AU2004283056A1 - Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds - Google Patents
Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds Download PDFInfo
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- AU2004283056A1 AU2004283056A1 AU2004283056A AU2004283056A AU2004283056A1 AU 2004283056 A1 AU2004283056 A1 AU 2004283056A1 AU 2004283056 A AU2004283056 A AU 2004283056A AU 2004283056 A AU2004283056 A AU 2004283056A AU 2004283056 A1 AU2004283056 A1 AU 2004283056A1
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP03103961 | 2003-10-24 | ||
EP03103961.3 | 2003-10-24 | ||
EP03103967.0 | 2003-10-27 | ||
EP03103967 | 2003-10-27 | ||
PCT/EP2004/052639 WO2005039550A2 (fr) | 2003-10-24 | 2004-10-22 | Nouvelles utilisations medicales de composes a activite antagoniste de cb1 et traitement combine impliquant ces composes |
Publications (1)
Publication Number | Publication Date |
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AU2004283056A1 true AU2004283056A1 (en) | 2005-05-06 |
Family
ID=34524748
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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AU2004283056A Abandoned AU2004283056A1 (en) | 2003-10-24 | 2004-10-22 | Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1753413A2 (fr) |
JP (1) | JP2007513872A (fr) |
AU (1) | AU2004283056A1 (fr) |
BR (1) | BRPI0415851A (fr) |
CA (1) | CA2543338A1 (fr) |
MX (1) | MXPA06004434A (fr) |
RU (1) | RU2006117627A (fr) |
WO (1) | WO2005039550A2 (fr) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2004058145A2 (fr) | 2002-12-19 | 2004-07-15 | Merck & Co., Inc. | Amides substitues |
AR046132A1 (es) * | 2003-10-24 | 2005-11-23 | Solvay Pharm Gmbh | Composicin farmaceutica que contiene al menos un compuesto con actividad de receptor de cb1, o un profarmaco , tautomero o sal del mismo, como componente activo adecuado para el tratamiento y/o profilaxis de enfermedades relacionadas con el receptor cb1 en pacientes juveniles y/o para el tratamiento |
MX2007003327A (es) | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Derivados heterociclicos, y su uso como mediadores de estearoil-coa desaturasa. |
JP5149009B2 (ja) | 2004-09-20 | 2013-02-20 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | ヒトステアロイル−CoAデサチュラーゼを阻害するためのピリダジン誘導体 |
BRPI0515483A (pt) | 2004-09-20 | 2008-07-22 | Xenon Pharmaceuticals Inc | derivados heterocìclicos para o tratamento de doenças mediadas por enzimas estearoil-coa desaturase |
EP1804799B1 (fr) | 2004-09-20 | 2013-08-21 | Xenon Pharmaceuticals Inc. | Dérivés hétérocycliques et leur utilisation en tant qu'agents thérapeutiques |
JP5043668B2 (ja) | 2004-09-20 | 2012-10-10 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | 複素環誘導体および治療薬としてのそれらの使用 |
TW200626154A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
MX2007003332A (es) | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como inhibidores de estearoil-coa-desaturasa. |
MX2007015216A (es) | 2005-06-03 | 2008-02-22 | Xenon Pharmaceuticals Inc | Derivados de aminotiazol y sus usos como agentes terapeuticos. |
EP1921073A1 (fr) | 2006-11-10 | 2008-05-14 | Laboratorios del Dr. Esteve S.A. | 1,2,4-Triazoles en tant qu'inhibiteurs du récepteur sigma |
WO2024154047A1 (fr) * | 2023-01-18 | 2024-07-25 | Brien Holden Vision Institute Limited | Compositions et/ou procédés pour la prévention et/ou le traitement de troubles oculaires secs |
Family Cites Families (16)
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JP3003148B2 (ja) * | 1989-01-05 | 2000-01-24 | 藤沢薬品工業株式会社 | チアゾール化合物、その製造法およびそれを含有する医薬組成物 |
CA2195847A1 (fr) * | 1994-07-27 | 1996-02-08 | John J. Talley | Thiazoles substitues destines au traitement de l'inflammation |
US5616601A (en) * | 1994-07-28 | 1997-04-01 | Gd Searle & Co | 1,2-aryl and heteroaryl substituted imidazolyl compounds for the treatment of inflammation |
US6492516B1 (en) * | 1999-05-14 | 2002-12-10 | Merck & Co., Inc. | Compounds having cytokine inhibitory activity |
EP1373216B1 (fr) * | 2001-03-22 | 2004-12-15 | Solvay Pharmaceuticals B.V. | Derives de 4,5-dihydro-1h-pyrazole ayant une activite d'antagoniste de cb 1 |
HUP0402113A3 (en) * | 2001-09-21 | 2012-05-29 | Solvay Pharm Bv | 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity, preparation and use thereof |
SI1429761T1 (sl) * | 2001-09-21 | 2007-02-28 | Solvay Pharm Bv | Novi 4,5-dihidro-1h-pirazolni derivati s cb1-antagonisticno aktivnostjo |
TWI231757B (en) * | 2001-09-21 | 2005-05-01 | Solvay Pharm Bv | 1H-Imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity |
PE20030547A1 (es) * | 2001-09-24 | 2003-08-18 | Bayer Corp | Derivados de imidazol para el tratamiento de la obesidad |
US20050004134A1 (en) * | 2001-11-08 | 2005-01-06 | Hideo Tsutsumi | Thiazole derivative and pharmaceutical use thereof |
TW200407110A (en) * | 2001-11-23 | 2004-05-16 | Astrazeneca Ab | New use for the treatment of gastroesophageal reflux disease |
US20040248956A1 (en) * | 2002-01-29 | 2004-12-09 | Hagmann William K | Substituted imidazoles as cannabinoid receptor modulators |
AR038966A1 (es) * | 2002-03-18 | 2005-02-02 | Solvay Pharm Bv | Derivados de tiazol que tienen actividad antagonista, agonista o agonista parcial de cb1 |
TW200412942A (en) * | 2002-08-06 | 2004-08-01 | Abbott Lab | Appetite control method |
US7319110B2 (en) * | 2002-09-19 | 2008-01-15 | Solvay Pharmaceuticals B.V. | 1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity |
GB0230087D0 (en) * | 2002-12-24 | 2003-01-29 | Astrazeneca Ab | Therapeutic agents |
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2004
- 2004-10-22 WO PCT/EP2004/052639 patent/WO2005039550A2/fr active Application Filing
- 2004-10-22 JP JP2006536096A patent/JP2007513872A/ja not_active Withdrawn
- 2004-10-22 RU RU2006117627/04A patent/RU2006117627A/ru not_active Application Discontinuation
- 2004-10-22 AU AU2004283056A patent/AU2004283056A1/en not_active Abandoned
- 2004-10-22 EP EP04817279A patent/EP1753413A2/fr not_active Withdrawn
- 2004-10-22 CA CA002543338A patent/CA2543338A1/fr not_active Abandoned
- 2004-10-22 MX MXPA06004434A patent/MXPA06004434A/es not_active Application Discontinuation
- 2004-10-22 BR BRPI0415851-2A patent/BRPI0415851A/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
BRPI0415851A (pt) | 2007-01-02 |
MXPA06004434A (es) | 2006-06-20 |
EP1753413A2 (fr) | 2007-02-21 |
JP2007513872A (ja) | 2007-05-31 |
CA2543338A1 (fr) | 2005-05-06 |
WO2005039550A2 (fr) | 2005-05-06 |
RU2006117627A (ru) | 2007-12-10 |
WO2005039550A3 (fr) | 2007-03-22 |
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