AU2015360364B2 - GLP-1 receptor modulators - Google Patents

GLP-1 receptor modulators Download PDF

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Publication number
AU2015360364B2
AU2015360364B2 AU2015360364A AU2015360364A AU2015360364B2 AU 2015360364 B2 AU2015360364 B2 AU 2015360364B2 AU 2015360364 A AU2015360364 A AU 2015360364A AU 2015360364 A AU2015360364 A AU 2015360364A AU 2015360364 B2 AU2015360364 B2 AU 2015360364B2
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Australia
Prior art keywords
certain embodiments
compound
butyl
compounds
phenyl
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AU2015360364A
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AU2015360364A1 (en
Inventor
Marcus F. Boehm
Enugurthi Brahmachary
Thomas Fowler
Daniel Glynn
Liming Huang
Michael Knaggs
Esther Martinborough
Premji Meghani
Mark Mills
Manisha Moorjani
Andrew Novak
Junko Tamiya
Adam R. Yeager
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Receptos LLC
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Receptos LLC
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Assigned to RECEPTOS LLC reassignment RECEPTOS LLC Request for Assignment Assignors: CELGENE INTERNATIONAL II SARL
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    • C—CHEMISTRY; METALLURGY
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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/26—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
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