DK228687A - 2-pyridyl-penem-forbindelser og salte deraf samt deres fremstilling og anvendelse - Google Patents

2-pyridyl-penem-forbindelser og salte deraf samt deres fremstilling og anvendelse

Info

Publication number
DK228687A
DK228687A DK228687A DK228687A DK228687A DK 228687 A DK228687 A DK 228687A DK 228687 A DK228687 A DK 228687A DK 228687 A DK228687 A DK 228687A DK 228687 A DK228687 A DK 228687A
Authority
DK
Denmark
Prior art keywords
pyridyl
compounds
salts
preparation
penem compounds
Prior art date
Application number
DK228687A
Other languages
English (en)
Other versions
DK169623B1 (da
DK228687D0 (da
Inventor
Marc Lang
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of DK228687D0 publication Critical patent/DK228687D0/da
Publication of DK228687A publication Critical patent/DK228687A/da
Application granted granted Critical
Publication of DK169623B1 publication Critical patent/DK169623B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK228687A 1986-05-06 1987-05-05 2-Pyridyl-penem-forbindelser og salte deraf, fremgangsmåde til deres fremstilling samt farmaceutiske præparater indeholdende disse forbindelser DK169623B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH184686 1986-05-06
CH184686 1986-05-06

Publications (3)

Publication Number Publication Date
DK228687D0 DK228687D0 (da) 1987-05-05
DK228687A true DK228687A (da) 1987-11-07
DK169623B1 DK169623B1 (da) 1994-12-27

Family

ID=4219979

Family Applications (1)

Application Number Title Priority Date Filing Date
DK228687A DK169623B1 (da) 1986-05-06 1987-05-05 2-Pyridyl-penem-forbindelser og salte deraf, fremgangsmåde til deres fremstilling samt farmaceutiske præparater indeholdende disse forbindelser

Country Status (14)

Country Link
US (1) US4826832A (da)
EP (1) EP0246187B1 (da)
JP (1) JPS62263183A (da)
AT (1) ATE72438T1 (da)
AU (1) AU603795B2 (da)
CA (1) CA1293502C (da)
DE (1) DE3776590D1 (da)
DK (1) DK169623B1 (da)
ES (1) ES2038207T3 (da)
GR (1) GR3003735T3 (da)
IE (1) IE59714B1 (da)
NZ (1) NZ220195A (da)
PT (1) PT84819B (da)
ZA (1) ZA873198B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0042026B1 (de) * 1978-02-02 1986-01-08 Ciba-Geigy Ag 3,4-Disubstituierte Azetidin-2-onverbindungen und Verfahren zu ihrer Herstellung
EP0215739B1 (de) * 1985-09-11 1993-09-01 Ciba-Geigy Ag Synthese von Beta-Lactamverbindungen
GB8716679D0 (en) * 1987-07-15 1987-08-19 Erba Farmitalia Penem derivatives
EP0462521A1 (en) * 1990-06-19 1991-12-27 Takeda Chemical Industries, Ltd. Crystalline penem, its production and use
US5492903A (en) * 1990-06-19 1996-02-20 Takeda Chemical Industries Ltd. Crystalline esters of (+)-(5R, 6S)-6-[(R)-1-hydroxyethyl]-3-(3-pyridyl)-7-oxo-4-thia-1-azabicyclo[3.2.0]he
CA2061245A1 (en) * 1991-02-15 1992-08-16 Yoshiharu Maeda Crystalline penem, its production and use
WO1992021304A1 (en) * 1991-06-06 1992-12-10 Cumming Stuart J Intraocular lens with haptic anchor plate
EP0597401A3 (en) * 1992-11-11 1995-07-26 Takeda Chemical Industries Ltd Preparation of penemes.
ATE260120T1 (de) * 1999-10-12 2004-03-15 Daiichi Suntory Pharma Co Ltd Arzneimittel zur oralen verabreichung
US20040202714A1 (en) * 1999-10-12 2004-10-14 Daiichi Suntory Pharma Co., Ltd. Oral pharmaceutical composition

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0042026B1 (de) * 1978-02-02 1986-01-08 Ciba-Geigy Ag 3,4-Disubstituierte Azetidin-2-onverbindungen und Verfahren zu ihrer Herstellung
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
US4272437A (en) * 1978-12-18 1981-06-09 Bristol-Myers Company Antibacterial agents, and 4-thio azetidinone intermediates
IL58576A (en) * 1978-12-18 1985-12-31 Bristol Myers Co 2-substituted and 2,6-disubstituted penem compounds,their preparation and pharmaceutical compositions containing them
US4386030A (en) * 1979-12-31 1983-05-31 Merck & Co., Inc. Process for preparing 6-(1'-hydroxyethyl)-2-substituted-pen-2-em-3-carboxylic acid
EP0180252B1 (en) * 1981-07-15 1989-04-26 Sumitomo Pharmaceuticals Company, Limited Process of preparing azetidinone compounds
NZ201471A (en) * 1981-08-10 1985-09-13 Merck & Co Inc Antibacterial compositions containing penems and dipeptidase inhibitors
DE3366926D1 (en) * 1982-11-16 1986-11-20 Schering Corp Penems, pharmaceutical compositions containing them, process for preparing them
EP0109362A1 (de) * 1982-11-16 1984-05-23 Ciba-Geigy Ag Heterocyclylverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verwendung von letzteren
US4540580A (en) * 1982-11-16 1985-09-10 Schering Corporation 2-[(1'R)-1'-Aminoalkyl]penems
DK613984A (da) * 1983-12-30 1985-07-01 Ciba Geigy Ag 2-heterocyclyl-6-hydroxylavalkyl-2-penem-forbindelser samt deres fremstilling og anvendelse
GB8416652D0 (en) * 1984-06-29 1984-08-01 Erba Farmitalia Penem derivatives
US4617300A (en) * 1984-09-21 1986-10-14 Schering Corporation 2(N-heterocyclyl) penems
EP0199675A1 (de) * 1985-04-17 1986-10-29 Ciba-Geigy Ag Heterocyclyl-penem-Verbindungen

Also Published As

Publication number Publication date
GR3003735T3 (da) 1993-03-16
PT84819B (pt) 1989-12-29
IE59714B1 (en) 1994-03-23
IE871182L (en) 1987-11-06
AU603795B2 (en) 1990-11-29
PT84819A (en) 1987-06-01
US4826832A (en) 1989-05-02
AU7251287A (en) 1987-11-12
CA1293502C (en) 1991-12-24
ZA873198B (en) 1987-12-30
ES2038207T3 (es) 1993-07-16
EP0246187A2 (de) 1987-11-19
DK169623B1 (da) 1994-12-27
NZ220195A (en) 1989-01-06
EP0246187A3 (en) 1988-03-16
DK228687D0 (da) 1987-05-05
JPS62263183A (ja) 1987-11-16
EP0246187B1 (de) 1992-02-05
ATE72438T1 (de) 1992-02-15
JPH0339514B2 (da) 1991-06-14
DE3776590D1 (de) 1992-03-19

Similar Documents

Publication Publication Date Title
NO931056L (no) Sulfonamido- og sulfonamidokarbonyl-pyridin-2-karboksylsyreamider samt deres pyridin-n-oksider, fremgangsmaater for fremstilling derav og anvendelse av forbindelsene som legemidler
CA2075173A1 (en) Compounds and methods for inhibition of hiv and related viruses
NO991206L (no) Benzamidinderivater substituert med sykliske aminosyre- eller sykliske hydroksysyrederivater, og deres anvendelse som antikoagulanter
DK58084A (da) Benzazocinon- og benzazoninonderivater og salte deraf samt deres fremstilling og anvendelse
DK0509398T3 (da) Quinoxaliner, fremgangsmåder til deres fremstilling samt deres anvendelse
DK0888271T3 (da) Benzamidinderivater substitueret med aminosyre- og hydroxysyrederivater og deres anvendelse som antikoagulerende midler
DK228687A (da) 2-pyridyl-penem-forbindelser og salte deraf samt deres fremstilling og anvendelse
IE830607L (en) Imidazolylphenylpyridazinones
GB8607921D0 (en) 3,4-disubstituted-2-azetidinone derivatives
DK0450420T3 (da) Heterocyclisk substituerede dihydropyridiner, fremgangsmåde til deres fremstilling og deres anvendelse i lægemidler
FR2549049B1 (fr) Nouvelles amidines, leur procede de preparation et leur application therapeutique
NO880811L (no) Krystalliserte cefam-syreaddisjonssalter og fremgangsmaatetil deres fremstilling.
MY127758A (en) Derivatives of homopiperidinyl substituted benzimidazole analogues
DK119188D0 (da) Substituerede pyridin-2,4-dicarboxylsyrederivater, fremgangsmaader til deres fremstilling samt laegemiddel indeholdende forbindelserne
DK314483D0 (da) Peenem-derivater, fremgangsmade til fremstilling deraf samt deres anvendelse som laegemidler
DK422688D0 (da) Substituerede pyridylethanolaminer og fysiologisk acceptable salte og n-oxider deraf, deres fremstilling og anvendelse samt mellemprodukter og disses fremstilling
EP0266559A3 (en) Therapeutic agent for the treatment of peptic ulcer disease
DK360584A (da) Triazol-pyrimidinderivater og fremgangsmaade til fremstilling deraf samt disses terapeutiske anvendelse som cardiotoniske midler
FR2529891B1 (da)
DK17581A (da) 2,3-dihydro-imidazo (1,2-b) pyridaziner fremgangsmaade til deres fremstilling samt deres anvendelse
NO880405L (no) Substituerte 3-fenyl-7h-tiazolo(3,2-b)(1,2,4)triazin-7-oner, fremgangsmaate til deres fremstilling og legemidler sominneholder dem, og deres anvendelse samt noen ved fremstillingen av de nevnte forbindelser dannede mellomprod.
DK490282A (da) 1-furyl-3,4-dihydroisoquinoliner, fremgangsmaade til deres fremstilling samt deres anvendelse
DK0413278T3 (da) Anvendelse af xanthinderivater mod mavesår
DK178384A (da) Iminosulfonamider samt deres fremstilling og anvendelse
EP0194164A3 (en) N-carboxyalcoyl-2-oxo-3-diaryl-5,6-triazines useful as therapeutic agents

Legal Events

Date Code Title Description
ATS Application withdrawn
B1 Patent granted (law 1993)
PUP Patent expired