AU2005326659A1 - Multicyclic bis-amide MMP inhibitors - Google Patents

Multicyclic bis-amide MMP inhibitors Download PDF

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Publication number
AU2005326659A1
AU2005326659A1 AU2005326659A AU2005326659A AU2005326659A1 AU 2005326659 A1 AU2005326659 A1 AU 2005326659A1 AU 2005326659 A AU2005326659 A AU 2005326659A AU 2005326659 A AU2005326659 A AU 2005326659A AU 2005326659 A1 AU2005326659 A1 AU 2005326659A1
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AU
Australia
Prior art keywords
alkyl
group
optionally substituted
cycloalkyl
aryl
Prior art date
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Abandoned
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AU2005326659A
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English (en)
Inventor
Ralf Biesinger
Harald Bluhm
Hongbo Deng
Rory Dodd
Brian M. Gallagher Jr.
Christian Gege
Matthias Hochgurtel
Andrew Kiely
Timothy Powers
Frank Richter
Mathias Schneider
Christoph Steeneck
Irving Sucholeiki
Arthur G. Taveras
Joshua Van Veldhuizen
Xinyuan Wu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Alantos Pharmaceuticals Holding Inc
Original Assignee
Alantos Pharmaceuticals Inc
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Filing date
Publication date
Application filed by Alantos Pharmaceuticals Inc filed Critical Alantos Pharmaceuticals Inc
Publication of AU2005326659A1 publication Critical patent/AU2005326659A1/en
Abandoned legal-status Critical Current

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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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AU2005326659A 2004-12-31 2005-12-31 Multicyclic bis-amide MMP inhibitors Abandoned AU2005326659A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US64079504P 2004-12-31 2004-12-31
US60/640,795 2004-12-31
US70626705P 2005-08-08 2005-08-08
US60/706,267 2005-08-08
PCT/US2005/047421 WO2006083454A1 (en) 2004-12-31 2005-12-31 Multicyclic bis-amide mmp inhibitors

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AU2005326659A1 true AU2005326659A1 (en) 2006-08-10

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AU2005326659A Abandoned AU2005326659A1 (en) 2004-12-31 2005-12-31 Multicyclic bis-amide MMP inhibitors

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US (1) US20060173183A1 (enExample)
EP (1) EP1843820A1 (enExample)
JP (1) JP2008526761A (enExample)
AU (1) AU2005326659A1 (enExample)
CA (1) CA2589328A1 (enExample)
MX (1) MX2007007895A (enExample)
WO (1) WO2006083454A1 (enExample)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006251989B2 (en) * 2005-05-20 2010-05-27 Alantos-Pharmaceuticals, Inc. Pyrimidine or triazine fused bicyclic metalloprotease inhibitors
US20070155738A1 (en) 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
US20070155737A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
WO2007079199A2 (en) * 2005-12-30 2007-07-12 Alantos Pharmaceuticals, Holding, Inc. Substituted bis-amide metalloprotease inhibitors
EP2069313A2 (en) * 2006-06-29 2009-06-17 Alantos Pharmaceuticals Holdings, Inc. Metalloprotease inhibitors
ATE528306T1 (de) * 2006-11-02 2011-10-15 Piramal Life Sciences Ltd Benzoxazepin-verbindungen, ihre herstellung und verwendung
US20080221092A1 (en) * 2006-11-20 2008-09-11 Harald Bluhm Heterobicyclic metalloprotease inhibitors
CA2670083A1 (en) * 2006-11-20 2008-05-29 Alantos Pharmaceuticals Holding, Inc. Heterobicyclic metalloprotease inhibitors
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