ATE396189T1 - Cyanopyrrolhaltige cyclische carbamat- und thiocarbamatbiaryle und verfahren zu deren herstellung - Google Patents

Cyanopyrrolhaltige cyclische carbamat- und thiocarbamatbiaryle und verfahren zu deren herstellung

Info

Publication number
ATE396189T1
ATE396189T1 AT05740218T AT05740218T ATE396189T1 AT E396189 T1 ATE396189 T1 AT E396189T1 AT 05740218 T AT05740218 T AT 05740218T AT 05740218 T AT05740218 T AT 05740218T AT E396189 T1 ATE396189 T1 AT E396189T1
Authority
AT
Austria
Prior art keywords
optionally substituted
methyl
alkyl
cyanopyrrole
aminoalkyl
Prior art date
Application number
AT05740218T
Other languages
English (en)
Inventor
Bogdan Wilk
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Application granted granted Critical
Publication of ATE396189T1 publication Critical patent/ATE396189T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT05740218T 2004-04-27 2005-04-25 Cyanopyrrolhaltige cyclische carbamat- und thiocarbamatbiaryle und verfahren zu deren herstellung ATE396189T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US56561604P 2004-04-27 2004-04-27

Publications (1)

Publication Number Publication Date
ATE396189T1 true ATE396189T1 (de) 2008-06-15

Family

ID=35242253

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05740218T ATE396189T1 (de) 2004-04-27 2005-04-25 Cyanopyrrolhaltige cyclische carbamat- und thiocarbamatbiaryle und verfahren zu deren herstellung

Country Status (14)

Country Link
US (3) US7582755B2 (de)
EP (1) EP1756095B1 (de)
JP (2) JP5108506B2 (de)
CN (1) CN1946716B (de)
AT (1) ATE396189T1 (de)
AU (1) AU2005238520B2 (de)
BR (1) BRPI0510278A (de)
CA (1) CA2562160C (de)
DE (1) DE602005007021D1 (de)
DK (1) DK1756095T3 (de)
ES (1) ES2306140T3 (de)
MX (1) MXPA06012402A (de)
PL (1) PL1756095T3 (de)
WO (1) WO2005105739A2 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA73119C2 (en) * 2000-04-19 2005-06-15 American Home Products Corpoir Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors
EP1756095B1 (de) * 2004-04-27 2008-05-21 Wyeth Cyanopyrrolhaltige cyclische carbamat- und thiocarbamatbiaryle und verfahren zu deren herstellung
MX2007013467A (es) * 2005-04-28 2008-01-21 Wyeth Corp Tanaproget micronizado y composiciones que contienen el mismo.
AU2006287925B2 (en) * 2005-04-28 2012-03-01 Wyeth Compositions containing micronized tanaproget
PT1896034E (pt) * 2005-04-28 2010-05-06 Wyeth Llc Composições de tanaproget micronizado e métodos para a sua preparação
PE20070220A1 (es) * 2005-07-29 2007-03-19 Wyeth Corp Proceso para la sintesis de moduladores del receptor de progesterona
PE20070341A1 (es) * 2005-07-29 2007-04-13 Wyeth Corp Derivados de pirrol como moduladores del receptor de progesterona
PE20070404A1 (es) 2005-07-29 2007-05-10 Wyeth Corp Compuestos derivados de cianopirrol-sulfonamida como moduladores del receptor de progesterona
PE20070182A1 (es) 2005-07-29 2007-03-06 Wyeth Corp Derivados cianopirrol-fenil amida como moduladores del receptor de progesterona
US20070213526A1 (en) * 2006-03-07 2007-09-13 Wyeth Purification of progesterone receptor modulators
US20080319204A1 (en) * 2007-06-25 2008-12-25 Wyeth Process for the synthesis of progesterone receptor modulators
EP2234491A4 (de) * 2007-12-20 2010-12-22 Teva Womens Health Inc Dosierungsschemata und pharmazeutische zusammensetzungen und packungen für die notfallkontrazeption
GB0817578D0 (en) * 2008-09-25 2008-11-05 3M Innovative Properties Co Method for treating wheel rims and composition for use therein

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US5194628A (en) * 1988-03-18 1993-03-16 Ciba-Geigy Corporation Process for the preparation of substituted difluorobenzo-1,3-dioxoles
EP0717740A1 (de) 1993-09-10 1996-06-26 Ciba SC Holding AG Photochrome verbindungen, verfahren und zwischenprodukte zu deren hestellung und deren verwendung
US6545108B1 (en) 1999-02-22 2003-04-08 Eastman Chemical Company Catalysts containing N-pyrrolyl substituted nitrogen donors
DE60014376T2 (de) 1999-02-22 2005-02-24 Eastman Chemical Co., Kingsport Katalysatoren, die n-pyrrolylsubstituierte stickstoffdonoren enthalten
DK1175411T3 (da) * 1999-05-04 2008-06-09 Wyeth Corp Cyclothiocarbamatderivater som progesteron-receptormodulatorer
CA2371651A1 (en) * 1999-05-04 2000-11-09 American Home Products Corporation Quinazolinone and benzoxazine derivatives as progesterone receptor modulators
US6407101B1 (en) * 1999-05-04 2002-06-18 American Home Products Corporation Cyanopyrroles
US6391907B1 (en) * 1999-05-04 2002-05-21 American Home Products Corporation Indoline derivatives
WO2000066560A1 (en) 1999-05-04 2000-11-09 American Home Products Corporation Quinazolinone and benzoxazine derivatives as progesterone receptor modulators
US6509334B1 (en) * 1999-05-04 2003-01-21 American Home Products Corporation Cyclocarbamate derivatives as progesterone receptor modulators
CA2371726A1 (en) * 1999-05-04 2000-11-09 American Home Products Corporation Cyclocarbamate derivatives as progesterone receptor modulators
US6566372B1 (en) * 1999-08-27 2003-05-20 Ligand Pharmaceuticals Incorporated Bicyclic androgen and progesterone receptor modulator compounds and methods
US20020065192A1 (en) * 2000-02-18 2002-05-30 Mackenzie Peter Borden Productivity catalysts and microstructure control
UA73119C2 (en) * 2000-04-19 2005-06-15 American Home Products Corpoir Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors
US6350837B1 (en) 2000-06-09 2002-02-26 Eastman Chemical Company Copolymerization of norbornene and functional norbornene monomers
EP1351997A2 (de) 2000-11-06 2003-10-15 Eastman Chemical Company Katalysatoren mit verbesserter produktivität und mikrostruktursteuerung
WO2002036642A2 (en) 2000-11-06 2002-05-10 Eastman Chemical Company Olefin polymerization processes using supported catalysts
US6387992B1 (en) * 2000-11-27 2002-05-14 Ciba Specialty Chemicals Corporation Substituted 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole UV absorbers, a process for preparation thereof and compositions stabilized therewith
AU2002218309A1 (en) 2000-11-27 2002-06-03 Ciba Specialty Chemicals Holding Inc. Substituted 5-aryl and 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole derivatives as uv absorbers
DE10111262A1 (de) 2001-03-09 2002-09-12 Studiengesellschaft Kohle Mbh Verfahren zur Herstellung von Vinyl- Aryl- und Heteroarylessigsäuren und ihrer Devivate
JP2005194190A (ja) 2001-10-05 2005-07-21 Fumie Satou １９−ノル−ビタミンｄ誘導体の製造法
DE10152989A1 (de) * 2001-10-26 2003-05-08 Bayer Ag Komplexe N-heterocyslischer Carbene und ihre Verwendung
AU2003223930A1 (en) 2002-06-14 2003-12-31 Novo Nordisk A/S Pharmaceutical use of boronic acids and esters thereof
CN1665510A (zh) * 2002-06-25 2005-09-07 惠氏公司 作为pr调节剂的环硫代氨基甲酸酯衍生物的衍生物和其用于治疗皮肤病的用途
TW200404548A (en) * 2002-06-25 2004-04-01 Wyeth Corp Pharmaceutical composition containing cyclothiocarbamate derivatives in treatment of hormone-related conditions
US7446211B2 (en) * 2004-04-27 2008-11-04 Wyeth Coupling process for generating reactive boron-containing derivatives of N-substituted pyrrole-2-carbonitriles to produce biaryls
BRPI0510260A (pt) * 2004-04-27 2007-10-23 Wyeth Corp método para purificar um composto, e, kit farmacêutico
EP1756095B1 (de) 2004-04-27 2008-05-21 Wyeth Cyanopyrrolhaltige cyclische carbamat- und thiocarbamatbiaryle und verfahren zu deren herstellung

Also Published As

Publication number Publication date
US20050239779A1 (en) 2005-10-27
CA2562160A1 (en) 2005-11-10
WO2005105739A3 (en) 2006-02-16
US8003784B2 (en) 2011-08-23
US8129524B2 (en) 2012-03-06
DE602005007021D1 (de) 2008-07-03
US20120016118A1 (en) 2012-01-19
US20090306371A1 (en) 2009-12-10
MXPA06012402A (es) 2007-01-17
EP1756095A2 (de) 2007-02-28
CN1946716A (zh) 2007-04-11
JP2013006853A (ja) 2013-01-10
EP1756095B1 (de) 2008-05-21
CN1946716B (zh) 2011-12-21
US7582755B2 (en) 2009-09-01
ES2306140T3 (es) 2008-11-01
JP2007534767A (ja) 2007-11-29
DK1756095T3 (da) 2008-08-11
WO2005105739A2 (en) 2005-11-10
AU2005238520A1 (en) 2005-11-10
CA2562160C (en) 2013-05-28
BRPI0510278A (pt) 2007-10-30
AU2005238520B2 (en) 2011-09-08
PL1756095T3 (pl) 2008-10-31
JP5108506B2 (ja) 2012-12-26

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