ATE537136T1 - Neues verfahren zur herstellung von säurechloriden - Google Patents

Neues verfahren zur herstellung von säurechloriden

Info

Publication number
ATE537136T1
ATE537136T1 AT06807399T AT06807399T ATE537136T1 AT E537136 T1 ATE537136 T1 AT E537136T1 AT 06807399 T AT06807399 T AT 06807399T AT 06807399 T AT06807399 T AT 06807399T AT E537136 T1 ATE537136 T1 AT E537136T1
Authority
AT
Austria
Prior art keywords
new process
acid chlorides
producing acid
preparation
producing
Prior art date
Application number
AT06807399T
Other languages
English (en)
Inventor
Ursula Hoffmann
Goesta Rimmler
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of ATE537136T1 publication Critical patent/ATE537136T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/58Preparation of carboxylic acid halides
    • C07C51/60Preparation of carboxylic acid halides by conversion of carboxylic acids or their anhydrides or esters, lactones, salts into halides with the same carboxylic acid part
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/38Acyl halides
    • C07C53/44Acyl halides containing rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT06807399T 2005-10-31 2006-10-19 Neues verfahren zur herstellung von säurechloriden ATE537136T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05110177 2005-10-31
PCT/EP2006/067570 WO2007051714A1 (en) 2005-10-31 2006-10-19 Novel process for the preparation of acid chlorides

Publications (1)

Publication Number Publication Date
ATE537136T1 true ATE537136T1 (de) 2011-12-15

Family

ID=37663247

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06807399T ATE537136T1 (de) 2005-10-31 2006-10-19 Neues verfahren zur herstellung von säurechloriden

Country Status (13)

Country Link
US (2) US7435849B2 (de)
EP (1) EP1945601B1 (de)
JP (1) JP5148500B2 (de)
KR (1) KR100980522B1 (de)
CN (1) CN101300219B (de)
AT (1) ATE537136T1 (de)
AU (1) AU2006310591B2 (de)
BR (1) BRPI0618267B1 (de)
CA (1) CA2626102C (de)
ES (1) ES2377570T3 (de)
IL (1) IL190551A (de)
TW (1) TWI313677B (de)
WO (1) WO2007051714A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7435849B2 (en) * 2005-10-31 2008-10-14 Hoffmann-La Roche Inc. Process for the production of acid chlorides
CA2684067A1 (en) * 2007-04-25 2008-11-06 F. Hoffmann-La Roche Ag Novel process for the preparation of acid chlorides
EP2274278B1 (de) * 2008-04-04 2016-08-17 F. Hoffmann-La Roche AG Neues verfahren zur herstellung von cyclohexancarboxylsäure-derivaten
KR101290935B1 (ko) * 2008-04-04 2013-07-29 에프. 호프만-라 로슈 아게 상응하는 사이클로헥세인카복스아마이드 유도체에 의한 사이클로헥세인카복실산 유도체의 신규한 제조 방법
AU2009259495B2 (en) 2008-06-17 2014-04-03 F. Hoffmann-La Roche Ag 1-(2-ethyl-butyl) -cyclohexanecarboxylic acid ester as an intermediate in the preparation of pharmaceutically active amides
US20110004011A1 (en) 2009-07-01 2011-01-06 Declan Costello Novel process
CN103097345A (zh) 2010-09-16 2013-05-08 霍夫曼-拉罗奇有限公司 新方法
EP2635263B1 (de) 2010-11-04 2015-09-23 F.Hoffmann-La Roche Ag Zusammensetzung umfassend s-[2-([[1-(2-ethylbutyl)-cyclohexyl]-carbonyl]amino)phenyl]2-methylpropanethioate und croscarmellose natrium
CA2818018C (en) 2010-12-08 2016-02-02 F. Hoffmann-La Roche Ag Liposomal formulation of dalcetrapib
EP2651882B1 (de) 2010-12-16 2018-11-14 F.Hoffmann-La Roche Ag Verfahren zur herstellung von aromatischen thiolderivaten durch hydrogenierung von disulfiden
JP2014505714A (ja) 2011-02-17 2014-03-06 エフ.ホフマン−ラ ロシュ アーゲー ホットメルト押出法による過冷却液体状態からの活性医薬成分の制御された結晶化方法
US8975438B2 (en) 2011-07-13 2015-03-10 Hoffmann-La Roche Inc. Process for the preparation of cyclohexanecarboxylic acid derivatives
KR20150016280A (ko) 2012-04-30 2015-02-11 에프. 호프만-라 로슈 아게 신규 제형
PT2978859T (pt) 2013-03-27 2018-10-04 Hoffmann La Roche Marcadores genéticos para previsão da capacidade de resposta à terapêutica
EP3082784A1 (de) 2013-12-19 2016-10-26 F.Hoffmann-La Roche Ag Cetp-modulator zur verwendung in der behandlung einer augenkrankheit
CN103755759A (zh) * 2014-01-26 2014-04-30 江西科技师范大学 一种合成核苷磷酰哌啶、磷酰吗啉及磷酰吡咯烷的方法
ES2825675T3 (es) 2014-07-30 2021-05-17 Hoffmann La Roche Marcadores genéticos para predecir la reactividad al tratamiento con un agente que aumenta las HDL o que imita las HDL
KR102807066B1 (ko) * 2019-09-30 2025-05-15 주식회사 엘지화학 아민계 화합물 제조방법
WO2025093129A1 (en) 2023-11-01 2025-05-08 Newamsterdam Pharma B.V. Treatment and prevention of age-related macular degeneration using a cetp inhibitor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2899458A (en) 1959-08-11 Process for producing oxy aromatic
US4129595A (en) * 1978-03-29 1978-12-12 Chevron Research Company Preparation of chloroacetyl chloride
JPS5740432A (en) * 1980-08-25 1982-03-06 Mitsubishi Chem Ind Ltd Production of carboxylic acid chloride
JP3290962B2 (ja) * 1997-02-12 2002-06-10 日本たばこ産業株式会社 Cetp活性阻害剤
JP2894445B2 (ja) 1997-02-12 1999-05-24 日本たばこ産業株式会社 Cetp活性阻害剤として有効な化合物
JP2002069033A (ja) * 2000-06-16 2002-03-08 Japan Tobacco Inc 1−置換−シクロヘキサンカルボニルハライド化合物の製造方法
GB0229803D0 (en) 2002-12-20 2003-01-29 Syngenta Ltd Chemical process
GB0304132D0 (en) * 2003-02-24 2003-03-26 Syngenta Ltd Chemical process
US7435849B2 (en) * 2005-10-31 2008-10-14 Hoffmann-La Roche Inc. Process for the production of acid chlorides

Also Published As

Publication number Publication date
CA2626102C (en) 2014-01-07
US20090036703A1 (en) 2009-02-05
IL190551A (en) 2012-08-30
US20070100154A1 (en) 2007-05-03
TWI313677B (en) 2009-08-21
KR20080061385A (ko) 2008-07-02
TW200720246A (en) 2007-06-01
BRPI0618267A2 (pt) 2011-08-23
IL190551A0 (en) 2008-11-03
JP5148500B2 (ja) 2013-02-20
US7728171B2 (en) 2010-06-01
JP2009513686A (ja) 2009-04-02
ES2377570T3 (es) 2012-03-29
AU2006310591A1 (en) 2007-05-10
US7435849B2 (en) 2008-10-14
KR100980522B1 (ko) 2010-09-06
CA2626102A1 (en) 2007-05-10
CN101300219A (zh) 2008-11-05
WO2007051714A1 (en) 2007-05-10
BRPI0618267B1 (pt) 2016-06-21
EP1945601A1 (de) 2008-07-23
EP1945601B1 (de) 2011-12-14
AU2006310591B2 (en) 2012-03-15
CN101300219B (zh) 2012-08-08

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