AU2003265901B2 - Pyrazolopyrimidines as cyclin dependent kinase inhibitors - Google Patents

Pyrazolopyrimidines as cyclin dependent kinase inhibitors Download PDF

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Publication number
AU2003265901B2
AU2003265901B2 AU2003265901A AU2003265901A AU2003265901B2 AU 2003265901 B2 AU2003265901 B2 AU 2003265901B2 AU 2003265901 A AU2003265901 A AU 2003265901A AU 2003265901 A AU2003265901 A AU 2003265901A AU 2003265901 B2 AU2003265901 B2 AU 2003265901B2
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Prior art keywords
compound
aryl
alkyl
group
cycloalkyl
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AU2003265901A1 (en
Inventor
Lawrence W. Dillard
Ronald J. Doll
Michael P. Dwyer
Viyyoor Moopil Girijavallabhan
Timothy J. Guzi
Zhen Min He
Ray Anthony James
Chad Knutson
Brian Mckittrick
Haengsoon Park
Kamil Paruch
Vinh D. Tran
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Merck Sharp and Dohme LLC
Pharmacopeia LLC
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Pharmacopeia Inc
Schering Corp
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Assigned to PHARMACOPEIA, INC., SCHERING CORPORATION reassignment PHARMACOPEIA, INC. Request for Assignment Assignors: PHARMACOPEIA DRUG DISCOVERY, INC., SCHERING CORPORATION
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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AU2003265901A 2002-09-04 2003-09-03 Pyrazolopyrimidines as cyclin dependent kinase inhibitors Ceased AU2003265901B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40818202P 2002-09-04 2002-09-04
US60/408,182 2002-09-04
PCT/US2003/027564 WO2004022062A1 (en) 2002-09-04 2003-09-03 Pyrazolopyrimidines as cyclin dependent kinase inhibitors

Publications (2)

Publication Number Publication Date
AU2003265901A1 AU2003265901A1 (en) 2004-03-29
AU2003265901B2 true AU2003265901B2 (en) 2006-09-14

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AU2003265901A Ceased AU2003265901B2 (en) 2002-09-04 2003-09-03 Pyrazolopyrimidines as cyclin dependent kinase inhibitors

Country Status (14)

Country Link
US (2) US7084271B2 (https=)
EP (1) EP1545533A1 (https=)
JP (2) JP2006500391A (https=)
KR (1) KR20050057072A (https=)
CN (1) CN1694705A (https=)
AR (1) AR041135A1 (https=)
AU (1) AU2003265901B2 (https=)
CA (1) CA2497539A1 (https=)
MX (1) MXPA05002574A (https=)
NZ (1) NZ539163A (https=)
PE (1) PE20040998A1 (https=)
TW (1) TW200412966A (https=)
WO (1) WO2004022062A1 (https=)
ZA (1) ZA200501854B (https=)

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US10953012B2 (en) 2011-04-26 2021-03-23 Bioenergenix Llc Heterocyclic compounds for the inhibition of pask
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US10392389B2 (en) 2012-10-25 2019-08-27 Bioenergenix Llc Heterocyclic compounds for the inhibition of PASK
KR20150130491A (ko) 2013-03-13 2015-11-23 제넨테크, 인크. 피라졸로 화합물 및 그것의 용도
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US7468372B2 (en) 2008-12-23
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US20060173017A1 (en) 2006-08-03
PE20040998A1 (es) 2004-12-30
NZ539163A (en) 2007-03-30
EP1545533A1 (en) 2005-06-29
US20040102452A1 (en) 2004-05-27
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CN1694705A (zh) 2005-11-09
US7084271B2 (en) 2006-08-01
JP2011074088A (ja) 2011-04-14
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