ATE73460T1 - Peptide aus alpha-aminoboronsaeuren. - Google Patents

Peptide aus alpha-aminoboronsaeuren.

Info

Publication number
ATE73460T1
ATE73460T1 AT84308405T AT84308405T ATE73460T1 AT E73460 T1 ATE73460 T1 AT E73460T1 AT 84308405 T AT84308405 T AT 84308405T AT 84308405 T AT84308405 T AT 84308405T AT E73460 T1 ATE73460 T1 AT E73460T1
Authority
AT
Austria
Prior art keywords
alpha
aminoboronic acid
acid peptides
peptides
aminoboronic
Prior art date
Application number
AT84308405T
Other languages
English (en)
Inventor
Ashokkumar Bhikkappa Shenvi
Charles A Kettner
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Application granted granted Critical
Publication of ATE73460T1 publication Critical patent/ATE73460T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0827Tripeptides containing heteroatoms different from O, S, or N
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT84308405T 1983-12-05 1984-12-04 Peptide aus alpha-aminoboronsaeuren. ATE73460T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/558,362 US4499082A (en) 1983-12-05 1983-12-05 α-Aminoboronic acid peptides
EP84308405A EP0145441B1 (de) 1983-12-05 1984-12-04 Peptide aus alpha-Aminoboronsäuren

Publications (1)

Publication Number Publication Date
ATE73460T1 true ATE73460T1 (de) 1992-03-15

Family

ID=24229258

Family Applications (1)

Application Number Title Priority Date Filing Date
AT84308405T ATE73460T1 (de) 1983-12-05 1984-12-04 Peptide aus alpha-aminoboronsaeuren.

Country Status (7)

Country Link
US (1) US4499082A (de)
EP (1) EP0145441B1 (de)
JP (2) JPH0717675B2 (de)
AT (1) ATE73460T1 (de)
CA (1) CA1253999A (de)
DE (1) DE3485568D1 (de)
HK (1) HK116893A (de)

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DE3840452A1 (de) * 1988-12-01 1990-06-07 Hoechst Ag (beta)-amino-boronsaeure-derivate
US5252463A (en) * 1990-06-22 1993-10-12 The Du Pont Merck Pharmaceutical Company Clipsin, a chymotrypsin-like protease and method of using same
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Also Published As

Publication number Publication date
JPH07173170A (ja) 1995-07-11
EP0145441A2 (de) 1985-06-19
EP0145441B1 (de) 1992-03-11
JPH0717675B2 (ja) 1995-03-01
JP2540290B2 (ja) 1996-10-02
EP0145441A3 (en) 1987-04-29
JPS60146900A (ja) 1985-08-02
US4499082A (en) 1985-02-12
CA1253999A (en) 1989-05-09
HK116893A (en) 1993-11-05
DE3485568D1 (de) 1992-04-16

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