ATE371645T1 - Naphthalinderivate, die sich an den ep4?rezeptor binden - Google Patents

Naphthalinderivate, die sich an den ep4?rezeptor binden

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Publication number
ATE371645T1
ATE371645T1 AT01271355T AT01271355T ATE371645T1 AT E371645 T1 ATE371645 T1 AT E371645T1 AT 01271355 T AT01271355 T AT 01271355T AT 01271355 T AT01271355 T AT 01271355T AT E371645 T1 ATE371645 T1 AT E371645T1
Authority
AT
Austria
Prior art keywords
bind
receptor
naphthaline derivatives
derivatives
naphthaline
Prior art date
Application number
AT01271355T
Other languages
English (en)
Inventor
Gerard Martin Paul Giblin
Haydn Terence Jones
Andrew Mason
Neil Miller
Susan Roomans
Stephen Shanahan
Ann Walker
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE371645T1 publication Critical patent/ATE371645T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/58—[b]- or [c]-condensed
    • C07D209/62—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles
    • C07D209/64—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles with an oxygen atom in position 1
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D209/56—Ring systems containing three or more rings
    • C07D209/58—[b]- or [c]-condensed
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    • C07D209/66—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles with oxygen atoms in positions 1 and 3

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AT01271355T 2000-12-21 2001-12-20 Naphthalinderivate, die sich an den ep4?rezeptor binden ATE371645T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0031302.3A GB0031302D0 (en) 2000-12-21 2000-12-21 Napthalene derivatives

Publications (1)

Publication Number Publication Date
ATE371645T1 true ATE371645T1 (de) 2007-09-15

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ID=9905630

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01271355T ATE371645T1 (de) 2000-12-21 2001-12-20 Naphthalinderivate, die sich an den ep4?rezeptor binden

Country Status (9)

Country Link
US (1) US6924297B2 (de)
EP (1) EP1351934B1 (de)
JP (1) JP4397586B2 (de)
AT (1) ATE371645T1 (de)
AU (1) AU2002216218A1 (de)
DE (1) DE60130256T2 (de)
ES (1) ES2290093T3 (de)
GB (1) GB0031302D0 (de)
WO (1) WO2002050032A1 (de)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN2001000224A (es) 2000-10-19 2002-06-13 Pfizer Compuestos de imidazol condensado con arilo o heteroarilo como agentes anti - inflamatorios y analgesicos.
GB0031295D0 (en) * 2000-12-21 2001-01-31 Glaxo Group Ltd Naphthalene derivatives
CA2563356A1 (en) * 2004-04-20 2005-11-03 Pfizer Products Inc. Combinations comprising alpha-2-delta ligands and ep4 receptor antagonists
ATE533766T1 (de) * 2005-05-19 2011-12-15 Merck Canada Inc Chinolinderivate als ep4-antagonisten
UY30121A1 (es) 2006-02-03 2007-08-31 Glaxo Group Ltd Nuevos compuestos
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DE60130256T2 (de) 2008-05-21
JP2004517099A (ja) 2004-06-10
AU2002216218A1 (en) 2002-07-01
WO2002050032A1 (en) 2002-06-27
EP1351934B1 (de) 2007-08-29
ES2290093T3 (es) 2008-02-16
US20040102508A1 (en) 2004-05-27
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