ATE536101T1 - Behandlung heilmittelresistenter proliferativer erkrankungen - Google Patents
Behandlung heilmittelresistenter proliferativer erkrankungenInfo
- Publication number
- ATE536101T1 ATE536101T1 AT06717284T AT06717284T ATE536101T1 AT E536101 T1 ATE536101 T1 AT E536101T1 AT 06717284 T AT06717284 T AT 06717284T AT 06717284 T AT06717284 T AT 06717284T AT E536101 T1 ATE536101 T1 AT E536101T1
- Authority
- AT
- Austria
- Prior art keywords
- treatment
- drug
- proliferative diseases
- resistant
- resistant proliferative
- Prior art date
Links
- 230000002062 proliferating effect Effects 0.000 title abstract 2
- 201000010099 disease Diseases 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
- 229940043355 kinase inhibitor Drugs 0.000 abstract 1
- 239000003757 phosphotransferase inhibitor Substances 0.000 abstract 1
- 229940124530 sulfonamide Drugs 0.000 abstract 1
- 150000003456 sulfonamides Chemical class 0.000 abstract 1
- 150000003457 sulfones Chemical class 0.000 abstract 1
- 150000003462 sulfoxides Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64137805P | 2005-01-05 | 2005-01-05 | |
| PCT/US2006/000059 WO2006074149A2 (en) | 2005-01-05 | 2006-01-04 | Treatment of drug-resistant proliferative disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE536101T1 true ATE536101T1 (de) | 2011-12-15 |
Family
ID=36648100
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT06717284T ATE536101T1 (de) | 2005-01-05 | 2006-01-04 | Behandlung heilmittelresistenter proliferativer erkrankungen |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20090306207A1 (de) |
| EP (1) | EP1841420B1 (de) |
| JP (1) | JP5156389B2 (de) |
| KR (2) | KR101427105B1 (de) |
| AT (1) | ATE536101T1 (de) |
| AU (1) | AU2006204103B2 (de) |
| CA (1) | CA2593523C (de) |
| IL (1) | IL184292A (de) |
| WO (1) | WO2006074149A2 (de) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090197893A1 (en) * | 2005-12-01 | 2009-08-06 | Bristol-Myers Squibb Company | Methods of Identifying and Treating Individuals Exhibiting Complex Karyotypes |
| KR101707669B1 (ko) * | 2008-04-17 | 2017-02-16 | 더 존스 홉킨스 유니버시티 | 약제-내성 종양에서 화학요법제 활성을 증강시키는 on01910.na |
| JP6348904B2 (ja) | 2012-09-20 | 2018-06-27 | テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイションTemple University−Of The Commonwealth System Of Higher Education | 置換アルキルジアリール誘導体、その製造方法及び使用 |
| US10383831B2 (en) | 2015-08-03 | 2019-08-20 | Temple University—Of the Commonwealth System of Higher Education | 2,4,6-trialkoxystryl aryl sulfones, sulfonamides and carboxamides, and methods of preparation and use |
| CN111926086B (zh) * | 2020-08-21 | 2022-05-31 | 云南农业大学 | 一种影响鸡体斜长的分子标记及其应用 |
| GB2628229A (en) * | 2021-08-12 | 2024-09-18 | Onconova Therapeutics Inc | Methods and compositions for treating cancer |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2210601C2 (ru) * | 1996-07-25 | 2003-08-20 | Ипкор Н.В. | Способ восстановления и плавления металла |
| BR9814059B1 (pt) * | 1997-10-03 | 2010-08-24 | composto e composiÇço farmacÉutica. | |
| US6548553B2 (en) * | 1997-10-03 | 2003-04-15 | Temple University-Of The Commonwealth System Of Higher Education | Styryl sulfone anticancer agents |
| EP1173160B1 (de) * | 1999-04-02 | 2005-06-22 | Temple University of the Commonwealth System of Higher Education | (e)-styrylsulfone als krebsbestreitende mittel |
| US6762207B1 (en) * | 1999-04-02 | 2004-07-13 | Temple University - Of The Commonwealth System Of Higher Education | (E)-styryl sulfone anticancer agents |
| US6767926B1 (en) * | 1999-10-12 | 2004-07-27 | Temple University - Of The Commonwealth System Of Higher Education | Method for protecting normal cells from cytotoxicity of chemotherapeutic agents |
| US6243322B1 (en) * | 1999-11-05 | 2001-06-05 | Wavemakers Research, Inc. | Method for estimating the distance of an acoustic signal |
| US6541475B2 (en) * | 2000-04-14 | 2003-04-01 | Temple University - Of The Commonwealth System Of Higher Education | α, β-unsaturated sulfones for treating proliferative disorders |
| US6486210B2 (en) * | 2000-04-14 | 2002-11-26 | Temple University—Of the Commonwealth System of Higher Education | Substituted styryl benzylsulfones for treating proliferative disorders |
| ATE406881T1 (de) * | 2001-02-28 | 2008-09-15 | Univ Temple | Verwendung von alpha, beta ungesättigten arylsulfonen zum schutz von zellen und geweben vor toxizität ionischer strahlung |
| JP4538233B2 (ja) * | 2002-02-28 | 2010-09-08 | テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション | 増殖性障害治療用の、アミノ置換されたスルホンアニリド及びその誘導体 |
| KR100972131B1 (ko) * | 2002-02-28 | 2010-07-26 | 템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션 | 증식성 질병 치료용 아미노-치환(e)-2,6-디알콕시스티릴 4-치환-벤질설폰 |
| DK1689706T3 (da) * | 2003-11-14 | 2017-04-03 | Temple Univ - Of The Commonwealth System Of Higher Education | Alfa, beta-umættede sulfoxider til behandling af proliferative forstyrrelser |
| US7932242B2 (en) * | 2004-03-16 | 2011-04-26 | Temple University - Of The Commonwealth System Of Higher Education | Substituted phenoxy-and phenylthio-derivatives for treating proliferative disorders |
-
2006
- 2006-01-04 WO PCT/US2006/000059 patent/WO2006074149A2/en not_active Ceased
- 2006-01-04 KR KR1020137020463A patent/KR101427105B1/ko not_active Expired - Lifetime
- 2006-01-04 CA CA2593523A patent/CA2593523C/en not_active Expired - Lifetime
- 2006-01-04 EP EP06717284A patent/EP1841420B1/de not_active Expired - Lifetime
- 2006-01-04 AT AT06717284T patent/ATE536101T1/de active
- 2006-01-04 AU AU2006204103A patent/AU2006204103B2/en not_active Expired
- 2006-01-04 US US11/794,524 patent/US20090306207A1/en not_active Abandoned
- 2006-01-04 JP JP2007550417A patent/JP5156389B2/ja not_active Expired - Lifetime
- 2006-01-04 KR KR1020077018000A patent/KR20070094956A/ko not_active Ceased
-
2007
- 2007-06-28 IL IL184292A patent/IL184292A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| US20090306207A1 (en) | 2009-12-10 |
| WO2006074149A3 (en) | 2007-11-15 |
| KR20070094956A (ko) | 2007-09-27 |
| EP1841420A2 (de) | 2007-10-10 |
| EP1841420A4 (de) | 2009-12-09 |
| AU2006204103A1 (en) | 2006-07-13 |
| EP1841420B1 (de) | 2011-12-07 |
| IL184292A (en) | 2012-10-31 |
| AU2006204103B2 (en) | 2011-11-24 |
| KR101427105B1 (ko) | 2014-08-07 |
| JP2008526852A (ja) | 2008-07-24 |
| WO2006074149A2 (en) | 2006-07-13 |
| JP5156389B2 (ja) | 2013-03-06 |
| IL184292A0 (en) | 2007-10-31 |
| KR20130091796A (ko) | 2013-08-19 |
| CA2593523A1 (en) | 2006-07-13 |
| CA2593523C (en) | 2014-04-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EA202092899A1 (ru) | Гетероарильные соединения для лечения болезни гентингтона | |
| DK2150530T3 (da) | Substituerede sulfonamid-derivater | |
| EA200900983A1 (ru) | Соединения и композиции в качестве ингибиторов киназы | |
| DOP2009000141A (es) | Derivados de dihidropiridina de utilidad como inhibidores de la proteína quinasa | |
| CR10072A (es) | Derivados de pirimidinil-aril-urea que son inhibidores de fgf | |
| MX383856B (es) | Compuestos y composiciones para inhibir la actividad de shp2. | |
| DK1625126T3 (da) | Imidazo- og thiazolopyridiner som JAK3-kinaseinhibitorer | |
| NO20082026L (no) | Deazapuriner som er nyttige som inhibitorer for Janus-kinaser | |
| EA200801291A1 (ru) | Карбониламинопирролопиразолы в качестве эффективных ингибиторов киназ | |
| NO20084652L (no) | Deazapuriner anvendelige som inhibitorer av januskinaser | |
| EA201200669A1 (ru) | ПИРИДОПИРИМИДИНОНОВЫЕ ИНГИБИТОРЫ PI3Kα | |
| EA200870193A1 (ru) | Цитотоксические агенты, включающие новые производные томаймицина, и их терапевтическое применение | |
| EA200970156A1 (ru) | Пиридизиноновые производные | |
| EA200801362A1 (ru) | Пиримидинил бензотиофеновые соединения | |
| EA201100447A1 (ru) | Органические соединения | |
| EA200700851A1 (ru) | Получение и применение бифенил-4-илкарбониламинокислотных производных для лечения ожирения | |
| EA200700489A1 (ru) | Новые бензоконденсированные гетероарилсульфамидные производные, полезные в качестве противоконвульсивных средств | |
| DE60206911D1 (de) | Imidazol-2-carbonsäureamid derivate als raf-kinase-inhibitoren | |
| EA201500403A1 (ru) | Соединения, активирующие теломеразу, и способы их применения | |
| NO20092130L (no) | Tricykliske heteroarylforbindelser anvendelige som inhibitorer of januskinase | |
| MA32505B1 (fr) | 5-alcynyl-pyrimidines | |
| CO6630193A2 (es) | Inhibidores de la actividad de la proteína tirosina quinasa seleccionada | |
| EA200600605A1 (ru) | Перегруппированные пентанолы, способ их получения и их применение в качестве противовоспалительных средств | |
| ATE502935T1 (de) | C-met-proteinkinasehemmer | |
| IL184292A0 (en) | Treatment of drug-resistant proliferative disorders |