ATE418543T1 - Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten - Google Patents

Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten

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Publication number
ATE418543T1
ATE418543T1 AT03773731T AT03773731T ATE418543T1 AT E418543 T1 ATE418543 T1 AT E418543T1 AT 03773731 T AT03773731 T AT 03773731T AT 03773731 T AT03773731 T AT 03773731T AT E418543 T1 ATE418543 T1 AT E418543T1
Authority
AT
Austria
Prior art keywords
dipiperidine
substituted
piperazine derivatives
neurokin antagonists
neurokin
Prior art date
Application number
AT03773731T
Other languages
English (en)
Inventor
Frans Eduard Janssens
Francois Maria Sommen
Boeck Benoit Christian Albert De
Joseph Elisabeth Leenaerts
Roosbroeck Yves Emiel Maria Van
Gaston Stanislas Marcella Diels
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2002/014836 external-priority patent/WO2004056772A1/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of ATE418543T1 publication Critical patent/ATE418543T1/de

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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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AT03773731T 2002-10-08 2003-10-07 Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten ATE418543T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0211328 2002-10-08
PCT/EP2002/014836 WO2004056772A1 (en) 2002-12-23 2002-12-23 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as tachykinin antagonists

Publications (1)

Publication Number Publication Date
ATE418543T1 true ATE418543T1 (de) 2009-01-15

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JP2006510602A (ja) 2006-03-30
EP1551804A1 (de) 2005-07-13
TWI324995B (en) 2010-05-21
CA2499903A1 (en) 2004-04-22
MY141736A (en) 2010-06-15
AU2003282115B2 (en) 2009-10-01
KR101049074B1 (ko) 2011-07-15
HRP20050309A2 (en) 2006-07-31
BR0315098A (pt) 2005-08-16
PA8584901A1 (es) 2005-10-28
HK1084394A1 (en) 2006-07-28
TW200413319A (en) 2004-08-01
US20060167008A1 (en) 2006-07-27
EP1551804B1 (de) 2008-12-24
EA009217B1 (ru) 2007-12-28
US7410970B2 (en) 2008-08-12
AU2003282115A1 (en) 2004-05-04
EA200500616A1 (ru) 2005-10-27
IL167885A (en) 2010-04-29
WO2004033428A1 (en) 2004-04-22
JP4674086B2 (ja) 2011-04-20
KR20050059164A (ko) 2005-06-17
DE60325493D1 (de) 2009-02-05
AR041545A1 (es) 2005-05-18
CA2499903C (en) 2011-06-14

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