AU2019249562B2 - Oxazole compound crystal - Google Patents

Oxazole compound crystal Download PDF

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Publication number
AU2019249562B2
AU2019249562B2 AU2019249562A AU2019249562A AU2019249562B2 AU 2019249562 B2 AU2019249562 B2 AU 2019249562B2 AU 2019249562 A AU2019249562 A AU 2019249562A AU 2019249562 A AU2019249562 A AU 2019249562A AU 2019249562 B2 AU2019249562 B2 AU 2019249562B2
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AU
Australia
Prior art keywords
crystal
type
compound
peaks
ointment
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
AU2019249562A
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English (en)
Other versions
AU2019249562A1 (en
Inventor
Ryosuke HIROTA
Naohiko KANAI
Takayuki YASUTOMI
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Otsuka Pharmaceutical Co Ltd
Original Assignee
Otsuka Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharmaceutical Co Ltd filed Critical Otsuka Pharmaceutical Co Ltd
Publication of AU2019249562A1 publication Critical patent/AU2019249562A1/en
Application granted granted Critical
Publication of AU2019249562B2 publication Critical patent/AU2019249562B2/en
Priority to AU2024220015A priority Critical patent/AU2024220015A1/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2019249562A 2018-04-04 2019-04-03 Oxazole compound crystal Active AU2019249562B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2024220015A AU2024220015A1 (en) 2018-04-04 2024-09-24 Oxazole compound crystal

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2018072717 2018-04-04
JP2018-072717 2018-04-04
PCT/JP2019/014730 WO2019194211A1 (en) 2018-04-04 2019-04-03 Oxazole compound crystal

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2024220015A Division AU2024220015A1 (en) 2018-04-04 2024-09-24 Oxazole compound crystal

Publications (2)

Publication Number Publication Date
AU2019249562A1 AU2019249562A1 (en) 2020-10-22
AU2019249562B2 true AU2019249562B2 (en) 2024-06-27

Family

ID=66223774

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2019249562A Active AU2019249562B2 (en) 2018-04-04 2019-04-03 Oxazole compound crystal
AU2024220015A Pending AU2024220015A1 (en) 2018-04-04 2024-09-24 Oxazole compound crystal

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2024220015A Pending AU2024220015A1 (en) 2018-04-04 2024-09-24 Oxazole compound crystal

Country Status (26)

Country Link
US (4) US11414391B2 (enExample)
EP (2) EP4400167A3 (enExample)
JP (4) JP7326295B2 (enExample)
KR (2) KR102764726B1 (enExample)
CN (1) CN111902402A (enExample)
AU (2) AU2019249562B2 (enExample)
BR (1) BR112020019377A2 (enExample)
CA (1) CA3095866A1 (enExample)
DK (1) DK3774745T3 (enExample)
EA (1) EA202092393A1 (enExample)
ES (1) ES2982586T3 (enExample)
FI (1) FI3774745T3 (enExample)
HR (1) HRP20240858T1 (enExample)
HU (1) HUE066793T2 (enExample)
IL (2) IL277730B2 (enExample)
LT (1) LT3774745T (enExample)
MX (1) MX2020010435A (enExample)
MY (1) MY202406A (enExample)
PH (1) PH12020551605A1 (enExample)
PL (1) PL3774745T3 (enExample)
PT (1) PT3774745T (enExample)
SG (1) SG11202009564TA (enExample)
SI (1) SI3774745T1 (enExample)
TW (2) TWI860993B (enExample)
WO (1) WO2019194211A1 (enExample)
ZA (1) ZA202006134B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK3774745T3 (da) * 2018-04-04 2024-06-17 Otsuka Pharma Co Ltd Krystal af en oxazolforbindelse
EP4501324A1 (en) 2022-03-25 2025-02-05 Otsuka Pharmaceutical Co., Ltd. Wound treatment composition
CN115887463A (zh) * 2022-12-27 2023-04-04 瑞石生物医药有限公司 一种含环酰胺化合物的药物组合物
GB202306663D0 (en) 2023-05-05 2023-06-21 Union Therapeutics As Combination therapy

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI330639B (en) * 2005-11-15 2010-09-21 Otsuka Pharma Co Ltd Oxazole compound and pharmaceutical composition
WO2014034958A1 (en) * 2012-08-30 2014-03-06 Otsuka Pharmaceutical Co., Ltd. Method for producing oxazole compound
TWI726027B (zh) 2015-12-28 2021-05-01 日商大塚製藥股份有限公司 軟膏
DK3774745T3 (da) * 2018-04-04 2024-06-17 Otsuka Pharma Co Ltd Krystal af en oxazolforbindelse

Also Published As

Publication number Publication date
KR20250022254A (ko) 2025-02-14
US11414391B2 (en) 2022-08-16
EP3774745B1 (en) 2024-05-29
BR112020019377A2 (pt) 2021-01-05
DK3774745T3 (da) 2024-06-17
US20210147370A1 (en) 2021-05-20
MY202406A (en) 2024-04-27
CN111902402A (zh) 2020-11-06
ES2982586T3 (es) 2024-10-16
TWI860993B (zh) 2024-11-11
EP3774745A1 (en) 2021-02-17
AU2024220015A1 (en) 2024-10-17
JP7326295B2 (ja) 2023-08-15
CA3095866A1 (en) 2019-10-10
WO2019194211A1 (en) 2019-10-10
US20220411386A1 (en) 2022-12-29
TW202515853A (zh) 2025-04-16
ZA202006134B (en) 2023-03-29
TW202012380A (zh) 2020-04-01
HUE066793T2 (hu) 2024-09-28
KR20200139736A (ko) 2020-12-14
MX2020010435A (es) 2020-10-28
SI3774745T1 (sl) 2024-08-30
EP4400167A3 (en) 2024-09-25
FI3774745T3 (fi) 2024-06-19
JP2025128238A (ja) 2025-09-02
IL277730B2 (en) 2025-02-01
PL3774745T3 (pl) 2024-08-19
SG11202009564TA (en) 2020-10-29
US20250250243A1 (en) 2025-08-07
JP2021517111A (ja) 2021-07-15
PT3774745T (pt) 2024-06-25
IL277730A (en) 2020-11-30
EP4400167A2 (en) 2024-07-17
IL277730B1 (en) 2024-10-01
LT3774745T (lt) 2024-07-10
JP2022037040A (ja) 2022-03-08
HRP20240858T1 (hr) 2024-10-11
PH12020551605A1 (en) 2021-04-26
KR102764726B1 (ko) 2025-02-11
IL315425A (en) 2024-11-01
US11840512B2 (en) 2023-12-12
AU2019249562A1 (en) 2020-10-22
EA202092393A1 (ru) 2021-01-25
JP2024001115A (ja) 2024-01-09
US20240076275A1 (en) 2024-03-07

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