AU2004283056A1 - Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds - Google Patents

Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds Download PDF

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Publication number
AU2004283056A1
AU2004283056A1 AU2004283056A AU2004283056A AU2004283056A1 AU 2004283056 A1 AU2004283056 A1 AU 2004283056A1 AU 2004283056 A AU2004283056 A AU 2004283056A AU 2004283056 A AU2004283056 A AU 2004283056A AU 2004283056 A1 AU2004283056 A1 AU 2004283056A1
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Australia
Prior art keywords
group
alkyl
substituted
compound
treatment
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Abandoned
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AU2004283056A
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English (en)
Inventor
Jochen Antel
Peter-Colin Gregory
Gunter Krause
Chris Kruse
Josephus Hubertus Maria Lange
Harald Waldeck
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Abbott Products GmbH
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Solvay Pharmaceuticals GmbH
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Publication of AU2004283056A1 publication Critical patent/AU2004283056A1/en
Abandoned legal-status Critical Current

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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Veterinary Medicine (AREA)
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  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Addiction (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
AU2004283056A 2003-10-24 2004-10-22 Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds Abandoned AU2004283056A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP03103961 2003-10-24
EP03103961.3 2003-10-24
EP03103967.0 2003-10-27
EP03103967 2003-10-27
PCT/EP2004/052639 WO2005039550A2 (fr) 2003-10-24 2004-10-22 Nouvelles utilisations medicales de composes a activite antagoniste de cb1 et traitement combine impliquant ces composes

Publications (1)

Publication Number Publication Date
AU2004283056A1 true AU2004283056A1 (en) 2005-05-06

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Application Number Title Priority Date Filing Date
AU2004283056A Abandoned AU2004283056A1 (en) 2003-10-24 2004-10-22 Novel medical uses of compounds showing CB1-antagonistic activity and combination treatment involving said compounds

Country Status (8)

Country Link
EP (1) EP1753413A2 (fr)
JP (1) JP2007513872A (fr)
AU (1) AU2004283056A1 (fr)
BR (1) BRPI0415851A (fr)
CA (1) CA2543338A1 (fr)
MX (1) MXPA06004434A (fr)
RU (1) RU2006117627A (fr)
WO (1) WO2005039550A2 (fr)

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WO2004058145A2 (fr) 2002-12-19 2004-07-15 Merck & Co., Inc. Amides substitues
AR046132A1 (es) * 2003-10-24 2005-11-23 Solvay Pharm Gmbh Composicin farmaceutica que contiene al menos un compuesto con actividad de receptor de cb1, o un profarmaco , tautomero o sal del mismo, como componente activo adecuado para el tratamiento y/o profilaxis de enfermedades relacionadas con el receptor cb1 en pacientes juveniles y/o para el tratamiento
MX2007003327A (es) 2004-09-20 2007-06-05 Xenon Pharmaceuticals Inc Derivados heterociclicos, y su uso como mediadores de estearoil-coa desaturasa.
JP5149009B2 (ja) 2004-09-20 2013-02-20 ゼノン・ファーマシューティカルズ・インコーポレイテッド ヒトステアロイル−CoAデサチュラーゼを阻害するためのピリダジン誘導体
BRPI0515483A (pt) 2004-09-20 2008-07-22 Xenon Pharmaceuticals Inc derivados heterocìclicos para o tratamento de doenças mediadas por enzimas estearoil-coa desaturase
EP1804799B1 (fr) 2004-09-20 2013-08-21 Xenon Pharmaceuticals Inc. Dérivés hétérocycliques et leur utilisation en tant qu'agents thérapeutiques
JP5043668B2 (ja) 2004-09-20 2012-10-10 ゼノン・ファーマシューティカルズ・インコーポレイテッド 複素環誘導体および治療薬としてのそれらの使用
TW200626154A (en) 2004-09-20 2006-08-01 Xenon Pharmaceuticals Inc Heterocyclic derivatives and their use as therapeutic agents
MX2007003332A (es) 2004-09-20 2007-06-05 Xenon Pharmaceuticals Inc Derivados heterociclicos y su uso como inhibidores de estearoil-coa-desaturasa.
MX2007015216A (es) 2005-06-03 2008-02-22 Xenon Pharmaceuticals Inc Derivados de aminotiazol y sus usos como agentes terapeuticos.
EP1921073A1 (fr) 2006-11-10 2008-05-14 Laboratorios del Dr. Esteve S.A. 1,2,4-Triazoles en tant qu'inhibiteurs du récepteur sigma
WO2024154047A1 (fr) * 2023-01-18 2024-07-25 Brien Holden Vision Institute Limited Compositions et/ou procédés pour la prévention et/ou le traitement de troubles oculaires secs

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JP3003148B2 (ja) * 1989-01-05 2000-01-24 藤沢薬品工業株式会社 チアゾール化合物、その製造法およびそれを含有する医薬組成物
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BRPI0415851A (pt) 2007-01-02
MXPA06004434A (es) 2006-06-20
EP1753413A2 (fr) 2007-02-21
JP2007513872A (ja) 2007-05-31
CA2543338A1 (fr) 2005-05-06
WO2005039550A2 (fr) 2005-05-06
RU2006117627A (ru) 2007-12-10
WO2005039550A3 (fr) 2007-03-22

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