AU2010272920B2 - Aminopyridine derivatives for treating tumors and inflammatory diseases - Google Patents

Aminopyridine derivatives for treating tumors and inflammatory diseases Download PDF

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Publication number
AU2010272920B2
AU2010272920B2 AU2010272920A AU2010272920A AU2010272920B2 AU 2010272920 B2 AU2010272920 B2 AU 2010272920B2 AU 2010272920 A AU2010272920 A AU 2010272920A AU 2010272920 A AU2010272920 A AU 2010272920A AU 2010272920 B2 AU2010272920 B2 AU 2010272920B2
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Prior art keywords
pyridin
pyrazol
benzimidazol
methyl
amino
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Ceased
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AU2010272920A
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AU2010272920A1 (en
Inventor
Michel Calderini
Christina Esdar
Ulrich Graedler
Margarita Wucherer-Plietker
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Merck Patent GmbH
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Merck Patent GmbH
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  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Immunology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
AU2010272920A 2009-07-15 2010-06-17 Aminopyridine derivatives for treating tumors and inflammatory diseases Ceased AU2010272920B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102009033208A DE102009033208A1 (de) 2009-07-15 2009-07-15 Aminopyridinderivate
DE102009033208.1 2009-07-15
PCT/EP2010/003659 WO2011006567A1 (de) 2009-07-15 2010-06-17 Aminopyridinderivate zur behandlung von tumoren und entzündungskrankheiten

Publications (2)

Publication Number Publication Date
AU2010272920A1 AU2010272920A1 (en) 2012-03-08
AU2010272920B2 true AU2010272920B2 (en) 2016-05-05

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AU2010272920A Ceased AU2010272920B2 (en) 2009-07-15 2010-06-17 Aminopyridine derivatives for treating tumors and inflammatory diseases

Country Status (11)

Country Link
US (1) US8648201B2 (enExample)
EP (1) EP2454253B1 (enExample)
JP (1) JP5681182B2 (enExample)
CN (1) CN102471317B (enExample)
AR (1) AR077567A1 (enExample)
AU (1) AU2010272920B2 (enExample)
CA (1) CA2768169C (enExample)
DE (1) DE102009033208A1 (enExample)
ES (1) ES2534095T3 (enExample)
IL (1) IL217467A (enExample)
WO (1) WO2011006567A1 (enExample)

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CA2955919A1 (en) 2014-07-25 2016-01-28 Piramal Enterprises Limited Substituted phenyl alkanoic acid compounds as gpr120 agonists and uses thereof
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TWI842978B (zh) 2018-07-13 2024-05-21 美商基利科學股份有限公司 衍生物
CN112457308B (zh) * 2019-09-09 2024-01-02 上海长森药业有限公司 新型三环芳香杂环化合物，及其制备方法、药物组合物和应用
US11767321B2 (en) 2020-10-05 2023-09-26 Enliven Inc. 5- and 6-azaindole compounds for inhibition of BCR-ABL tyrosine kinases
JP2025507902A (ja) * 2022-03-02 2025-03-21 杭州百誠医薬科技股▲ふん▼有限公司 ヒスタミンｈ３受容体阻害剤及びその医薬における使用

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EP2454253B1 (de) 2015-01-21
WO2011006567A1 (de) 2011-01-20
IL217467A0 (en) 2012-03-01
CA2768169A1 (en) 2011-01-20
JP5681182B2 (ja) 2015-03-04
IL217467A (en) 2015-09-24
DE102009033208A1 (de) 2011-01-20
EP2454253A1 (de) 2012-05-23
AU2010272920A1 (en) 2012-03-08
CA2768169C (en) 2017-06-13
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US8648201B2 (en) 2014-02-11
JP2012532899A (ja) 2012-12-20
AR077567A1 (es) 2011-09-07

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