AU2012295802B2 - Tricyclic heterocyclic compounds and JAK inhibitors - Google Patents

Tricyclic heterocyclic compounds and JAK inhibitors Download PDF

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Publication number
AU2012295802B2
AU2012295802B2 AU2012295802A AU2012295802A AU2012295802B2 AU 2012295802 B2 AU2012295802 B2 AU 2012295802B2 AU 2012295802 A AU2012295802 A AU 2012295802A AU 2012295802 A AU2012295802 A AU 2012295802A AU 2012295802 B2 AU2012295802 B2 AU 2012295802B2
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Australia
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group
groups
aromatic heterocyclyl
membered
substituted
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AU2012295802A1 (en
Inventor
Keishi Hayashi
Junji Kamon
Masataka Minami
Mariko Nasu
Koji Toyama
Miyuki UNI
Tsuneo Watanabe
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Nissan Chemical Corp
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Nissan Chemical Corp
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/5365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
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    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
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    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

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AU2012295802A 2011-08-12 2012-08-10 Tricyclic heterocyclic compounds and JAK inhibitors Ceased AU2012295802B2 (en)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
JP2011-177289 2011-08-12
JP2011-177270 2011-08-12
JP2011177289 2011-08-12
JP2011177270 2011-08-12
JP2012097073 2012-04-20
JP2012-097073 2012-04-20
JP2012103516 2012-04-27
JP2012-103517 2012-04-27
JP2012-103516 2012-04-27
JP2012103517 2012-04-27
PCT/JP2012/070876 WO2013024895A1 (en) 2011-08-12 2012-08-10 Tricyclic heterocyclic compounds and jak inhibitors

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AU2012295802A1 AU2012295802A1 (en) 2014-02-27
AU2012295802B2 true AU2012295802B2 (en) 2017-03-30

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AU2012295802A Ceased AU2012295802B2 (en) 2011-08-12 2012-08-10 Tricyclic heterocyclic compounds and JAK inhibitors

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US (2) US9216999B2 (cg-RX-API-DMAC10.html)
EP (2) EP2742049A1 (cg-RX-API-DMAC10.html)
JP (2) JP6123804B2 (cg-RX-API-DMAC10.html)
KR (1) KR102021159B1 (cg-RX-API-DMAC10.html)
CN (2) CN105001226B (cg-RX-API-DMAC10.html)
AU (1) AU2012295802B2 (cg-RX-API-DMAC10.html)
BR (1) BR112014002472A2 (cg-RX-API-DMAC10.html)
CA (1) CA2841458C (cg-RX-API-DMAC10.html)
IL (2) IL230812A0 (cg-RX-API-DMAC10.html)
IN (1) IN2014MN00228A (cg-RX-API-DMAC10.html)
MX (1) MX365311B (cg-RX-API-DMAC10.html)
MY (2) MY176647A (cg-RX-API-DMAC10.html)
PH (1) PH12013502670A1 (cg-RX-API-DMAC10.html)
RU (1) RU2632870C2 (cg-RX-API-DMAC10.html)
TW (1) TWI601727B (cg-RX-API-DMAC10.html)
UA (1) UA114606C2 (cg-RX-API-DMAC10.html)
WO (1) WO2013024895A1 (cg-RX-API-DMAC10.html)

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