AU603795B2 - Pyridine compounds - Google Patents

Pyridine compounds Download PDF

Info

Publication number
AU603795B2
AU603795B2 AU72512/87A AU7251287A AU603795B2 AU 603795 B2 AU603795 B2 AU 603795B2 AU 72512/87 A AU72512/87 A AU 72512/87A AU 7251287 A AU7251287 A AU 7251287A AU 603795 B2 AU603795 B2 AU 603795B2
Authority
AU
Australia
Prior art keywords
formula
lower alkyl
compounds
carboxy
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU72512/87A
Other languages
English (en)
Other versions
AU7251287A (en
Inventor
Marc Lang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU7251287A publication Critical patent/AU7251287A/en
Application granted granted Critical
Publication of AU603795B2 publication Critical patent/AU603795B2/en
Assigned to NOVARTIS AG reassignment NOVARTIS AG Request to Amend Deed and Register Assignors: CIBA-GEIGY AG
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU72512/87A 1986-05-06 1987-05-05 Pyridine compounds Expired AU603795B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1846/86 1986-05-06
CH184686 1986-05-06

Publications (2)

Publication Number Publication Date
AU7251287A AU7251287A (en) 1987-11-12
AU603795B2 true AU603795B2 (en) 1990-11-29

Family

ID=4219979

Family Applications (1)

Application Number Title Priority Date Filing Date
AU72512/87A Expired AU603795B2 (en) 1986-05-06 1987-05-05 Pyridine compounds

Country Status (14)

Country Link
US (1) US4826832A (enExample)
EP (1) EP0246187B1 (enExample)
JP (1) JPS62263183A (enExample)
AT (1) ATE72438T1 (enExample)
AU (1) AU603795B2 (enExample)
CA (1) CA1293502C (enExample)
DE (1) DE3776590D1 (enExample)
DK (1) DK169623B1 (enExample)
ES (1) ES2038207T3 (enExample)
GR (1) GR3003735T3 (enExample)
IE (1) IE59714B1 (enExample)
NZ (1) NZ220195A (enExample)
PT (1) PT84819B (enExample)
ZA (1) ZA873198B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0003960B1 (de) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-Substituierte Thia-Azaverbindungen, ihre Herstellung und diese enthaltende pharmazeutische Präparate
EP0215739B1 (de) * 1985-09-11 1993-09-01 Ciba-Geigy Ag Synthese von Beta-Lactamverbindungen
GB8716679D0 (en) * 1987-07-15 1987-08-19 Erba Farmitalia Penem derivatives
EP0462521A1 (en) * 1990-06-19 1991-12-27 Takeda Chemical Industries, Ltd. Crystalline penem, its production and use
US5492903A (en) * 1990-06-19 1996-02-20 Takeda Chemical Industries Ltd. Crystalline esters of (+)-(5R, 6S)-6-[(R)-1-hydroxyethyl]-3-(3-pyridyl)-7-oxo-4-thia-1-azabicyclo[3.2.0]he
EP0499274A1 (en) * 1991-02-15 1992-08-19 Takeda Chemical Industries, Ltd. Crystalline penem, its production and use
DE69130022T2 (de) * 1991-06-06 1999-05-27 Medevec Licensing B.V., Amsterdam Intraokuläre linse mit einer haptischen verankerungsplatte
EP0597401A3 (en) * 1992-11-11 1995-07-26 Takeda Chemical Industries Ltd Preparation of penemes.
US20040202714A1 (en) * 1999-10-12 2004-10-14 Daiichi Suntory Pharma Co., Ltd. Oral pharmaceutical composition
EP1138333B1 (en) * 1999-10-12 2004-02-25 Daiichi Suntory Pharma Co., Ltd. Medicinal compositions for oral use

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU5378779A (en) * 1978-12-18 1980-08-28 Bristol-Myers Company 2-penem antibiotics
AU8605382A (en) * 1981-07-15 1983-01-20 Sumitomo Chemical Company, Limited Penicillins and azetidinones

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0003960B1 (de) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-Substituierte Thia-Azaverbindungen, ihre Herstellung und diese enthaltende pharmazeutische Präparate
US4272437A (en) * 1978-12-18 1981-06-09 Bristol-Myers Company Antibacterial agents, and 4-thio azetidinone intermediates
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
US4386030A (en) * 1979-12-31 1983-05-31 Merck & Co., Inc. Process for preparing 6-(1'-hydroxyethyl)-2-substituted-pen-2-em-3-carboxylic acid
NZ201471A (en) * 1981-08-10 1985-09-13 Merck & Co Inc Antibacterial compositions containing penems and dipeptidase inhibitors
EP0109362A1 (de) * 1982-11-16 1984-05-23 Ciba-Geigy Ag Heterocyclylverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verwendung von letzteren
US4540580A (en) * 1982-11-16 1985-09-10 Schering Corporation 2-[(1'R)-1'-Aminoalkyl]penems
DE3366926D1 (en) * 1982-11-16 1986-11-20 Schering Corp Penems, pharmaceutical compositions containing them, process for preparing them
DK613984A (da) * 1983-12-30 1985-07-01 Ciba Geigy Ag 2-heterocyclyl-6-hydroxylavalkyl-2-penem-forbindelser samt deres fremstilling og anvendelse
GB8416652D0 (en) * 1984-06-29 1984-08-01 Erba Farmitalia Penem derivatives
US4617300A (en) * 1984-09-21 1986-10-14 Schering Corporation 2(N-heterocyclyl) penems
EP0199675A1 (de) * 1985-04-17 1986-10-29 Ciba-Geigy Ag Heterocyclyl-penem-Verbindungen

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU5378779A (en) * 1978-12-18 1980-08-28 Bristol-Myers Company 2-penem antibiotics
AU8605382A (en) * 1981-07-15 1983-01-20 Sumitomo Chemical Company, Limited Penicillins and azetidinones

Also Published As

Publication number Publication date
US4826832A (en) 1989-05-02
IE871182L (en) 1987-11-06
NZ220195A (en) 1989-01-06
DK228687D0 (da) 1987-05-05
AU7251287A (en) 1987-11-12
JPS62263183A (ja) 1987-11-16
PT84819A (en) 1987-06-01
CA1293502C (en) 1991-12-24
IE59714B1 (en) 1994-03-23
EP0246187B1 (de) 1992-02-05
JPH0339514B2 (enExample) 1991-06-14
ZA873198B (en) 1987-12-30
DK169623B1 (da) 1994-12-27
DE3776590D1 (de) 1992-03-19
ES2038207T3 (es) 1993-07-16
PT84819B (pt) 1989-12-29
DK228687A (da) 1987-11-07
ATE72438T1 (de) 1992-02-15
EP0246187A3 (en) 1988-03-16
GR3003735T3 (enExample) 1993-03-16
EP0246187A2 (de) 1987-11-19

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