ATE495172T1 - Neue azabizyklische arylderivate und medizinische verwendung damit - Google Patents

Neue azabizyklische arylderivate und medizinische verwendung damit

Info

Publication number
ATE495172T1
ATE495172T1 AT05797020T AT05797020T ATE495172T1 AT E495172 T1 ATE495172 T1 AT E495172T1 AT 05797020 T AT05797020 T AT 05797020T AT 05797020 T AT05797020 T AT 05797020T AT E495172 T1 ATE495172 T1 AT E495172T1
Authority
AT
Austria
Prior art keywords
diseases
disorders
compounds
pyridazinyl
medical use
Prior art date
Application number
AT05797020T
Other languages
English (en)
Inventor
Dan Peters
Daniel B Timmermann
Gunnar M Olsen
Elsebet Ystergaard Nielsen
Tino Dyhring Jyrgensen
Original Assignee
Neurosearch As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurosearch As filed Critical Neurosearch As
Application granted granted Critical
Publication of ATE495172T1 publication Critical patent/ATE495172T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
AT05797020T 2004-10-15 2005-10-14 Neue azabizyklische arylderivate und medizinische verwendung damit ATE495172T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US61859804P 2004-10-15 2004-10-15
DKPA200401582 2004-10-15
PCT/EP2005/055263 WO2006040352A1 (en) 2004-10-15 2005-10-14 Novel azabicyclic aryl derivatives and their medical use

Publications (1)

Publication Number Publication Date
ATE495172T1 true ATE495172T1 (de) 2011-01-15

Family

ID=38744785

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05797020T ATE495172T1 (de) 2004-10-15 2005-10-14 Neue azabizyklische arylderivate und medizinische verwendung damit

Country Status (9)

Country Link
US (1) US7652010B2 (de)
EP (1) EP1802616B1 (de)
CN (1) CN100588657C (de)
AT (1) ATE495172T1 (de)
AU (1) AU2005293510A1 (de)
CA (1) CA2584836A1 (de)
DE (1) DE602005025902D1 (de)
HK (1) HK1106513A1 (de)
WO (1) WO2006040352A1 (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0220581D0 (en) 2002-09-04 2002-10-09 Novartis Ag Organic Compound
PE20060437A1 (es) 2004-06-18 2006-06-08 Novartis Ag COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR
GB0415746D0 (en) 2004-07-14 2004-08-18 Novartis Ag Organic compounds
GB0521508D0 (en) 2005-10-21 2005-11-30 Novartis Ag Organic compounds
GB0525672D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
GB0525673D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
WO2007093601A1 (en) 2006-02-14 2007-08-23 Neurosearch A/S 3, 9-diazabicyclo(3.3.1)non-3-yl-aryl methanone derivatives as nicotinic acetylcholine receptor agonists
ATE455114T1 (de) * 2006-02-16 2010-01-15 Neurosearch As Enantiomerenreine chinuclidinyloxy-pyridazine und ihre verwendung als nikotin-acetylcholin- rezeptorliganden
US8314119B2 (en) * 2006-11-06 2012-11-20 Abbvie Inc. Azaadamantane derivatives and methods of use
JO3250B1 (ar) 2009-09-22 2018-09-16 Novartis Ag إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7
SG2014013460A (en) 2010-09-23 2014-09-26 Abbvie Inc Monohydrate of an azaadamantane derivative
WO2016100184A1 (en) 2014-12-16 2016-06-23 Forum Pharmaceuticals, Inc. Geminal substituted quinuclidine amide compounds as agonists of alpha-7 nicotinic acetylcholine receptors
CA2988968A1 (en) 2015-06-10 2016-12-15 Forum Pharmaceuticals, Inc. Aminobenzisoxazole compounds as agonists of a7-nicotinic acetylcholine receptors
WO2017027600A1 (en) 2015-08-12 2017-02-16 Forum Pharmaceuticals, Inc. GEMINAL SUBSTITUTED AMINOBENZISOXAZOLE COMPOUNDS AS AGONISTS OF α7-NICOTINIC ACETYLCHOLINE RECEPTORS
CN109593088B (zh) * 2018-12-27 2022-03-25 华东理工大学 氮杂双环衍生物及其制备和应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2791678B1 (fr) * 1999-03-30 2001-05-04 Synthelabo Derives de 1,4-diazabicyclo [3.2.2] nonane-4-carboxylates et -carboxamides, leur preparation et leur application en therapeutique
US6492385B2 (en) * 2000-08-18 2002-12-10 Pharmacia & Upjohn Company Quinuclidine-substituted heteroaryl moieties for treatment of disease
DE50305587D1 (en) * 2002-06-10 2006-12-14 Bayer Healthcare Ag 2-heteroarylcarbonsäureamide
SE0202430D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab New Compounds
GB0415746D0 (en) 2004-07-14 2004-08-18 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
CA2584836A1 (en) 2006-04-20
CN101027300A (zh) 2007-08-29
EP1802616B1 (de) 2011-01-12
WO2006040352A1 (en) 2006-04-20
EP1802616A1 (de) 2007-07-04
US7652010B2 (en) 2010-01-26
AU2005293510A1 (en) 2006-04-20
DE602005025902D1 (de) 2011-02-24
HK1106513A1 (en) 2008-03-14
CN100588657C (zh) 2010-02-10
US20070299082A1 (en) 2007-12-27

Similar Documents

Publication Publication Date Title
ATE495172T1 (de) Neue azabizyklische arylderivate und medizinische verwendung damit
ATE493415T1 (de) Neue diazabizyklische arylderivate und medizinische verwendung dafür
ATE481407T1 (de) Neue diazabicyclische arylderivate und medizinische verwendung dafür
ATE385497T1 (de) 3-substituierte quinuclidin-derivate und deren verwendung als nikotinischen agonisten
ATE477253T1 (de) Neuartige oxadiazol-derivate und deren medizinische verwendung
ATE473978T1 (de) Neue diazabicyclische arylderivate und medizinische verwendung dafür
ATE450263T1 (de) Diazabicyclische aryl-derivate als cholinerge rezeptor-modulatoren
ATE437880T1 (de) Dimere azacyclische verbindungen und deren verwendung
DE602007004307D1 (de) Enantiomerenreine chinuclidinyloxy-pyridazine und ihre verwendung als nikotin-acetylcholin-rezeptorliganden
ATE287888T1 (de) Aryl- und heteroaryldiazabicycloalkane, deren zubereitung und verwendung
DK1506200T3 (da) Diazabicykliske biarylderivater
ATE345342T1 (de) 1,4-dizabicyclo(3,2,2)nonane derivative, verfahren zur ihre herstellung und therapeutical verwendung
HK1079528A1 (en) Azacyclic ethynyl derivatives
DE60215172D1 (de) Neue verbindungen, deren herstellung und verwendung
ATE445618T1 (de) Neue diazabicyclische arylderivate
ATE334129T1 (de) 3-substituierte chinuklidine und deren verwendung
MX2007003331A (es) Nuevos derivados de arilo diazabiciclico.
ATE460416T1 (de) Neuartige 1,4-diazabicycloä3.2.2ünonan-derivate und deren medizinische verwendung
DE602006019561D1 (de) Diazabicyclische arylderivate und ihre verwendung als chinolinergische liganden an nikotin-acetylcholin-rezeptoren
DE602004031124D1 (de) Neue chinuklidinderivative und deren pharmazeutische verwendung
ATE478869T1 (de) Diazabicycloalkan-derivate und ihre medizinische verwendung
MX2007004245A (es) Nuevos derivados de arilo azabiciclicos y su uso medico.

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties