ATE403657T1 - Chemische verbindungen - Google Patents

Chemische verbindungen

Info

Publication number
ATE403657T1
ATE403657T1 AT02776075T AT02776075T ATE403657T1 AT E403657 T1 ATE403657 T1 AT E403657T1 AT 02776075 T AT02776075 T AT 02776075T AT 02776075 T AT02776075 T AT 02776075T AT E403657 T1 ATE403657 T1 AT E403657T1
Authority
AT
Austria
Prior art keywords
chemical compounds
derivatives
methods
pyrazolo
diseases
Prior art date
Application number
AT02776075T
Other languages
English (en)
Inventor
Jerry Adams
Jiri Kasparec
Domingos Silva
Catherine Yuan
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Application granted granted Critical
Publication of ATE403657T1 publication Critical patent/ATE403657T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT02776075T 2001-10-02 2002-10-01 Chemische verbindungen ATE403657T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32650601P 2001-10-02 2001-10-02

Publications (1)

Publication Number Publication Date
ATE403657T1 true ATE403657T1 (de) 2008-08-15

Family

ID=23272496

Family Applications (1)

Application Number Title Priority Date Filing Date
AT02776075T ATE403657T1 (de) 2001-10-02 2002-10-01 Chemische verbindungen

Country Status (8)

Country Link
US (1) US7217710B2 (de)
EP (1) EP1432714B1 (de)
JP (1) JP4459619B2 (de)
AT (1) ATE403657T1 (de)
AU (1) AU2002341920A1 (de)
DE (1) DE60228103D1 (de)
ES (1) ES2309206T3 (de)
WO (1) WO2003029209A2 (de)

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JO3367B1 (ar) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
KR102414246B1 (ko) 2014-01-21 2022-06-27 얀센 파마슈티카 엔.브이. 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
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Also Published As

Publication number Publication date
JP4459619B2 (ja) 2010-04-28
JP2005504828A (ja) 2005-02-17
AU2002341920A1 (en) 2003-04-14
WO2003029209A2 (en) 2003-04-10
US20040198751A1 (en) 2004-10-07
DE60228103D1 (de) 2008-09-18
ES2309206T3 (es) 2008-12-16
EP1432714A2 (de) 2004-06-30
WO2003029209A3 (en) 2004-02-12
EP1432714B1 (de) 2008-08-06
US7217710B2 (en) 2007-05-15
EP1432714A4 (de) 2005-10-19

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