AU2013221613A1 - Solid forms comprising inhibitors of HCV NS5A, compositions thereof, and uses therewith - Google Patents
Solid forms comprising inhibitors of HCV NS5A, compositions thereof, and uses therewith Download PDFInfo
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- AU2013221613A1 AU2013221613A1 AU2013221613A AU2013221613A AU2013221613A1 AU 2013221613 A1 AU2013221613 A1 AU 2013221613A1 AU 2013221613 A AU2013221613 A AU 2013221613A AU 2013221613 A AU2013221613 A AU 2013221613A AU 2013221613 A1 AU2013221613 A1 AU 2013221613A1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261598249P | 2012-02-13 | 2012-02-13 | |
| US61/598,249 | 2012-02-13 | ||
| PCT/US2013/025995 WO2013123092A1 (en) | 2012-02-13 | 2013-02-13 | Solid forms comprising inhibitors of hcv ns5a, compositions thereof, and uses therewith |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2013221613A1 true AU2013221613A1 (en) | 2014-09-04 |
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| AU2013221613A Abandoned AU2013221613A1 (en) | 2012-02-13 | 2013-02-13 | Solid forms comprising inhibitors of HCV NS5A, compositions thereof, and uses therewith |
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| US9717712B2 (en) | 2013-07-02 | 2017-08-01 | Bristol-Myers Squibb Company | Combinations comprising tricyclohexadecahexaene derivatives for use in the treatment of hepatitis C virus |
| US20150023913A1 (en) | 2013-07-02 | 2015-01-22 | Bristol-Myers Squibb Company | Hepatitis C Virus Inhibitors |
| WO2015009744A1 (en) | 2013-07-17 | 2015-01-22 | Bristol-Myers Squibb Company | Combinations comprising biphenyl derivatives for use in the treatment of hcv |
| TWI679203B (zh) | 2014-06-11 | 2019-12-11 | 美商基利法瑪席特有限責任公司 | 製備抗病毒化合物之方法 |
| ITUB20152784A1 (it) * | 2015-08-03 | 2017-02-03 | Chemelectiva S R L | Processo per la sintesi di ravidasvir |
| US10617675B2 (en) | 2015-08-06 | 2020-04-14 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| CN109134439A (zh) * | 2017-06-15 | 2019-01-04 | 歌礼生物科技（杭州）有限公司 | 丙肝治疗药物Ravidasvir的制备方法 |
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| GB2438802A (en) * | 2005-02-28 | 2007-12-05 | Univ Rockefeller | Structure of the hepatitis C virus NS5A protein |
| KR101784830B1 (ko) * | 2008-12-03 | 2017-10-16 | 프레시디오 파마슈티칼스, 인코포레이티드 | Ｈｃｖ ｎｓ5ａ의 억제제 |
| CN102427731B (zh) * | 2009-02-27 | 2015-05-13 | 英安塔制药有限公司 | 丙型肝炎病毒抑制剂 |
| WO2011004276A1 (en) * | 2009-07-06 | 2011-01-13 | Pfizer Limited | Hepatitis c virus inhibitors |
| UA108211C2 (uk) * | 2009-11-04 | 2015-04-10 | Янссен Рід Айрленд | Бензімідазолімідазольні похідні |
| KR20120124495A (ko) * | 2010-03-04 | 2012-11-13 | 이난타 파마슈티칼스, 인코포레이티드 | Ｈｃｖ 복제의 억제제로서의 조합 제약 작용제 |
| EP2575866A4 (en) * | 2010-05-24 | 2013-10-16 | Presidio Pharmaceuticals Inc | HCV NS5A INHIBITORS |
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2013
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- 2013-02-13 BR BR112014019585A patent/BR112014019585A8/pt not_active IP Right Cessation
- 2013-02-13 PE PE2014001253A patent/PE20142462A1/es not_active Application Discontinuation
- 2013-02-13 KR KR1020147025614A patent/KR20140145126A/ko not_active Withdrawn
- 2013-02-13 EP EP13749094.2A patent/EP2814322A4/en not_active Withdrawn
- 2013-02-13 CN CN201380019234.4A patent/CN104219953A/zh active Pending
- 2013-02-13 US US14/377,846 patent/US20150203474A1/en not_active Abandoned
- 2013-02-13 EA EA201491442A patent/EA201491442A1/ru unknown
- 2013-02-13 SG SG11201404754TA patent/SG11201404754TA/en unknown
- 2013-02-13 WO PCT/US2013/025995 patent/WO2013123092A1/en not_active Ceased
- 2013-02-13 IN IN1671MUN2014 patent/IN2014MN01671A/en unknown
- 2013-02-13 AR ARP130100443A patent/AR093738A1/es unknown
- 2013-02-13 MX MX2014009693A patent/MX2014009693A/es unknown
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- 2013-02-18 TW TW102105671A patent/TW201339153A/zh unknown
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- 2014-09-11 ZA ZA2014/06740A patent/ZA201406740B/en unknown
- 2014-09-11 CO CO14201398A patent/CO7061084A2/es unknown
Also Published As
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| CL2014002138A1 (es) | 2014-11-28 |
| MX2014009693A (es) | 2014-09-08 |
| HK1204433A1 (en) | 2015-11-20 |
| EA201491442A1 (ru) | 2015-01-30 |
| PE20142462A1 (es) | 2015-02-01 |
| US20150203474A1 (en) | 2015-07-23 |
| EP2814322A1 (en) | 2014-12-24 |
| CO7061084A2 (es) | 2014-09-19 |
| SG11201404754TA (en) | 2014-09-26 |
| CN104219953A (zh) | 2014-12-17 |
| TW201339153A (zh) | 2013-10-01 |
| ZA201406740B (en) | 2016-02-24 |
| KR20140145126A (ko) | 2014-12-22 |
| CA2864342A1 (en) | 2013-08-22 |
| IN2014MN01671A (enExample) | 2015-05-29 |
| JP2015506987A (ja) | 2015-03-05 |
| WO2013123092A1 (en) | 2013-08-22 |
| BR112014019585A8 (pt) | 2017-07-11 |
| AR093738A1 (es) | 2015-06-24 |
| EP2814322A4 (en) | 2015-09-23 |
| PH12014501781A1 (en) | 2014-11-10 |
| BR112014019585A2 (enExample) | 2017-06-20 |
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| Date | Code | Title | Description |
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| MK5 | Application lapsed section 142(2)(e) - patent request and compl. specification not accepted |