AU573027B2 - 6-(pyrrol-1-yl)pyran-2-one derivatives - Google Patents

6-(pyrrol-1-yl)pyran-2-one derivatives

Info

Publication number
AU573027B2
AU573027B2 AU46867/85A AU4686785A AU573027B2 AU 573027 B2 AU573027 B2 AU 573027B2 AU 46867/85 A AU46867/85 A AU 46867/85A AU 4686785 A AU4686785 A AU 4686785A AU 573027 B2 AU573027 B2 AU 573027B2
Authority
AU
Australia
Prior art keywords
pyrrol
pyran
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU46867/85A
Other languages
English (en)
Other versions
AU4686785A (en
Inventor
Milton Louis Hoefle
Bruce D. Roth
Charlotte D. Stratton
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Warner Lambert Co LLC
Original Assignee
Warner Lambert Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co LLC filed Critical Warner Lambert Co LLC
Publication of AU4686785A publication Critical patent/AU4686785A/en
Application granted granted Critical
Publication of AU573027B2 publication Critical patent/AU573027B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
AU46867/85A 1984-09-24 1985-08-29 6-(pyrrol-1-yl)pyran-2-one derivatives Ceased AU573027B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US65379884A 1984-09-24 1984-09-24
US653798 1984-09-24
US679676 1984-12-10
US06/679,676 US4647576A (en) 1984-09-24 1984-12-10 Trans-6-[2-(substitutedpyrrol-1-yl)alkyl]-pyran-2-one inhibitors of cholesterol synthesis

Publications (2)

Publication Number Publication Date
AU4686785A AU4686785A (en) 1986-04-10
AU573027B2 true AU573027B2 (en) 1988-05-26

Family

ID=27096596

Family Applications (1)

Application Number Title Priority Date Filing Date
AU46867/85A Ceased AU573027B2 (en) 1984-09-24 1985-08-29 6-(pyrrol-1-yl)pyran-2-one derivatives

Country Status (12)

Country Link
US (1) US4647576A (enExample)
EP (1) EP0179559A3 (enExample)
KR (2) KR890001449B1 (enExample)
AU (1) AU573027B2 (enExample)
CA (1) CA1242721A (enExample)
DK (1) DK430485A (enExample)
ES (1) ES8701756A1 (enExample)
FI (1) FI853632L (enExample)
GR (1) GR852297B (enExample)
NO (1) NO853725L (enExample)
NZ (1) NZ213252A (enExample)
PT (1) PT81179B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU601981B2 (en) * 1986-05-30 1990-09-27 Warner-Lambert Company Llc Trans- (2-(3 or 4-carboxamido-substituted pyrrol-1-yl) alkyl)-4-hydroxypyran-2-one inhibitors of cholesterol synthesis

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US4647576A (en) 1987-03-03
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KR860002503A (ko) 1986-04-26
ES8701756A1 (es) 1986-12-01
KR890001449B1 (en) 1989-05-03
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PT81179B (en) 1987-02-13
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NO853725L (no) 1986-03-25
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