AU2003232215B2 - Thiazole derivatives as phosphodiesterase IV inhibitors - Google Patents

Thiazole derivatives as phosphodiesterase IV inhibitors Download PDF

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Publication number
AU2003232215B2
AU2003232215B2 AU2003232215A AU2003232215A AU2003232215B2 AU 2003232215 B2 AU2003232215 B2 AU 2003232215B2 AU 2003232215 A AU2003232215 A AU 2003232215A AU 2003232215 A AU2003232215 A AU 2003232215A AU 2003232215 B2 AU2003232215 B2 AU 2003232215B2
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disease
asthma
chronic
group
pathogenesis
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AU2003232215A1 (en
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Hans-Michael Eggenweiler
Michael Wolf
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Merck Patent GmbH
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Merck Patent GmbH
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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biotechnology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
AU2003232215A 2002-06-19 2003-04-28 Thiazole derivatives as phosphodiesterase IV inhibitors Ceased AU2003232215B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10227269A DE10227269A1 (de) 2002-06-19 2002-06-19 Thiazolderivate
DE10227269.7 2002-06-19
PCT/EP2003/004434 WO2004000839A1 (de) 2002-06-19 2003-04-28 Thiazolderivate als phosphodiesterase iv-inhibtoren

Publications (2)

Publication Number Publication Date
AU2003232215A1 AU2003232215A1 (en) 2004-01-06
AU2003232215B2 true AU2003232215B2 (en) 2009-04-30

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ID=29719229

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003232215A Ceased AU2003232215B2 (en) 2002-06-19 2003-04-28 Thiazole derivatives as phosphodiesterase IV inhibitors

Country Status (15)

Country Link
US (1) US7790723B2 (enExample)
EP (1) EP1513837B1 (enExample)
JP (1) JP4555076B2 (enExample)
AR (1) AR039695A1 (enExample)
AT (1) ATE338041T1 (enExample)
AU (1) AU2003232215B2 (enExample)
BR (1) BR0311879A (enExample)
CA (1) CA2489902C (enExample)
DE (2) DE10227269A1 (enExample)
ES (1) ES2271642T3 (enExample)
MX (1) MXPA04012428A (enExample)
PL (1) PL372123A1 (enExample)
RU (1) RU2005101202A (enExample)
WO (1) WO2004000839A1 (enExample)
ZA (1) ZA200500484B (enExample)

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DE10227269A1 (de) * 2002-06-19 2004-01-08 Merck Patent Gmbh Thiazolderivate
AR044519A1 (es) 2003-05-02 2005-09-14 Novartis Ag Derivados de piridin-tiazol amina y de pirimidin-tiazol amina
GB0401334D0 (en) 2004-01-21 2004-02-25 Novartis Ag Organic compounds
AU2005247906B2 (en) 2004-05-18 2011-08-25 Merck Sharp & Dohme Corp. Substituted 2-quinolyl-oxazoles useful as PDE4 inhibitors
GB0411056D0 (en) 2004-05-18 2004-06-23 Novartis Ag Organic compounds
GT200500281A (es) 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
GB0424284D0 (en) 2004-11-02 2004-12-01 Novartis Ag Organic compounds
GB0426164D0 (en) 2004-11-29 2004-12-29 Novartis Ag Organic compounds
GB0507577D0 (en) 2005-04-14 2005-05-18 Novartis Ag Organic compounds
GB0510390D0 (en) 2005-05-20 2005-06-29 Novartis Ag Organic compounds
US7910708B2 (en) 2005-10-21 2011-03-22 Novartis Ag Anti-IL13 human antibodies
GB0526244D0 (en) 2005-12-22 2006-02-01 Novartis Ag Organic compounds
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
ATE549337T1 (de) 2006-04-21 2012-03-15 Novartis Ag Purinderivate zur verwendung als adenosin-a2a- rezeptoragonisten
KR20090073121A (ko) 2006-09-29 2009-07-02 노파르티스 아게 Ｐｉ3ｋ 지질 키나제 억제제로서의 피라졸로피리미딘
KR20090075714A (ko) 2006-10-30 2009-07-08 노파르티스 아게 소염제로서의 헤테로시클릭 화합물
RS51644B (sr) 2007-01-10 2011-10-31 Irm Llc. Jedinjenja i preparati kao inhibitori kanal aktivirajuće proteaze
KR20100005730A (ko) 2007-05-07 2010-01-15 노파르티스 아게 유기 화합물
EA017919B1 (ru) 2007-12-10 2013-04-30 Новартис Аг Производные пиразин-2-карбоксамида для лечения заболеваний, которые поддаются лечению путем блокирования эпителиальных натриевых каналов
EP2231642B1 (en) 2008-01-11 2013-10-23 Novartis AG Pyrimidines as kinase inhibitors
KR20110040818A (ko) 2008-06-10 2011-04-20 노파르티스 아게 상피 나트륨 채널 차단제로서의 피라진 유도체
WO2010009243A1 (en) 2008-07-15 2010-01-21 Theracos, Inc. Deuterated benzylbenzene derivatives and methods of use
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US20050222160A1 (en) 2005-10-06
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