AU2006233502B2 - Beta-2 adrenoceptor agonists for treating connective tissue diseases of the skin - Google Patents

Beta-2 adrenoceptor agonists for treating connective tissue diseases of the skin Download PDF

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Publication number
AU2006233502B2
AU2006233502B2 AU2006233502A AU2006233502A AU2006233502B2 AU 2006233502 B2 AU2006233502 B2 AU 2006233502B2 AU 2006233502 A AU2006233502 A AU 2006233502A AU 2006233502 A AU2006233502 A AU 2006233502A AU 2006233502 B2 AU2006233502 B2 AU 2006233502B2
Authority
AU
Australia
Prior art keywords
beta
agonist
composition
skin
lupus erythematosus
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2006233502A
Other languages
English (en)
Other versions
AU2006233502A1 (en
Inventor
Morten Sloth Weidner
Hans Christian Wulff
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astion Pharma AS
Original Assignee
Astion Pharma AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astion Pharma AS filed Critical Astion Pharma AS
Publication of AU2006233502A1 publication Critical patent/AU2006233502A1/en
Application granted granted Critical
Publication of AU2006233502B2 publication Critical patent/AU2006233502B2/en
Assigned to Cipher Pharmaceuticals, Inc. reassignment Cipher Pharmaceuticals, Inc. Request for Assignment Assignors: ASTION PHARMA A/S
Assigned to ASTION PHARMA A/S reassignment ASTION PHARMA A/S Request for Assignment Assignors: Cipher Pharmaceuticals, Inc.
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Transplantation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU2006233502A 2005-04-13 2006-04-12 Beta-2 adrenoceptor agonists for treating connective tissue diseases of the skin Ceased AU2006233502B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200500529 2005-04-13
DKPA200500529 2005-04-13
PCT/DK2006/050013 WO2006108424A2 (en) 2005-04-13 2006-04-12 Beta-2 adrenoceptor agonists for treating connective tissue diseases of the skin

Publications (2)

Publication Number Publication Date
AU2006233502A1 AU2006233502A1 (en) 2006-10-19
AU2006233502B2 true AU2006233502B2 (en) 2011-07-28

Family

ID=36703472

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2006233502A Ceased AU2006233502B2 (en) 2005-04-13 2006-04-12 Beta-2 adrenoceptor agonists for treating connective tissue diseases of the skin

Country Status (28)

Country Link
US (4) US8426475B2 (enExample)
EP (1) EP1719507B1 (enExample)
JP (1) JP5021621B2 (enExample)
KR (1) KR101355422B1 (enExample)
CN (1) CN101203214B (enExample)
AR (1) AR054249A1 (enExample)
AT (1) ATE473735T1 (enExample)
AU (1) AU2006233502B2 (enExample)
BR (1) BRPI0609361A2 (enExample)
CA (1) CA2604758C (enExample)
CY (1) CY1111541T1 (enExample)
DE (1) DE602006015387D1 (enExample)
DK (1) DK1719507T3 (enExample)
EA (1) EA016082B1 (enExample)
ES (1) ES2348920T3 (enExample)
HR (1) HRP20100552T1 (enExample)
IL (1) IL186491A (enExample)
MX (1) MX2007012794A (enExample)
MY (1) MY147864A (enExample)
NO (1) NO331211B1 (enExample)
NZ (1) NZ562940A (enExample)
PL (1) PL1719507T3 (enExample)
PT (1) PT1719507E (enExample)
RS (1) RS51464B (enExample)
SI (1) SI1719507T1 (enExample)
TW (1) TWI366457B (enExample)
WO (1) WO2006108424A2 (enExample)
ZA (1) ZA200708748B (enExample)

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GB0604826D0 (en) * 2006-03-09 2006-04-19 Arakis Ltd The treatment of inflammatory disorders and pain
CA2656312C (en) 2006-07-10 2014-09-09 Intervet International B.V. Zilpaterol enantiomer compositions and methods of making and using such compositions
GB0624757D0 (en) * 2006-12-12 2007-01-17 Sosei R & D Ltd Novel compounds
GB0805535D0 (en) * 2008-03-27 2008-04-30 Univ Leicester Scar prevention
US20120252831A1 (en) * 2011-03-31 2012-10-04 Mustafa Nevzat Ilac Sanayii A.S. Compositions of opioid antagonists and methods for treating scleroderma therewith
CN102267917B (zh) * 2011-06-15 2013-07-31 浙江工业大学 一种盐酸甲氧那明的合成方法
EP2849577A1 (en) * 2012-05-18 2015-03-25 Intervet International B.V. A method of enhancing performance in broiler chickens
GB2513297A (en) 2013-03-08 2014-10-29 Univ Leicester Methods
CN104606177B (zh) * 2014-11-21 2018-02-02 苏州君宁新药开发中心有限公司 左旋(r)沙丁胺醇制剂在治疗皮肤及粘膜创伤溃疡的药物应用
WO2018000098A1 (en) * 2016-06-30 2018-01-04 Cipher Pharmaceuticals Inc. Treatment of inflammatory myopathies
CN106580978A (zh) * 2016-11-30 2017-04-26 郑州仁宏医药科技有限公司 一种治疗皮炎的西药组合物及其应用
US10576043B2 (en) * 2017-08-10 2020-03-03 Avro Life Sciences, Inc. Transdermal drug delivery system
GB201714745D0 (en) * 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714734D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201903832D0 (en) 2019-03-20 2019-05-01 Atrogi Ab New compounds and methods
BR112021018481A2 (pt) * 2019-03-27 2021-11-23 Curasen Therapeutics Inc Agonista adrenérgico beta e métodos para usar o mesmo
CA3161376A1 (en) 2019-12-18 2021-06-24 Anthony P. FORD Methods for improving neurological diseases and disorders
CN112300237A (zh) * 2020-04-13 2021-02-02 苏州恩泰新材料科技有限公司 海豹胆酸的制备方法及其应用
KR20230084242A (ko) * 2020-10-09 2023-06-12 엠씨2 테라퓨틱스 리미티드 피부과적 병태의 치료
CN116236467B (zh) * 2023-02-07 2023-10-27 中国人民解放军总医院 西马特罗或其衍生物的新用途

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US5919827A (en) * 1990-07-11 1999-07-06 Sepracor Inc. Method for treating asthma using optically pure R(-) salmeterol
US6068833A (en) * 1991-04-05 2000-05-30 Sepracor Inc. Methods and compositions for treating pulmonary disorders using optically pure (R,R) formoterol
US6110974A (en) * 1997-04-30 2000-08-29 Bridge Pharma, Inc. Methods of accelerating muscle growth and improving feed efficiency in animals by using optically pure eutomers of adrenergic beta-2 receptor agonists, and food supplements containing the same
US6254882B1 (en) * 1997-09-16 2001-07-03 Sepracor Inc. Methods and compositions for treating pulmonary disorders using optically pure (S)—salmeterol
WO2003092617A2 (en) * 2002-05-03 2003-11-13 Combinatorx, Incorporated Combinations for the treatment of inflammatory skin disorders
WO2003097073A1 (en) * 2002-04-19 2003-11-27 Astion Development A/S Combination of a beta-2 adrenoceptor agonists and an aminosugars and their use for the treatment immunomodulatory disorders
WO2004073614A2 (en) * 2003-02-14 2004-09-02 Combinatorx, Incorporated Combination therapy for the treatment of immunoinflammatory disorders
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US5919827A (en) * 1990-07-11 1999-07-06 Sepracor Inc. Method for treating asthma using optically pure R(-) salmeterol
GB2255503A (en) * 1991-04-05 1992-11-11 Sandoz Ltd Bronchodilator enantiomers
US6068833A (en) * 1991-04-05 2000-05-30 Sepracor Inc. Methods and compositions for treating pulmonary disorders using optically pure (R,R) formoterol
US6110974A (en) * 1997-04-30 2000-08-29 Bridge Pharma, Inc. Methods of accelerating muscle growth and improving feed efficiency in animals by using optically pure eutomers of adrenergic beta-2 receptor agonists, and food supplements containing the same
US6254882B1 (en) * 1997-09-16 2001-07-03 Sepracor Inc. Methods and compositions for treating pulmonary disorders using optically pure (S)—salmeterol
WO2003097073A1 (en) * 2002-04-19 2003-11-27 Astion Development A/S Combination of a beta-2 adrenoceptor agonists and an aminosugars and their use for the treatment immunomodulatory disorders
WO2003092617A2 (en) * 2002-05-03 2003-11-13 Combinatorx, Incorporated Combinations for the treatment of inflammatory skin disorders
WO2004073614A2 (en) * 2003-02-14 2004-09-02 Combinatorx, Incorporated Combination therapy for the treatment of immunoinflammatory disorders
AU2004292445A1 (en) * 2003-11-21 2005-06-09 Zalicus Inc. Methods and reagents for the treatment of inflammatory disorders

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Also Published As

Publication number Publication date
US20170157068A1 (en) 2017-06-08
PL1719507T3 (pl) 2010-12-31
IL186491A0 (en) 2008-08-07
MY147864A (en) 2013-01-31
KR101355422B1 (ko) 2014-02-06
ZA200708748B (en) 2010-03-31
TW200719882A (en) 2007-06-01
WO2006108424A2 (en) 2006-10-19
CA2604758A1 (en) 2006-10-19
CN101203214B (zh) 2012-11-21
JP5021621B2 (ja) 2012-09-12
CN101203214A (zh) 2008-06-18
CA2604758C (en) 2014-11-25
DK1719507T3 (da) 2010-11-01
SI1719507T1 (sl) 2010-11-30
AU2006233502A1 (en) 2006-10-19
JP2008535873A (ja) 2008-09-04
NZ562940A (en) 2010-02-26
HK1091739A1 (en) 2007-01-26
PT1719507E (pt) 2010-10-21
EA200702204A1 (ru) 2008-04-28
HRP20100552T1 (hr) 2010-11-30
EP1719507A1 (en) 2006-11-08
RS51464B (sr) 2011-04-30
ATE473735T1 (de) 2010-07-15
KR20080005957A (ko) 2008-01-15
TWI366457B (en) 2012-06-21
CY1111541T1 (el) 2015-08-05
US20060235048A1 (en) 2006-10-19
WO2006108424A9 (en) 2007-08-09
US8426475B2 (en) 2013-04-23
EP1719507B1 (en) 2010-07-14
US20130237607A1 (en) 2013-09-12
AR054249A1 (es) 2007-06-13
US9907765B2 (en) 2018-03-06
IL186491A (en) 2011-12-29
MX2007012794A (es) 2008-02-22
NO20075527L (no) 2008-01-14
NO331211B1 (no) 2011-10-31
US20190125699A1 (en) 2019-05-02
BRPI0609361A2 (pt) 2010-03-30
DE602006015387D1 (de) 2010-08-26
WO2006108424A3 (en) 2006-12-14
EA016082B1 (ru) 2012-02-28
ES2348920T3 (es) 2010-12-17

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Legal Events

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FGA Letters patent sealed or granted (standard patent)
PC Assignment registered

Owner name: CIPHER PHARMACEUTICALS, INC.

Free format text: FORMER OWNER WAS: ASTION PHARMA A/S

PC Assignment registered

Owner name: ASTION PHARMA A/S

Free format text: FORMER OWNER(S): CIPHER PHARMACEUTICALS, INC.

MK14 Patent ceased section 143(a) (annual fees not paid) or expired