AU2006225355B2 - Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications - Google Patents

Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications Download PDF

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Publication number
AU2006225355B2
AU2006225355B2 AU2006225355A AU2006225355A AU2006225355B2 AU 2006225355 B2 AU2006225355 B2 AU 2006225355B2 AU 2006225355 A AU2006225355 A AU 2006225355A AU 2006225355 A AU2006225355 A AU 2006225355A AU 2006225355 B2 AU2006225355 B2 AU 2006225355B2
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hydroxy
group
acrylamide
compound
cancer
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AU2006225355A1 (en
Inventor
Ken Chi Lik Lee
Eric T. Sun
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Helsinn Healthcare SA
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Helsinn Healthcare SA
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
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    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
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  • Rheumatology (AREA)
  • Biotechnology (AREA)
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AU2006225355A 2005-03-21 2006-03-20 Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications Ceased AU2006225355B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US66326505P 2005-03-21 2005-03-21
US60/663,265 2005-03-21
US75954406P 2006-01-18 2006-01-18
US60/759,544 2006-01-18
PCT/SG2006/000064 WO2006101455A1 (en) 2005-03-21 2006-03-20 Imidazo[1,2-a]pyridine derivatives: preparation and pharmaceutical applications

Publications (2)

Publication Number Publication Date
AU2006225355A1 AU2006225355A1 (en) 2006-09-28
AU2006225355B2 true AU2006225355B2 (en) 2010-12-09

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AU2006225355A Ceased AU2006225355B2 (en) 2005-03-21 2006-03-20 Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications

Country Status (12)

Country Link
EP (1) EP1863811B1 (cg-RX-API-DMAC10.html)
JP (1) JP5206405B2 (cg-RX-API-DMAC10.html)
KR (1) KR101300831B1 (cg-RX-API-DMAC10.html)
CN (1) CN101218238B (cg-RX-API-DMAC10.html)
AR (1) AR056187A1 (cg-RX-API-DMAC10.html)
AU (1) AU2006225355B2 (cg-RX-API-DMAC10.html)
CA (1) CA2602328C (cg-RX-API-DMAC10.html)
ES (1) ES2470766T3 (cg-RX-API-DMAC10.html)
MX (1) MX2007011710A (cg-RX-API-DMAC10.html)
MY (1) MY147647A (cg-RX-API-DMAC10.html)
TW (1) TW200714600A (cg-RX-API-DMAC10.html)
WO (1) WO2006101455A1 (cg-RX-API-DMAC10.html)

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WO2010032195A1 (en) * 2008-09-16 2010-03-25 Csir Imidazopyridines and imidazopyrimidines as hiv-i reverse transcriptase inhibitors
US20110212943A1 (en) * 2008-10-15 2011-09-01 Orchid Research Laboratories Limited Novel bridged cyclic compounds as histone deacetylase inhibitors
CA2807230A1 (en) * 2010-08-03 2012-02-09 The Regents Of The University Of California Compounds and compositions for mitigating tissue damage and lethality
KR20140048079A (ko) 2011-02-01 2014-04-23 교와 핫꼬 기린 가부시키가이샤 축환 복소환 유도체
JP2014509616A (ja) * 2011-03-31 2014-04-21 エーエムベーエルエーエム テクノロジー トランスファー ゲーエムベーハー 治療用イミダゾ［１，２−ａ］ピリジン化合物
US8883819B2 (en) 2011-09-01 2014-11-11 Irm Llc Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
CN104619707A (zh) * 2012-07-31 2015-05-13 协和发酵麒麟株式会社 稠环杂环化合物
US9073921B2 (en) 2013-03-01 2015-07-07 Novartis Ag Salt forms of bicyclic heterocyclic derivatives
CN105164126B (zh) * 2013-04-30 2017-05-31 豪夫迈·罗氏有限公司 吡唑酰胺的Pd‑催化偶联
WO2014187922A1 (en) * 2013-05-24 2014-11-27 Iomet Pharma Ltd. Slc2a transporter inhibitors
CA2913785C (en) * 2013-06-25 2021-08-31 F. Hoffmann-La Roche Ag Compounds for treating spinal muscular atrophy
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US10723705B2 (en) 2015-08-14 2020-07-28 Incyte Corporation Heterocyclic compounds and uses thereof
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JP5206405B2 (ja) 2013-06-12
KR20080005207A (ko) 2008-01-10
CA2602328A1 (en) 2006-09-28
CA2602328C (en) 2014-07-29
MY147647A (en) 2012-12-31
EP1863811B1 (en) 2014-03-12
EP1863811A4 (en) 2008-11-12
TW200714600A (en) 2007-04-16
ES2470766T3 (es) 2014-06-24
KR101300831B1 (ko) 2013-08-30
JP2008533198A (ja) 2008-08-21
EP1863811A1 (en) 2007-12-12
MX2007011710A (es) 2007-11-20
CN101218238A (zh) 2008-07-09
AR056187A1 (es) 2007-09-26
CN101218238B (zh) 2011-10-26
WO2006101455A1 (en) 2006-09-28
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