AU467361B2 - Q-aryl-4-substituted piperidinoalkanol derivatives - Google Patents

Q-aryl-4-substituted piperidinoalkanol derivatives

Info

Publication number
AU467361B2
AU467361B2 AU49893/72A AU4989372A AU467361B2 AU 467361 B2 AU467361 B2 AU 467361B2 AU 49893/72 A AU49893/72 A AU 49893/72A AU 4989372 A AU4989372 A AU 4989372A AU 467361 B2 AU467361 B2 AU 467361B2
Authority
AU
Australia
Prior art keywords
aryl
piperidinoalkanol derivatives
substituted
substituted piperidinoalkanol
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU49893/72A
Other languages
English (en)
Other versions
AU4989372A (en
Inventor
and CLYDE RICHARD KINSOLVING ALBERT ANTHONY CARR
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Merrell Dow Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22829539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU467361(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merrell Dow Pharmaceuticals Inc filed Critical Merrell Dow Pharmaceuticals Inc
Publication of AU4989372A publication Critical patent/AU4989372A/en
Application granted granted Critical
Publication of AU467361B2 publication Critical patent/AU467361B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU49893/72A 1972-01-28 1972-12-11 Q-aryl-4-substituted piperidinoalkanol derivatives Ceased AU467361B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22182172A 1972-01-28 1972-01-28
USUS221,821 1972-01-28

Publications (2)

Publication Number Publication Date
AU4989372A AU4989372A (en) 1974-06-13
AU467361B2 true AU467361B2 (en) 1975-11-27

Family

ID=22829539

Family Applications (1)

Application Number Title Priority Date Filing Date
AU49893/72A Ceased AU467361B2 (en) 1972-01-28 1972-12-11 Q-aryl-4-substituted piperidinoalkanol derivatives

Country Status (26)

Country Link
JP (1) JPS5115035B2 (ja)
AR (1) AR195314A1 (ja)
AT (2) AT323742B (ja)
AU (1) AU467361B2 (ja)
BE (1) BE794597A (ja)
CA (1) CA978946A (ja)
CH (2) CH587820A5 (ja)
CS (1) CS177834B2 (ja)
DD (1) DD103239A5 (ja)
DE (1) DE2303306C3 (ja)
DK (1) DK136713B (ja)
ES (1) ES410731A1 (ja)
FR (1) FR2181690B1 (ja)
GB (1) GB1413138A (ja)
HU (1) HU166477B (ja)
IE (1) IE36983B1 (ja)
IL (1) IL41060A (ja)
LU (1) LU66916A1 (ja)
NL (1) NL175410C (ja)
NO (1) NO140057C (ja)
PH (1) PH10264A (ja)
PL (1) PL89095B1 (ja)
SE (1) SE382058B (ja)
SU (1) SU464997A3 (ja)
YU (1) YU36013B (ja)
ZA (1) ZA728544B (ja)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3941795A (en) 1974-02-08 1976-03-02 Richardson-Merrell Inc. α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES
US4254129A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
US4254130A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
IT1200123B (it) * 1985-09-27 1989-01-05 Ind Chimica Srl Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo
US4742175A (en) * 1986-05-07 1988-05-03 Merrell Dow Pharmaceuticals Inc. Preparation of polymorphically pure terfenadine
JPS63101760U (ja) * 1986-12-19 1988-07-02
IT1205685B (it) * 1987-05-26 1989-03-31 Erregierre Spa Processo per la preparazione di alfa-(alchilfenil)-4-(idrossi difenilmetil)-1-piperidina butanolo
ZA901360B (en) * 1989-02-28 1990-11-28 Merrell Dow Pharma Preparation of the low-melting polymorphic form of terfenadine
CA2015390A1 (en) * 1989-05-01 1990-11-01 Frederick J. Mccarty Process for the preparation of the high melting polymorphic of terfenadine
DE3917241A1 (de) * 1989-05-26 1990-11-29 Schaper & Bruemmer Gmbh 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate
US5466691A (en) * 1991-08-09 1995-11-14 Yoshitomi Pharmaceutical Industries, Ltd. Thiophene compound
KR19990008406A (ko) * 1995-05-08 1999-01-25 스티븐엘.네스비트 알파-(치환된 알킬페닐)-4-(히드록시디페닐메틸)-1-피페리딘 부탄올 유도체들, 그들의 제조 방법 및 항히스타민제, 항알러지제및 기관지 확장제로서 그들의 용도
EP0864653B1 (de) * 1997-03-11 2004-03-03 Aventis Pharmaceuticals Inc. Verfahren zur Herstellung von 4-(4-(4-(Hydroxydiphenyl)-1-piperidinyl)-1-hydroxybutyl)-alpha,alpha-dimenthylphenylessigsäure und phosphorylierter Derivate
US7498345B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of piperidine derivatives
US8153385B2 (en) 2004-10-18 2012-04-10 Reverse Proteomics Research Institute Co., Ltd. Target protein and target gene in drug designing and screening method

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3081303A (en) * 1961-10-13 1963-03-12 Searle & Co 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols
GB1242169A (en) * 1969-04-09 1971-08-11 Ucb Sa Piperidine derivatives

Also Published As

Publication number Publication date
DK136713C (ja) 1978-05-01
FR2181690B1 (ja) 1976-05-14
SE382058B (sv) 1976-01-12
AU4989372A (en) 1974-06-13
DE2303306B2 (de) 1978-09-28
HU166477B (ja) 1975-03-28
IL41060A (en) 1975-06-25
NL175410C (nl) 1984-11-01
CH593259A5 (ja) 1977-11-30
YU3473A (en) 1981-02-28
NL175410B (nl) 1984-06-01
IE36983B1 (en) 1977-04-13
SU464997A3 (ru) 1975-03-25
CH587820A5 (ja) 1977-05-13
JPS4885578A (ja) 1973-11-13
AR195314A1 (es) 1973-09-28
IL41060A0 (en) 1973-02-28
PL89095B1 (ja) 1976-10-30
FR2181690A1 (ja) 1973-12-07
ZA728544B (en) 1974-02-27
LU66916A1 (ja) 1973-07-27
GB1413138A (en) 1975-11-05
YU36013B (en) 1981-11-13
DE2303306A1 (de) 1973-08-02
AT321917B (de) 1975-04-25
DK136713B (da) 1977-11-14
DD103239A5 (ja) 1974-01-12
BE794597A (fr) 1973-05-16
IE36983L (en) 1973-07-28
NO140057B (no) 1979-03-19
DE2303306C3 (de) 1979-05-31
NL7300873A (ja) 1973-07-31
NO140057C (no) 1979-07-04
JPS5115035B2 (ja) 1976-05-13
CS177834B2 (ja) 1977-08-31
CA978946A (en) 1975-12-02
PH10264A (en) 1976-10-20
ES410731A1 (es) 1976-04-01
AT323742B (de) 1975-07-25

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