA2056009A1 (OSRAM)
DE (1) DE4037427A1 (OSRAM)
FI (1) FI915518A7 (OSRAM)
HU (1) HUT62004A (OSRAM)
IE (1) IE914074A1 (OSRAM)
IL (1) IL99949A0 (OSRAM)
MX (1) MX9102192A (OSRAM)
NO (1) NO914577L (OSRAM)
PT (1) PT99570A (OSRAM)
TW (1) TW218876B (OSRAM)
ZA (1) ZA918341B (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2667068B1 (fr) * 1990-09-26 1994-09-09 Adir Nouvelles amines alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
AU638154B2 (en) * 1990-10-04 1993-06-17 Suntory Limited Benzoxazine derivative and herbicide containing same as an active ingredient
AU5979494A (en) * 1993-02-05 1994-08-29 Yamanouchi Pharmaceutical Co., Ltd. Novel benzoxazine derivative, medicine containing the same, and intermediate therefor
FR2702477B1 (fr) * 1993-03-08 1995-04-28 Synthelabo Dérivés de benzoxazine, leur préparation et leur application en thérapeutique.
FR2755690B1 (fr) * 1996-11-08 1998-12-18 Adir Nouveaux derives aminomethyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6853187A (en) * 1986-02-11 1987-08-13 Takeda Chemical Industries Ltd. 1,4-benzoxazine derivatives
AU8471191A (en) * 1990-09-26 1992-04-16 Adir Et Compagnie New heterocycle-substituted alkylamines, process for preparing these and pharmaceutical compositions containing them

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1244481A (en) * 1967-11-08 1971-09-02 Wyeth John & Brother Ltd Benzothiazine derivatives and the preparation thereof
EP0186310A1 (en) * 1984-11-28 1986-07-02 Takeda Chemical Industries, Ltd. 1,4-Benzothiazine Derivatives, their production and use

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6853187A (en) * 1986-02-11 1987-08-13 Takeda Chemical Industries Ltd. 1,4-benzoxazine derivatives
AU8471191A (en) * 1990-09-26 1992-04-16 Adir Et Compagnie New heterocycle-substituted alkylamines, process for preparing these and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
FI915518A0 (fi) 1991-11-22
JPH05140156A (ja) 1993-06-08
FI915518L (fi) 1992-05-25
TW218876B (OSRAM) 1994-01-11
EP0488008A1 (de) 1992-06-03
IE914074A1 (en) 1992-06-03
HUT62004A (en) 1993-03-29
NO914577D0 (no) 1991-11-22
KR920009826A (ko) 1992-06-25
NO914577L (no) 1992-05-25
HU913482D0 (en) 1992-01-28
CA2056009A1 (en) 1992-05-25
DE4037427A1 (de) 1992-05-27
ZA918341B (en) 1992-07-29
MX9102192A (es) 1994-08-31
FI915518A7 (fi) 1992-05-25
AU8809191A (en) 1992-05-28
PT99570A (pt) 1992-10-30
IL99949A0 (en) 1992-08-18
CN1062140A (zh) 1992-06-24

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