AU2013304133B2 - Azaindole carboxylic acid amides and azaindole thiocarboxylic acid amides for use as insecticides and acaricides - Google Patents

Azaindole carboxylic acid amides and azaindole thiocarboxylic acid amides for use as insecticides and acaricides Download PDF

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Publication number
AU2013304133B2
AU2013304133B2 AU2013304133A AU2013304133A AU2013304133B2 AU 2013304133 B2 AU2013304133 B2 AU 2013304133B2 AU 2013304133 A AU2013304133 A AU 2013304133A AU 2013304133 A AU2013304133 A AU 2013304133A AU 2013304133 B2 AU2013304133 B2 AU 2013304133B2
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AU
Australia
Prior art keywords
spp
methyl
formula
ethyl
compounds
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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AU2013304133A
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English (en)
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AU2013304133A1 (en
Inventor
Roland Andree
Ulrich Goergens
Markus Heil
Eike Kevin Heilmann
Kerstin Ilg
Peter Jeschke
Matthias RIEDRICH
Arnd Voerste
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Bayer CropScience AG
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Bayer CropScience AG
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Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Publication of AU2013304133A1 publication Critical patent/AU2013304133A1/en
Application granted granted Critical
Publication of AU2013304133B2 publication Critical patent/AU2013304133B2/en
Expired - Fee Related legal-status Critical Current
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N53/00—Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
AU2013304133A 2012-08-17 2013-08-13 Azaindole carboxylic acid amides and azaindole thiocarboxylic acid amides for use as insecticides and acaricides Expired - Fee Related AU2013304133B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12180826.5 2012-08-17
EP12180826 2012-08-17
PCT/EP2013/066905 WO2014026984A1 (de) 2012-08-17 2013-08-13 Azaindolcarbonsäure- und -thiocarbonsäureamide als insektizide und akarizide

Publications (2)

Publication Number Publication Date
AU2013304133A1 AU2013304133A1 (en) 2015-02-26
AU2013304133B2 true AU2013304133B2 (en) 2017-02-23

Family

ID=46940225

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2013304133A Expired - Fee Related AU2013304133B2 (en) 2012-08-17 2013-08-13 Azaindole carboxylic acid amides and azaindole thiocarboxylic acid amides for use as insecticides and acaricides

Country Status (17)

Country Link
US (1) US9345247B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP2885301A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JP2015530990A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR20150044895A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN104718206B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU2013304133B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR112015003098A2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2881995A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CL (1) CL2015000336A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CO (1) CO7200270A2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IN (1) IN2015DN01061A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX2015001897A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PE (1) PE20150634A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PH (1) PH12015500334A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
RU (1) RU2015109064A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
WO (1) WO2014026984A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (1) ZA201501211B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

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US8957078B2 (en) 2013-03-15 2015-02-17 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
WO2014143240A1 (en) 2013-03-15 2014-09-18 Vertex Pharmaceuticals Incorporated Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase
US8969360B2 (en) 2013-03-15 2015-03-03 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
SG11201604519PA (en) 2013-12-06 2016-07-28 Vertex Pharma 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, its preparation, different solid forms and radiolabelled derivatives thereof
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WO2015187451A1 (en) 2014-06-05 2015-12-10 Vertex Pharmacetucals Incorporated Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof
SG10201811175WA (en) 2014-06-17 2019-01-30 Vertex Pharma Method for treating cancer using a combination of chk1 and atr inhibitors
CN104974075A (zh) * 2015-08-07 2015-10-14 新秀化学（烟台）有限公司 一种n, n-二(2,2,6,6-四甲基-4-哌啶基) -1,3-苯二甲酰胺的制备方法
KR102678021B1 (ko) 2015-09-30 2024-06-26 버텍스 파마슈티칼스 인코포레이티드 Dna 손상제와 병용되는, atr 저해제를 포함하는 암 치료용 약제학적 조성물
US12084472B2 (en) 2015-12-18 2024-09-10 Ardelyx, Inc. Substituted 4-phenyl pyridine compounds as non-systemic TGR5 agonists
TW202246215A (zh) 2015-12-18 2022-12-01 美商亞德利克斯公司 作為非全身ｔｇｒ５促效劑之經取代之４－苯基吡啶化合物
CN107094790A (zh) * 2017-06-12 2017-08-29 刘鸿宇 一种具有协同杀虫作用的农药组合物
EP4034108A4 (en) * 2019-09-26 2023-09-13 The Global Alliance for TB Drug Development, Inc. AZAINDOLE CARBOXAMIDE COMPOUNDS FOR THE TREATMENT OF MYCOBACTERIAL INFECTIONS

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Also Published As

Publication number Publication date
PH12015500334A1 (en) 2015-04-20
IN2015DN01061A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 2015-06-26
EP2885301A1 (de) 2015-06-24
US9345247B2 (en) 2016-05-24
CO7200270A2 (es) 2015-02-27
WO2014026984A1 (de) 2014-02-20
RU2015109064A (ru) 2016-10-10
CN104718206B (zh) 2017-03-08
PE20150634A1 (es) 2015-05-08
MX2015001897A (es) 2015-05-11
US20150216175A1 (en) 2015-08-06
CA2881995A1 (en) 2014-02-20
JP2015530990A (ja) 2015-10-29
CL2015000336A1 (es) 2015-06-26
KR20150044895A (ko) 2015-04-27
ZA201501211B (en) 2016-10-26
CN104718206A (zh) 2015-06-17
AU2013304133A1 (en) 2015-02-26
BR112015003098A2 (pt) 2017-08-22

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