AU2020346057A1 - Thyroid hormone receptor beta agonist compounds - Google Patents

Thyroid hormone receptor beta agonist compounds Download PDF

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Publication number
AU2020346057A1
AU2020346057A1 AU2020346057A AU2020346057A AU2020346057A1 AU 2020346057 A1 AU2020346057 A1 AU 2020346057A1 AU 2020346057 A AU2020346057 A AU 2020346057A AU 2020346057 A AU2020346057 A AU 2020346057A AU 2020346057 A1 AU2020346057 A1 AU 2020346057A1
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AU
Australia
Prior art keywords
alkyl
compound
groups
pharmaceutically acceptable
acceptable salt
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Pending
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AU2020346057A
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English (en)
Inventor
Randall HALCOMB
Thorsten A. Kirschberg
F. Anthony Romero
Yingzi XU
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Terns Pharmaceuticals Inc
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Terns Pharmaceuticals Inc
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Application filed by Terns Pharmaceuticals Inc filed Critical Terns Pharmaceuticals Inc
Publication of AU2020346057A1 publication Critical patent/AU2020346057A1/en
Pending legal-status Critical Current

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/14Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2020346057A 2019-09-12 2020-09-11 Thyroid hormone receptor beta agonist compounds Pending AU2020346057A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962899581P 2019-09-12 2019-09-12
US62/899,581 2019-09-12
PCT/US2020/050497 WO2021050945A1 (en) 2019-09-12 2020-09-11 Thyroid hormone receptor beta agonist compounds

Publications (1)

Publication Number Publication Date
AU2020346057A1 true AU2020346057A1 (en) 2022-04-21

Family

ID=74866716

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2020346057A Pending AU2020346057A1 (en) 2019-09-12 2020-09-11 Thyroid hormone receptor beta agonist compounds

Country Status (7)

Country Link
US (1) US12398127B2 (https=)
EP (1) EP4028008A4 (https=)
JP (2) JP2022548250A (https=)
CN (1) CN114375193B (https=)
AU (1) AU2020346057A1 (https=)
CA (1) CA3154391A1 (https=)
WO (1) WO2021050945A1 (https=)

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Also Published As

Publication number Publication date
EP4028008A1 (en) 2022-07-20
JP2026027279A (ja) 2026-02-18
CN114375193B (zh) 2024-05-14
US12398127B2 (en) 2025-08-26
CN114375193A (zh) 2022-04-19
WO2021050945A1 (en) 2021-03-18
JP2022548250A (ja) 2022-11-17
US20220356177A1 (en) 2022-11-10
CA3154391A1 (en) 2021-03-18
EP4028008A4 (en) 2023-09-13

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