ATE546450T1 - Microkristall of (e)-8-(3,4-dimethoxystyryl)-1,3- diethyl-7-methyl-3,7-dihydro-1h-purine-2,6-dion - Google Patents
Microkristall of (e)-8-(3,4-dimethoxystyryl)-1,3- diethyl-7-methyl-3,7-dihydro-1h-purine-2,6-dionInfo
- Publication number
- ATE546450T1 ATE546450T1 AT04731752T AT04731752T ATE546450T1 AT E546450 T1 ATE546450 T1 AT E546450T1 AT 04731752 T AT04731752 T AT 04731752T AT 04731752 T AT04731752 T AT 04731752T AT E546450 T1 ATE546450 T1 AT E546450T1
- Authority
- AT
- Austria
- Prior art keywords
- dimethoxystyryl
- dione
- purine
- dihydro
- diethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2003131417 | 2003-05-09 | ||
PCT/JP2004/006495 WO2004099207A1 (ja) | 2003-05-09 | 2004-05-07 | 微細結晶 |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE546450T1 true ATE546450T1 (de) | 2012-03-15 |
Family
ID=33432132
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT04731752T ATE546450T1 (de) | 2003-05-09 | 2004-05-07 | Microkristall of (e)-8-(3,4-dimethoxystyryl)-1,3- diethyl-7-methyl-3,7-dihydro-1h-purine-2,6-dion |
Country Status (10)
Country | Link |
---|---|
US (1) | US7541363B2 (de) |
EP (1) | EP1626049B1 (de) |
JP (2) | JP4606326B2 (de) |
KR (2) | KR20110128216A (de) |
CN (1) | CN100395245C (de) |
AT (1) | ATE546450T1 (de) |
AU (1) | AU2004236101B2 (de) |
CA (1) | CA2525037C (de) |
ES (1) | ES2384685T3 (de) |
WO (1) | WO2004099207A1 (de) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7247639B2 (en) * | 2003-06-06 | 2007-07-24 | Endacea, Inc. | A1 adenosine receptor antagonists |
TW200507882A (en) * | 2003-07-17 | 2005-03-01 | Kyowa Hakko Kogyo Kk | Solid formulations |
JP7382737B2 (ja) * | 2019-05-13 | 2023-11-17 | 東和薬品株式会社 | イストラデフィリン製剤 |
CN113024558A (zh) * | 2021-03-15 | 2021-06-25 | 山东新华制药股份有限公司 | 伊曲茶碱的晶体的制备方法和应用 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0059091A1 (de) * | 1981-02-25 | 1982-09-01 | Leslie Stott | Einrichtung zum Regeln der Ausflussmenge |
US5484920A (en) | 1992-04-08 | 1996-01-16 | Kyowa Hakko Kogyo Co., Ltd. | Therapeutic agent for Parkinson's disease |
JP2928386B2 (ja) * | 1992-07-08 | 1999-08-03 | 協和醗酵工業株式会社 | うつ病治療剤 |
JP2613355B2 (ja) * | 1992-09-28 | 1997-05-28 | 協和醗酵工業株式会社 | パーキンソン氏病治療剤 |
ATE240734T1 (de) * | 1995-07-26 | 2003-06-15 | Kyowa Hakko Kogyo Kk | Zubereitung von xanthinderivaten als feste dispersion |
JPH0940652A (ja) * | 1995-07-28 | 1997-02-10 | Kyowa Hakko Kogyo Co Ltd | ウラシル誘導体の製造方法 |
TW200507882A (en) * | 2003-07-17 | 2005-03-01 | Kyowa Hakko Kogyo Kk | Solid formulations |
-
2004
- 2004-05-07 EP EP04731752A patent/EP1626049B1/de not_active Expired - Lifetime
- 2004-05-07 CA CA2525037A patent/CA2525037C/en not_active Expired - Fee Related
- 2004-05-07 WO PCT/JP2004/006495 patent/WO2004099207A1/ja active Application Filing
- 2004-05-07 CN CNB2004800118737A patent/CN100395245C/zh not_active Expired - Fee Related
- 2004-05-07 JP JP2005506044A patent/JP4606326B2/ja not_active Expired - Lifetime
- 2004-05-07 AU AU2004236101A patent/AU2004236101B2/en not_active Ceased
- 2004-05-07 AT AT04731752T patent/ATE546450T1/de active
- 2004-05-07 US US10/554,511 patent/US7541363B2/en active Active
- 2004-05-07 ES ES04731752T patent/ES2384685T3/es not_active Expired - Lifetime
- 2004-05-07 KR KR1020117026513A patent/KR20110128216A/ko not_active Application Discontinuation
- 2004-05-07 KR KR1020057020738A patent/KR101229594B1/ko active IP Right Grant
-
2010
- 2010-06-17 JP JP2010138014A patent/JP2010195836A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
EP1626049A4 (de) | 2008-07-02 |
AU2004236101A1 (en) | 2004-11-18 |
JP2010195836A (ja) | 2010-09-09 |
KR20110128216A (ko) | 2011-11-28 |
KR101229594B1 (ko) | 2013-02-05 |
EP1626049A1 (de) | 2006-02-15 |
US7541363B2 (en) | 2009-06-02 |
CN100395245C (zh) | 2008-06-18 |
ES2384685T3 (es) | 2012-07-11 |
CN1784405A (zh) | 2006-06-07 |
JPWO2004099207A1 (ja) | 2006-07-13 |
US20060205745A1 (en) | 2006-09-14 |
KR20060015570A (ko) | 2006-02-17 |
JP4606326B2 (ja) | 2011-01-05 |
CA2525037C (en) | 2011-12-20 |
CA2525037A1 (en) | 2004-11-18 |
EP1626049B1 (de) | 2012-02-22 |
WO2004099207A1 (ja) | 2004-11-18 |
AU2004236101B2 (en) | 2010-11-11 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CA2398887A1 (en) | 2,4,di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineoplastic agents | |
DE502004007000D1 (de) | Stickstoff substituierte hexahydro-pyrazino 1,2-a pyrimidin-4,7-dionderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel | |
WO2001049688A8 (en) | Purine derivatives, process for their preparation and use thereof | |
WO2004018451A8 (en) | Pyridazinone-derivatives as pde4 inhibitors | |
WO2003041647A3 (en) | Synthesis and purification of valacyclovir | |
ZA200506253B (en) | Pyrimidine derivatives for the prevention of HIV infection | |
PL1613304T3 (pl) | Inhibitory DPP-IV | |
WO2003093269A3 (de) | Substituierte pyrazolo-pyrimidin-4-one | |
MY133479A (en) | Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions | |
ATE500254T1 (de) | Die replikation von hiv hemmende purinderivate | |
AU2002357773A1 (en) | 1,6 naphthyridines useful as inhibitors of syk kinase | |
WO2003050087A3 (en) | Novel herbicides | |
WO2005063744A3 (en) | IMIDAZO[4,5-c]PYRIDINE COMPOUNDS AND METHODS OF ANTIVIRAL TREATMENT | |
CY1105553T1 (el) | Υποκαταστατα 2-πυριμιδινυλιο-6,7,8,9-τετραϋδροπυριμιδο[1,2-α]πυριμιδιν-4-ονιο και 7-πυριμιδινυλιο-2,3-διυδροιμιδαζο[1,2-α]πυριμιδιν-5(1η)ονιο για νευροεκφυλιστικες διαταραχες | |
WO2006031281A3 (en) | Orientation-insensitive ultra-wideband coupling capacitor and method of making | |
JP2007510401A5 (de) | ||
HK1064096A1 (en) | Purine derivatives as a2b adenosine receptor antagonists. | |
CA2166800A1 (en) | 4-substituted piperidine derivatives useful as neurokinin antagonists | |
ATE472548T1 (de) | Substituierte hexahydro-pyrazino(1,2-a)pyrimidin- 4,7-dionderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel | |
WO2001084962A3 (de) | Zusammensetzungen enthaltend folsäure und reduziertes folat | |
WO2003022216A3 (en) | Biaryl substituted purine derivatives as potent antiproliferative agents | |
CA2419665A1 (en) | Novel 2-phenylpiperazine derivatives | |
ATE546450T1 (de) | Microkristall of (e)-8-(3,4-dimethoxystyryl)-1,3- diethyl-7-methyl-3,7-dihydro-1h-purine-2,6-dion | |
WO2002094020A8 (de) | Verwendung von triazolopyrimidin-derivaten als mikrobizide im materialschutz | |
EP1647275A4 (de) | Feste pharmazeutische zubereitung |