AU2014367781B2 - Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain - Google Patents

Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain Download PDF

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Publication number
AU2014367781B2
AU2014367781B2 AU2014367781A AU2014367781A AU2014367781B2 AU 2014367781 B2 AU2014367781 B2 AU 2014367781B2 AU 2014367781 A AU2014367781 A AU 2014367781A AU 2014367781 A AU2014367781 A AU 2014367781A AU 2014367781 B2 AU2014367781 B2 AU 2014367781B2
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AU
Australia
Prior art keywords
pain
dihydro
inden
sulfamide
mmol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
AU2014367781A
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English (en)
Other versions
AU2014367781A1 (en
Inventor
Keisuke Hashimoto
Hiroyuki Higashiyama
Yuji Kazuta
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eisai R&D Management Co Ltd
Original Assignee
Eisai R&D Management Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Management Co Ltd filed Critical Eisai R&D Management Co Ltd
Publication of AU2014367781A1 publication Critical patent/AU2014367781A1/en
Application granted granted Critical
Publication of AU2014367781B2 publication Critical patent/AU2014367781B2/en
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Anticipated expiration legal-status Critical

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0021Intradermal administration, e.g. through microneedle arrays, needleless injectors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
AU2014367781A 2013-12-19 2014-12-17 Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain Active AU2014367781B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2013262743 2013-12-19
JP2013-262743 2013-12-19
PCT/JP2014/083374 WO2015093515A1 (ja) 2013-12-19 2014-12-17 1-インダンスルファミド誘導体を含む疼痛の治療および/または予防剤

Publications (2)

Publication Number Publication Date
AU2014367781A1 AU2014367781A1 (en) 2016-06-23
AU2014367781B2 true AU2014367781B2 (en) 2019-07-04

Family

ID=53402860

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2014367781A Active AU2014367781B2 (en) 2013-12-19 2014-12-17 Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain

Country Status (14)

Country Link
US (1) US9610262B2 (enExample)
EP (1) EP3085369B1 (enExample)
JP (1) JP6518595B2 (enExample)
KR (1) KR102250214B1 (enExample)
CN (1) CN105792821B (enExample)
AU (1) AU2014367781B2 (enExample)
BR (1) BR112016012833B1 (enExample)
CA (1) CA2932529C (enExample)
ES (1) ES2673876T3 (enExample)
IL (1) IL246036B (enExample)
MX (1) MX370898B (enExample)
RU (1) RU2678571C1 (enExample)
SG (1) SG11201604484UA (enExample)
WO (1) WO2015093515A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11660275B2 (en) * 2018-03-20 2023-05-30 Eisai R&D Management Co., Ltd. Epilepsy treatment agent
KR20250005086A (ko) 2022-04-27 2025-01-09 에자이 알앤드디 매니지먼트 가부시키가이샤 파킨슨병의 치료를 위한 약학적 조성물
KR102803991B1 (ko) 2022-11-11 2025-05-13 덕산에테르씨티 주식회사 내화성능 및 강도가 보강된 압력용기
KR102815520B1 (ko) 2022-11-11 2025-06-04 덕산에테르씨티 주식회사 내화성능 및 강도가 보강된 압력용기
KR102815521B1 (ko) 2022-11-11 2025-06-04 덕산에테르씨티 주식회사 내화성능 및 강도가 보강된 압력용기
KR20250063588A (ko) 2023-11-01 2025-05-08 덕산에테르씨티 주식회사 압력 용기의 숄더부 보호용 커버
KR20250063587A (ko) 2023-11-01 2025-05-08 덕산에테르씨티 주식회사 압력 용기의 숄더부 보호용 커버
KR20250063589A (ko) 2023-11-01 2025-05-08 덕산에테르씨티 주식회사 압력 용기의 숄더부 보호용 커버

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013191144A1 (ja) * 2012-06-21 2013-12-27 エーザイ・アール・アンド・ディー・マネジメント株式会社 新規インダンスルファミド誘導体

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8716231B2 (en) * 2005-12-19 2014-05-06 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
US20070191452A1 (en) * 2006-02-15 2007-08-16 Smith-Swintosky Virginia L Use of benzo-heteroaryl sulfamide derivatives for the treatment of pain
CL2007002994A1 (es) 2006-10-19 2008-02-08 Wyeth Corp Compuestos derivados heterociclicos que contienen sulfamoilo, inhibidores de hsp90; composicion farmaceutica; y uso para el tratamiento del cancer, tal como cancer de mama, de colon y prostata, entre otros.
TWI433674B (zh) 2006-12-28 2014-04-11 Infinity Discovery Inc 環杷明(cyclopamine)類似物類
EP2417101B1 (en) 2009-04-09 2013-10-23 Merck Sharp & Dohme B.V. Indane derivatives
TW201217312A (en) * 2010-09-22 2012-05-01 Gruenenthal Gmbh Substituted benzamide compounds
RU2508295C2 (ru) * 2012-03-22 2014-02-27 Общество с ограниченной ответственностью "Биофармокс" Синтетические пептиды с ненаркотическим типом анальгетического действия

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013191144A1 (ja) * 2012-06-21 2013-12-27 エーザイ・アール・アンド・ディー・マネジメント株式会社 新規インダンスルファミド誘導体

Also Published As

Publication number Publication date
ES2673876T3 (es) 2018-06-26
CN105792821B (zh) 2018-05-04
CA2932529C (en) 2022-03-22
CN105792821A (zh) 2016-07-20
EP3085369B1 (en) 2018-04-04
EP3085369A1 (en) 2016-10-26
IL246036B (en) 2018-11-29
CA2932529A1 (en) 2015-06-25
US20160303058A1 (en) 2016-10-20
BR112016012833B1 (pt) 2022-11-16
WO2015093515A1 (ja) 2015-06-25
SG11201604484UA (en) 2016-07-28
KR102250214B1 (ko) 2021-05-07
JP6518595B2 (ja) 2019-05-22
JPWO2015093515A1 (ja) 2017-03-23
AU2014367781A1 (en) 2016-06-23
KR20160106053A (ko) 2016-09-09
RU2678571C1 (ru) 2019-01-30
EP3085369A4 (en) 2017-05-10
US9610262B2 (en) 2017-04-04
IL246036A0 (en) 2016-07-31
MX370898B (es) 2020-01-09
BR112016012833A2 (enExample) 2017-08-08
MX2016007370A (es) 2016-10-03
RU2016122189A (ru) 2018-01-24

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